Found 21 hits for monomerid = 50005944 Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
Sterol O-acyltransferase 1
(Homo sapiens (Human)) | BDBM50005944
![PNG](/data/jpeg/tenK5000/BindingDB_50005944.png) (2,2-Dimethyl-dodecanoic acid (2,4,6-trimethoxy-phe...)Show InChI InChI=1S/C23H39NO4/c1-7-8-9-10-11-12-13-14-15-23(2,3)22(25)24-21-19(27-5)16-18(26-4)17-20(21)28-6/h16-17H,7-15H2,1-6H3,(H,24,25) | PDB
KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
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Similars
| PDB PubMed
| n/a | n/a | 619 | n/a | n/a | n/a | n/a | n/a | n/a |
Azwell Inc.
Curated by ChEMBL
| Assay Description Compound was tested for inhibitory activity against ACAT from canine intestine |
Bioorg Med Chem Lett 9: 2039-42 (1999)
BindingDB Entry DOI: 10.7270/Q2FF3RJJ |
More data for this Ligand-Target Pair | ![3D 3D](/images/Docked_3d.png) 3D Structure (crystal) |
Acyl coenzyme A:cholesterol acyltransferase 1
(Mus musculus) | BDBM50005944
![PNG](/data/jpeg/tenK5000/BindingDB_50005944.png) (2,2-Dimethyl-dodecanoic acid (2,4,6-trimethoxy-phe...)Show InChI InChI=1S/C23H39NO4/c1-7-8-9-10-11-12-13-14-15-23(2,3)22(25)24-21-19(27-5)16-18(26-4)17-20(21)28-6/h16-17H,7-15H2,1-6H3,(H,24,25) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
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Similars
| PDB Article PubMed
| n/a | n/a | 310 | n/a | n/a | n/a | n/a | n/a | n/a |
Kowa Co., Ltd.
Curated by ChEMBL
| Assay Description Inhibition of ACAT1 in mouse J774 cells assessed as reduction in esterified cholesterol accumulation after 18 hrs in presence of 25-hydroxycholestero... |
Bioorg Med Chem 26: 4001-4013 (2018)
Article DOI: 10.1016/j.bmc.2018.06.024 BindingDB Entry DOI: 10.7270/Q22F7R3T |
More data for this Ligand-Target Pair | ![3D 3D](/images/Docked_3d.png) 3D Structure (crystal) |
Sterol O-acyltransferase 1
(Homo sapiens (Human)) | BDBM50005944
![PNG](/data/jpeg/tenK5000/BindingDB_50005944.png) (2,2-Dimethyl-dodecanoic acid (2,4,6-trimethoxy-phe...)Show InChI InChI=1S/C23H39NO4/c1-7-8-9-10-11-12-13-14-15-23(2,3)22(25)24-21-19(27-5)16-18(26-4)17-20(21)28-6/h16-17H,7-15H2,1-6H3,(H,24,25) | PDB
KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
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| PDB PubMed
| n/a | n/a | 838 | n/a | n/a | n/a | n/a | n/a | n/a |
Azwell Inc.
Curated by ChEMBL
| Assay Description Compound was tested for inhibitory activity against ACAT from HepG2 microsome in human |
Bioorg Med Chem Lett 9: 2039-42 (1999)
BindingDB Entry DOI: 10.7270/Q2FF3RJJ |
More data for this Ligand-Target Pair | ![3D 3D](/images/Docked_3d.png) 3D Structure (crystal) |
Sterol O-acyltransferase 1
(Homo sapiens (Human)) | BDBM50005944
![PNG](/data/jpeg/tenK5000/BindingDB_50005944.png) (2,2-Dimethyl-dodecanoic acid (2,4,6-trimethoxy-phe...)Show InChI InChI=1S/C23H39NO4/c1-7-8-9-10-11-12-13-14-15-23(2,3)22(25)24-21-19(27-5)16-18(26-4)17-20(21)28-6/h16-17H,7-15H2,1-6H3,(H,24,25) | PDB
KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
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| PDB PubMed
| n/a | n/a | 926 | n/a | n/a | n/a | n/a | n/a | n/a |
Azwell Inc.
Curated by ChEMBL
| Assay Description Compound was tested for inhibitory activity against ACAT from U937 microsome in human |
Bioorg Med Chem Lett 9: 2039-42 (1999)
BindingDB Entry DOI: 10.7270/Q2FF3RJJ |
More data for this Ligand-Target Pair | ![3D 3D](/images/Docked_3d.png) 3D Structure (crystal) |
Sterol O-acyltransferase 1
(Homo sapiens (Human)) | BDBM50005944
![PNG](/data/jpeg/tenK5000/BindingDB_50005944.png) (2,2-Dimethyl-dodecanoic acid (2,4,6-trimethoxy-phe...)Show InChI InChI=1S/C23H39NO4/c1-7-8-9-10-11-12-13-14-15-23(2,3)22(25)24-21-19(27-5)16-18(26-4)17-20(21)28-6/h16-17H,7-15H2,1-6H3,(H,24,25) | PDB
KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
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| PDB PubMed
| n/a | n/a | 4.59E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Azwell Inc.
Curated by ChEMBL
| Assay Description Compound was tested for inhibitory activity against ACAT from HepG2 microsome in human |
Bioorg Med Chem Lett 9: 2039-42 (1999)
BindingDB Entry DOI: 10.7270/Q2FF3RJJ |
More data for this Ligand-Target Pair | ![3D 3D](/images/Docked_3d.png) 3D Structure (crystal) |
Acyl-CoA:cholesterol acyltransferase
(Oryctolagus cuniculus) | BDBM50005944
![PNG](/data/jpeg/tenK5000/BindingDB_50005944.png) (2,2-Dimethyl-dodecanoic acid (2,4,6-trimethoxy-phe...)Show InChI InChI=1S/C23H39NO4/c1-7-8-9-10-11-12-13-14-15-23(2,3)22(25)24-21-19(27-5)16-18(26-4)17-20(21)28-6/h16-17H,7-15H2,1-6H3,(H,24,25) | PDB
Reactome pathway KEGG
UniProtKB/TrEMBL
DrugBank GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
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| n/a | n/a | 1.95E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Azwell Inc.
Curated by ChEMBL
| Assay Description Compound was tested for inhibitory activity against ACAT from rabbit adrenal gland |
Bioorg Med Chem Lett 9: 2039-42 (1999)
BindingDB Entry DOI: 10.7270/Q2FF3RJJ |
More data for this Ligand-Target Pair | ![3D 3D](/images/Docked_3d.png) 3D Structure (crystal) |
Acyl-CoA:cholesterol acyltransferase
(Oryctolagus cuniculus) | BDBM50005944
![PNG](/data/jpeg/tenK5000/BindingDB_50005944.png) (2,2-Dimethyl-dodecanoic acid (2,4,6-trimethoxy-phe...)Show InChI InChI=1S/C23H39NO4/c1-7-8-9-10-11-12-13-14-15-23(2,3)22(25)24-21-19(27-5)16-18(26-4)17-20(21)28-6/h16-17H,7-15H2,1-6H3,(H,24,25) | PDB
Reactome pathway KEGG
UniProtKB/TrEMBL
DrugBank GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
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| PDB PubMed
| n/a | n/a | 191 | n/a | n/a | n/a | n/a | n/a | n/a |
Azwell Inc.
Curated by ChEMBL
| Assay Description Compound was tested for inhibitory activity against ACAT from rabbit liver |
Bioorg Med Chem Lett 9: 2039-42 (1999)
BindingDB Entry DOI: 10.7270/Q2FF3RJJ |
More data for this Ligand-Target Pair | ![3D 3D](/images/Docked_3d.png) 3D Structure (crystal) |
Acyl-CoA:cholesterol acyltransferase
(Oryctolagus cuniculus) | BDBM50005944
![PNG](/data/jpeg/tenK5000/BindingDB_50005944.png) (2,2-Dimethyl-dodecanoic acid (2,4,6-trimethoxy-phe...)Show InChI InChI=1S/C23H39NO4/c1-7-8-9-10-11-12-13-14-15-23(2,3)22(25)24-21-19(27-5)16-18(26-4)17-20(21)28-6/h16-17H,7-15H2,1-6H3,(H,24,25) | PDB
Reactome pathway KEGG
UniProtKB/TrEMBL
DrugBank GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
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| PDB PubMed
| n/a | n/a | 152 | n/a | n/a | n/a | n/a | n/a | n/a |
Azwell Inc.
Curated by ChEMBL
| Assay Description Compound was tested for inhibitory activity against ACAT from Caco-2 microsome in human |
Bioorg Med Chem Lett 9: 2039-42 (1999)
BindingDB Entry DOI: 10.7270/Q2FF3RJJ |
More data for this Ligand-Target Pair | ![3D 3D](/images/Docked_3d.png) 3D Structure (crystal) |
Sterol O-acyltransferase 1
(Homo sapiens (Human)) | BDBM50005944
![PNG](/data/jpeg/tenK5000/BindingDB_50005944.png) (2,2-Dimethyl-dodecanoic acid (2,4,6-trimethoxy-phe...)Show InChI InChI=1S/C23H39NO4/c1-7-8-9-10-11-12-13-14-15-23(2,3)22(25)24-21-19(27-5)16-18(26-4)17-20(21)28-6/h16-17H,7-15H2,1-6H3,(H,24,25) | PDB
KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
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| PDB PubMed
| n/a | n/a | 4.65E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Azwell Inc.
Curated by ChEMBL
| Assay Description Compound was tested for inhibitory activity against ACAT from canine adrenal gland |
Bioorg Med Chem Lett 9: 2039-42 (1999)
BindingDB Entry DOI: 10.7270/Q2FF3RJJ |
More data for this Ligand-Target Pair | ![3D 3D](/images/Docked_3d.png) 3D Structure (crystal) |
Sterol O-acyltransferase, Soat
(Rattus norvegicus) | BDBM50005944
![PNG](/data/jpeg/tenK5000/BindingDB_50005944.png) (2,2-Dimethyl-dodecanoic acid (2,4,6-trimethoxy-phe...)Show InChI InChI=1S/C23H39NO4/c1-7-8-9-10-11-12-13-14-15-23(2,3)22(25)24-21-19(27-5)16-18(26-4)17-20(21)28-6/h16-17H,7-15H2,1-6H3,(H,24,25) | PDB
KEGG
UniProtKB/SwissProt
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| n/a | n/a | 110 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description Concentration required for the in vitro inhibition of Acyl coenzyme A:cholesterol acyltransferase (ACAT) in liver microsomes isolated from cholestero... |
Bioorg Med Chem Lett 5: 289-294 (1995)
Article DOI: 10.1016/0960-894X(95)00024-N BindingDB Entry DOI: 10.7270/Q2FQ9WKP |
More data for this Ligand-Target Pair | ![3D 3D](/images/Docked_3d.png) 3D Structure (crystal) |
Sterol O-acyltransferase, Soat
(Rattus norvegicus) | BDBM50005944
![PNG](/data/jpeg/tenK5000/BindingDB_50005944.png) (2,2-Dimethyl-dodecanoic acid (2,4,6-trimethoxy-phe...)Show InChI InChI=1S/C23H39NO4/c1-7-8-9-10-11-12-13-14-15-23(2,3)22(25)24-21-19(27-5)16-18(26-4)17-20(21)28-6/h16-17H,7-15H2,1-6H3,(H,24,25) | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
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| n/a | n/a | 110 | n/a | n/a | n/a | n/a | n/a | n/a |
Warner-Lambert Company
Curated by ChEMBL
| Assay Description Concentration required for the in vitro inhibition of Acyl coenzyme A:cholesterol acyltransferase (ACAT) in liver microsomes isolated from cholestero... |
Bioorg Med Chem Lett 5: 295-300 (1995)
BindingDB Entry DOI: 10.7270/Q29Z94WS |
More data for this Ligand-Target Pair | ![3D 3D](/images/Docked_3d.png) 3D Structure (crystal) |
Acyl coenzyme A:cholesterol acyltransferase 1
(Mus musculus) | BDBM50005944
![PNG](/data/jpeg/tenK5000/BindingDB_50005944.png) (2,2-Dimethyl-dodecanoic acid (2,4,6-trimethoxy-phe...)Show InChI InChI=1S/C23H39NO4/c1-7-8-9-10-11-12-13-14-15-23(2,3)22(25)24-21-19(27-5)16-18(26-4)17-20(21)28-6/h16-17H,7-15H2,1-6H3,(H,24,25) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
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| PDB Article
| n/a | n/a | 400 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description Compound was tested for its ability to penetrate the cell wall and inhibit macrophage ACAT in cell culture using murine IC-21 macrophages (MAI) |
Bioorg Med Chem Lett 6: 1753-1758 (1996)
Article DOI: 10.1016/0960-894X(96)00310-1 BindingDB Entry DOI: 10.7270/Q2VD6ZF6 |
More data for this Ligand-Target Pair | ![3D 3D](/images/Docked_3d.png) 3D Structure (crystal) |
Sterol O-acyltransferase, Soat
(Rattus norvegicus) | BDBM50005944
![PNG](/data/jpeg/tenK5000/BindingDB_50005944.png) (2,2-Dimethyl-dodecanoic acid (2,4,6-trimethoxy-phe...)Show InChI InChI=1S/C23H39NO4/c1-7-8-9-10-11-12-13-14-15-23(2,3)22(25)24-21-19(27-5)16-18(26-4)17-20(21)28-6/h16-17H,7-15H2,1-6H3,(H,24,25) | PDB
KEGG
UniProtKB/SwissProt
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| PDB PubMed
| n/a | n/a | 6.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute
Curated by ChEMBL
| Assay Description In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase 1, rat liver microsomal assay |
J Med Chem 38: 1600-7 (1995)
BindingDB Entry DOI: 10.7270/Q26T0KN9 |
More data for this Ligand-Target Pair | ![3D 3D](/images/Docked_3d.png) 3D Structure (crystal) |
Acyl-CoA:cholesterol acyltransferase
(Oryctolagus cuniculus) | BDBM50005944
![PNG](/data/jpeg/tenK5000/BindingDB_50005944.png) (2,2-Dimethyl-dodecanoic acid (2,4,6-trimethoxy-phe...)Show InChI InChI=1S/C23H39NO4/c1-7-8-9-10-11-12-13-14-15-23(2,3)22(25)24-21-19(27-5)16-18(26-4)17-20(21)28-6/h16-17H,7-15H2,1-6H3,(H,24,25) | PDB
Reactome pathway KEGG
UniProtKB/TrEMBL
DrugBank GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
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| PDB Article PubMed
| n/a | n/a | 140 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute for Bio-Medical Research
Curated by ChEMBL
| Assay Description Inhibitory activity against Acyl coenzyme A:cholesterol acyltransferase 1 obtained from rabbit intestine microsomes |
J Med Chem 39: 1262-70 (1996)
Article DOI: 10.1021/jm950828+ BindingDB Entry DOI: 10.7270/Q24T6HGW |
More data for this Ligand-Target Pair | ![3D 3D](/images/Docked_3d.png) 3D Structure (crystal) |
Sterol O-acyltransferase, Soat
(Rattus norvegicus) | BDBM50005944
![PNG](/data/jpeg/tenK5000/BindingDB_50005944.png) (2,2-Dimethyl-dodecanoic acid (2,4,6-trimethoxy-phe...)Show InChI InChI=1S/C23H39NO4/c1-7-8-9-10-11-12-13-14-15-23(2,3)22(25)24-21-19(27-5)16-18(26-4)17-20(21)28-6/h16-17H,7-15H2,1-6H3,(H,24,25) | PDB
KEGG
UniProtKB/SwissProt
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| PDB PubMed
| n/a | n/a | 6.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute
Curated by ChEMBL
| Assay Description Concentration required for 50% inhibition of Acyl coenzyme A:cholesterol acyltransferase activity using microsomal ACAT assay |
J Med Chem 37: 1733-6 (1994)
BindingDB Entry DOI: 10.7270/Q20P0Z20 |
More data for this Ligand-Target Pair | ![3D 3D](/images/Docked_3d.png) 3D Structure (crystal) |
Acyl-CoA:cholesterol acyltransferase
(Oryctolagus cuniculus) | BDBM50005944
![PNG](/data/jpeg/tenK5000/BindingDB_50005944.png) (2,2-Dimethyl-dodecanoic acid (2,4,6-trimethoxy-phe...)Show InChI InChI=1S/C23H39NO4/c1-7-8-9-10-11-12-13-14-15-23(2,3)22(25)24-21-19(27-5)16-18(26-4)17-20(21)28-6/h16-17H,7-15H2,1-6H3,(H,24,25) | PDB
Reactome pathway KEGG
UniProtKB/TrEMBL
DrugBank GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
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| PDB PubMed
| n/a | n/a | 73 | n/a | n/a | n/a | n/a | n/a | n/a |
Warner-Lambert Company
Curated by ChEMBL
| Assay Description In vitro inhibition of acyl coenzyme A:cholesterol acyltransferase, in intestinal microsomes isolated from cholesterol-fed rabbits |
J Med Chem 35: 1609-17 (1992)
BindingDB Entry DOI: 10.7270/Q2G44QXN |
More data for this Ligand-Target Pair | ![3D 3D](/images/Docked_3d.png) 3D Structure (crystal) |
Sterol O-acyltransferase, Soat
(Rattus norvegicus) | BDBM50005944
![PNG](/data/jpeg/tenK5000/BindingDB_50005944.png) (2,2-Dimethyl-dodecanoic acid (2,4,6-trimethoxy-phe...)Show InChI InChI=1S/C23H39NO4/c1-7-8-9-10-11-12-13-14-15-23(2,3)22(25)24-21-19(27-5)16-18(26-4)17-20(21)28-6/h16-17H,7-15H2,1-6H3,(H,24,25) | PDB
KEGG
UniProtKB/SwissProt
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| PDB Article PubMed
| n/a | n/a | 149 | n/a | n/a | n/a | n/a | n/a | n/a |
Institute for Bio-Medical Research
Curated by ChEMBL
| Assay Description Inhibitory activity of the compound against Acyl coenzyme A:cholesterol acyltransferase 1 obtained from rat liver microsomes |
J Med Chem 39: 1262-70 (1996)
Article DOI: 10.1021/jm950828+ BindingDB Entry DOI: 10.7270/Q24T6HGW |
More data for this Ligand-Target Pair | ![3D 3D](/images/Docked_3d.png) 3D Structure (crystal) |
Sterol O-acyltransferase, Soat
(Rattus norvegicus) | BDBM50005944
![PNG](/data/jpeg/tenK5000/BindingDB_50005944.png) (2,2-Dimethyl-dodecanoic acid (2,4,6-trimethoxy-phe...)Show InChI InChI=1S/C23H39NO4/c1-7-8-9-10-11-12-13-14-15-23(2,3)22(25)24-21-19(27-5)16-18(26-4)17-20(21)28-6/h16-17H,7-15H2,1-6H3,(H,24,25) | PDB
KEGG
UniProtKB/SwissProt
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| PDB PubMed
| n/a | n/a | 73 | n/a | n/a | n/a | n/a | n/a | n/a |
Parke-Davis Pharmaceutical Research
Curated by ChEMBL
| Assay Description In vitro inhibition of rat intestinal acyl coenzyme A:cholesterol acyltransferase using [1-14C]oleolyl-CoA |
J Med Chem 37: 1810-22 (1994)
BindingDB Entry DOI: 10.7270/Q2CR5V0V |
More data for this Ligand-Target Pair | ![3D 3D](/images/Docked_3d.png) 3D Structure (crystal) |
Sterol O-acyltransferase 1
(Homo sapiens (Human)) | BDBM50005944
![PNG](/data/jpeg/tenK5000/BindingDB_50005944.png) (2,2-Dimethyl-dodecanoic acid (2,4,6-trimethoxy-phe...)Show InChI InChI=1S/C23H39NO4/c1-7-8-9-10-11-12-13-14-15-23(2,3)22(25)24-21-19(27-5)16-18(26-4)17-20(21)28-6/h16-17H,7-15H2,1-6H3,(H,24,25) | PDB
KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
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| PDB PubMed
| n/a | n/a | 4.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description Inhibition of Acyl coenzyme A:cholesterol acyltransferase (ACAT) |
J Med Chem 24: 496-9 (1981)
BindingDB Entry DOI: 10.7270/Q2K64JTV |
More data for this Ligand-Target Pair | ![3D 3D](/images/Docked_3d.png) 3D Structure (crystal) |
Sterol O-acyltransferase 1
(Homo sapiens (Human)) | BDBM50005944
![PNG](/data/jpeg/tenK5000/BindingDB_50005944.png) (2,2-Dimethyl-dodecanoic acid (2,4,6-trimethoxy-phe...)Show InChI InChI=1S/C23H39NO4/c1-7-8-9-10-11-12-13-14-15-23(2,3)22(25)24-21-19(27-5)16-18(26-4)17-20(21)28-6/h16-17H,7-15H2,1-6H3,(H,24,25) | PDB
KEGG
UniProtKB/SwissProt
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| PDB Article PubMed
| n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
Kansas State University
Curated by ChEMBL
| Assay Description Inhibition of ACAT activity in human MC65 cells using NBD-cholesterol staining after 48 hrs by fluorescence assay |
J Med Chem 55: 8969-73 (2012)
Article DOI: 10.1021/jm3012189 BindingDB Entry DOI: 10.7270/Q2000370 |
More data for this Ligand-Target Pair | ![3D 3D](/images/Docked_3d.png) 3D Structure (crystal) |
Sterol O-acyltransferase 1
(Homo sapiens (Human)) | BDBM50005944
![PNG](/data/jpeg/tenK5000/BindingDB_50005944.png) (2,2-Dimethyl-dodecanoic acid (2,4,6-trimethoxy-phe...)Show InChI InChI=1S/C23H39NO4/c1-7-8-9-10-11-12-13-14-15-23(2,3)22(25)24-21-19(27-5)16-18(26-4)17-20(21)28-6/h16-17H,7-15H2,1-6H3,(H,24,25) | PDB
KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
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CHEMBL PC cid PC sid PDB UniChem
Patents
Similars
| PDB PubMed
| n/a | n/a | 5.87E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Azwell Inc.
Curated by ChEMBL
| Assay Description Compound was tested for inhibitory activity against ACAT from U937 microsome in human |
Bioorg Med Chem Lett 9: 2039-42 (1999)
BindingDB Entry DOI: 10.7270/Q2FF3RJJ |
More data for this Ligand-Target Pair | ![3D 3D](/images/Docked_3d.png) 3D Structure (crystal) |