null
SMILES: [#6]-[#8]-c1ccc(cc1)-[#6](=[#6]\[#6]=[#6]\[#6](=O)-[#7]-c1ccc(cc1)-c1cccnc1)\c1ccc(-[#8]-[#6])cc1
InChI Key: InChIKey=AHPDSBLXHZAIHR-XVNBXDOJSA-N
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018347 (5,5-Bis-(4-methoxy-phenyl)-penta-2,4-dienoic acid ...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand | J Med Chem 32: 1820-35 (1989) BindingDB Entry DOI: 10.7270/Q2NZ86MR | |||||||||||
More data for this Ligand-Target Pair |