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SMILES: Cc1cccn2c(ncc12)C1(CC1)NC(=O)[C@@H]1[C@H]2CNC[C@@H]12

InChI Key: InChIKey=LGGFQBURWYHOSH-IMRBUKKESA-N

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 312009   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Somatostatin receptor type 4 (Homo sapiens (Human))	BDBM312009 (US10166214, Example 145 | US10675268, Example 145) Show SMILES Cc1cccn2c(ncc12)C1(CC1)NC(=O)[C@@H]1[C@H]2CNC[C@@H]12 |r| Show InChI InChI=1S/C17H20N4O/c1-10-3-2-6-21-13(10)9-19-16(21)17(4-5-17)20-15(22)14-11-7-18-8-12(11)14/h2-3,6,9,11-12,14,18H,4-5,7-8H2,1H3,(H,20,22)/t11-,12+,14+	PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	0.900	n/a	n/a	n/a	n/a
Centrexion Therapeutics Corporation US Patent					Assay Description The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...				US Patent US10675268 (2020) BindingDB Entry DOI: 10.7270/Q21C20XK
					More data for this Ligand-Target Pair
Somatostatin receptor type 4 (Homo sapiens (Human))	BDBM312009 (US10166214, Example 145 | US10675268, Example 145) Show SMILES Cc1cccn2c(ncc12)C1(CC1)NC(=O)[C@@H]1[C@H]2CNC[C@@H]12 |r| Show InChI InChI=1S/C17H20N4O/c1-10-3-2-6-21-13(10)9-19-16(21)17(4-5-17)20-15(22)14-11-7-18-8-12(11)14/h2-3,6,9,11-12,14,18H,4-5,7-8H2,1H3,(H,20,22)/t11-,12+,14+	PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	n/a	n/a	0.900	n/a	n/a	n/a	n/a
Centrexion Therapeutics Corporation US Patent					Assay Description The activation of the SSTR4 receptor (Gi coupled) causes an inhibition of intracellular cAMP after stimulation with Forskolin, which can be quantifia...				US Patent US10166214 (2019) BindingDB Entry DOI: 10.7270/Q2D50Q16
					More data for this Ligand-Target Pair