null

SMILES: CN(c1ccc(Oc2nc(O)c3ccncc3n2)cc1)c1cccc(c1)C1=CCN(C)CC1

InChI Key: InChIKey=VFLAYFWGNVAVEN-UHFFFAOYSA-N

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 347132   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM347132 (2-(4-(methyl(3-(1-methyl-1,2,3,6- tetrahydropyridi...) Show SMILES CN(c1ccc(Oc2nc(O)c3ccncc3n2)cc1)c1cccc(c1)C1=CCN(C)CC1 |t:30| Show InChI InChI=1S/C26H25N5O2/c1-30-14-11-18(12-15-30)19-4-3-5-21(16-19)31(2)20-6-8-22(9-7-20)33-26-28-24-17-27-13-10-23(24)25(32)29-26/h3-11,13,16-17H,12,14-15H2,1-2H3,(H,28,29,32)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<100	n/a	n/a	n/a	n/a	n/a	n/a
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate-format under the following reaction conditions: 0.3 ...				US Patent US10208039 (2019) BindingDB Entry DOI: 10.7270/Q241706J
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM347132 (2-(4-(methyl(3-(1-methyl-1,2,3,6- tetrahydropyridi...) Show SMILES CN(c1ccc(Oc2nc(O)c3ccncc3n2)cc1)c1cccc(c1)C1=CCN(C)CC1 |t:30| Show InChI InChI=1S/C26H25N5O2/c1-30-14-11-18(12-15-30)19-4-3-5-21(16-19)31(2)20-6-8-22(9-7-20)33-26-28-24-17-27-13-10-23(24)25(32)29-26/h3-11,13,16-17H,12,14-15H2,1-2H3,(H,28,29,32)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<100	n/a	n/a	n/a	n/a	n/a	n/a
CELGENE QUANTICEL RESEARCH, INC. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate-format under the following reaction conditions: 0.3 ...				US Patent US10202381 (2019) BindingDB Entry DOI: 10.7270/Q2SX6GBM
					More data for this Ligand-Target Pair