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SMILES: [#6]-[#8]-c1ccccc1\[#6](=[#6]\[#6]=[#6]\[#6](=O)-[#7]-[#6]-[#6]-[#6]-[#6]-c1cccnc1)-c1ccccc1-[#8]-[#6]

InChI Key: InChIKey=CPGHLTGASAARCO-GIJQJNRQSA-N

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50018359   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kcal/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Platelet-activating factor receptor


(Homo sapiens (Human))		BDBM50018359
PNG
(5,5-Bis-(2-methoxy-phenyl)-penta-2,4-dienoic acid ...)
Show SMILES [#6]-[#8]-c1ccccc1\[#6](=[#6]\[#6]=[#6]\[#6](=O)-[#7]-[#6]-[#6]-[#6]-[#6]-c1cccnc1)-c1ccccc1-[#8]-[#6]
Show InChI InChI=1S/C28H30N2O3/c1-32-26-16-5-3-13-24(26)23(25-14-4-6-17-27(25)33-2)15-9-18-28(31)30-20-8-7-11-22-12-10-19-29-21-22/h3-6,9-10,12-19,21H,7-8,11,20H2,1-2H3,(H,30,31)/b18-9+
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n/an/a 40n/an/an/an/an/an/a



Roche Research Center

Curated by ChEMBL


Assay Description
Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand

J Med Chem 32: 1820-35 (1989)


BindingDB Entry DOI: 10.7270/Q2NZ86MR
More data for this
Ligand-Target Pair