BDBM213761 US9284299, 12::US9738628, Compound 12
SMILES: On1nnc2cc(CCc3nn[nH]n3)ccc12
InChI Key: InChIKey=ILSPBLDTHMAASO-UHFFFAOYSA-N
Data: 12 KI
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Catenin beta-1 [138-686] (Homo sapiens (Human)) | BDBM213761 (US9284299, 12 | US9738628, Compound 12) | PDB GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 3.14E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Utah Research Foundation US Patent | Assay Description Experiments were performed in white opaque 384-well plates from PerkinElmer (Waltham, Mass.), and the samples were read on a Synergy 2 plate reader (... | US Patent US9738628 (2017) BindingDB Entry DOI: 10.7270/Q27P91H7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Catenin beta-1 [138-686] (Homo sapiens (Human)) | BDBM213761 (US9284299, 12 | US9738628, Compound 12) | PDB GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 3.14E+3 | -7.50 | n/a | n/a | n/a | n/a | n/a | n/a | 25 |
University of Utah Research Foundation US Patent | Assay Description Experiments were performed in 96-well Microfluor 2 black plates (Waltham, Mass.), and the samples were read by a Synergy 2 plate reader (Biotek, Wino... | US Patent US9284299 (2016) BindingDB Entry DOI: 10.7270/Q2WW7GGC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Catenin beta-1 [138-686]/Transcription factor 4 [7-51] (Homo sapiens (Human)) | BDBM213761 (US9284299, 12 | US9738628, Compound 12) | PDB GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 3.14E+3 | -7.50 | n/a | n/a | n/a | n/a | n/a | n/a | 25 |
University of Utah Research Foundation US Patent | Assay Description Experiments were performed in 96-well Microfluor 2 black plates (Waltham, Mass.), and the samples were read by a Synergy 2 plate reader (Biotek, Wino... | US Patent US9284299 (2016) BindingDB Entry DOI: 10.7270/Q2WW7GGC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Catenin beta-1 [138-686] (Homo sapiens (Human)) | BDBM213761 (US9284299, 12 | US9738628, Compound 12) | PDB GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 3.83E+3 | -7.38 | n/a | n/a | n/a | n/a | n/a | n/a | 25 |
University of Utah Research Foundation US Patent | Assay Description Experiments were performed in 96-well Microfluor 2 black plates (Waltham, Mass.), and the samples were read by a Synergy 2 plate reader (Biotek, Wino... | US Patent US9284299 (2016) BindingDB Entry DOI: 10.7270/Q2WW7GGC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Catenin beta-1 [138-686]/Transcription factor 4 [7-51] (Homo sapiens (Human)) | BDBM213761 (US9284299, 12 | US9738628, Compound 12) | PDB GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 3.83E+3 | -7.38 | n/a | n/a | n/a | n/a | n/a | 7.4 | 25 |
University of Utah Research Foundation US Patent | Assay Description Experiments were performed in white opaque 384-well plates from PerkinElmer (Waltham, Mass.), and the samples were read on a Synergy 2 plate reader (... | US Patent US9284299 (2016) BindingDB Entry DOI: 10.7270/Q2WW7GGC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Catenin beta-1 [138-686] (Homo sapiens (Human)) | BDBM213761 (US9284299, 12 | US9738628, Compound 12) | PDB GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 7.60E+3 | -6.98 | n/a | n/a | n/a | n/a | n/a | 7.4 | 25 |
University of Utah Research Foundation US Patent | Assay Description Experiments were performed in white opaque 384-well plates from PerkinElmer (Waltham, Mass.), and the samples were read on a Synergy 2 plate reader (... | US Patent US9284299 (2016) BindingDB Entry DOI: 10.7270/Q2WW7GGC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Catenin beta-1 [138-686] (Homo sapiens (Human)) | BDBM213761 (US9284299, 12 | US9738628, Compound 12) | PDB GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 7.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Utah Research Foundation US Patent | Assay Description Experiments were performed in 96-well Microfluor 2 black plates (Waltham, Mass.), and the samples were read by a Synergy 2 plate reader (Biotek, Wino... | US Patent US9738628 (2017) BindingDB Entry DOI: 10.7270/Q27P91H7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Catenin beta-1 [138-686] (Homo sapiens (Human)) | BDBM213761 (US9284299, 12 | US9738628, Compound 12) | PDB GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 5.42E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Utah Research Foundation US Patent | Assay Description Experiments were performed in white opaque 384-well plates from PerkinElmer (Waltham, Mass.), and the samples were read on a Synergy 2 plate reader (... | US Patent US9738628 (2017) BindingDB Entry DOI: 10.7270/Q27P91H7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cadherin-1 [819-873]/Catenin beta-1 [138-686] (Homo sapiens (Human)) | BDBM213761 (US9284299, 12 | US9738628, Compound 12) | PDB GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 1.04E+5 | -5.43 | n/a | n/a | n/a | n/a | n/a | n/a | 25 |
University of Utah Research Foundation US Patent | Assay Description Experiments were performed in 96-well Microfluor 2 black plates (Waltham, Mass.), and the samples were read by a Synergy 2 plate reader (Biotek, Wino... | US Patent US9284299 (2016) BindingDB Entry DOI: 10.7270/Q2WW7GGC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cadherin-1 [819-873]/Catenin beta-1 [138-686] (Homo sapiens (Human)) | BDBM213761 (US9284299, 12 | US9738628, Compound 12) | PDB GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 1.05E+5 | -5.42 | n/a | n/a | n/a | n/a | n/a | 7.4 | 25 |
University of Utah Research Foundation US Patent | Assay Description Experiments were performed in white opaque 384-well plates from PerkinElmer (Waltham, Mass.), and the samples were read on a Synergy 2 plate reader (... | US Patent US9284299 (2016) BindingDB Entry DOI: 10.7270/Q2WW7GGC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenomatous polyposis coli protein [1477-1519]/Catenin beta-1 [138-686] (Homo sapiens (Human)) | BDBM213761 (US9284299, 12 | US9738628, Compound 12) | PDB GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 1.71E+5 | -5.14 | n/a | n/a | n/a | n/a | n/a | 7.4 | 25 |
University of Utah Research Foundation US Patent | Assay Description Experiments were performed in white opaque 384-well plates from PerkinElmer (Waltham, Mass.), and the samples were read on a Synergy 2 plate reader (... | US Patent US9284299 (2016) BindingDB Entry DOI: 10.7270/Q2WW7GGC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenomatous polyposis coli protein [1477-1519]/Catenin beta-1 [138-686] (Homo sapiens (Human)) | BDBM213761 (US9284299, 12 | US9738628, Compound 12) | PDB GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 1.76E+5 | -5.12 | n/a | n/a | n/a | n/a | n/a | n/a | 25 |
University of Utah Research Foundation US Patent | Assay Description Experiments were performed in 96-well Microfluor 2 black plates (Waltham, Mass.), and the samples were read by a Synergy 2 plate reader (Biotek, Wino... | US Patent US9284299 (2016) BindingDB Entry DOI: 10.7270/Q2WW7GGC | |||||||||||
More data for this Ligand-Target Pair |