BDBM223137 P5i-6
SMILES: NC(=O)N\N=C\c1ccc(o1)-c1ccc(Cl)cc1
InChI Key: InChIKey=ANUWWIQYOYPMTQ-VIZOYTHASA-N
Data: 6 IC50
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Protein-arginine N-methyltransferase 1 (Homo sapiens (Human)) | BDBM223137 (P5i-6) | PDB B.MOAD GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | 25 |
Sichuan University | Assay Description All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the... | Chem Biol Drug Des 89: 585-598 (2017) Article DOI: 10.1111/cbdd.12881 BindingDB Entry DOI: 10.7270/Q21V5CTR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein arginine methyltransferase 3 (PRMT3) (Homo sapiens (Human)) | BDBM223137 (P5i-6) | PDB B.MOAD GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | 25 |
Sichuan University | Assay Description All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the... | Chem Biol Drug Des 89: 585-598 (2017) Article DOI: 10.1111/cbdd.12881 BindingDB Entry DOI: 10.7270/Q21V5CTR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein arginine methyltransferase 8 (PRMT8) (Homo sapiens (Human)) | BDBM223137 (P5i-6) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | 25 |
Sichuan University | Assay Description All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the... | Chem Biol Drug Des 89: 585-598 (2017) Article DOI: 10.1111/cbdd.12881 BindingDB Entry DOI: 10.7270/Q21V5CTR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein arginine N-methyltransferase 6 (Homo sapiens (Human)) | BDBM223137 (P5i-6) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | 25 |
Sichuan University | Assay Description All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the... | Chem Biol Drug Des 89: 585-598 (2017) Article DOI: 10.1111/cbdd.12881 BindingDB Entry DOI: 10.7270/Q21V5CTR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein arginine methyltransferase 7 (PRMT7) (Homo sapiens (Human)) | BDBM223137 (P5i-6) | PDB UniProtKB/SwissProt UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | 25 |
Sichuan University | Assay Description All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the... | Chem Biol Drug Des 89: 585-598 (2017) Article DOI: 10.1111/cbdd.12881 BindingDB Entry DOI: 10.7270/Q21V5CTR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone-arginine methyltransferase CARM1 (Homo sapiens (Human)) | BDBM223137 (P5i-6) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | 25 |
Sichuan University | Assay Description All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the... | Chem Biol Drug Des 89: 585-598 (2017) Article DOI: 10.1111/cbdd.12881 BindingDB Entry DOI: 10.7270/Q21V5CTR | |||||||||||
More data for this Ligand-Target Pair |