null
SMILES: CCOC(=O)C1C(c2c(C)noc2CCc2ccccc2)C(C(=O)OCC)=C(C)N=C1C
InChI Key: InChIKey=REQVROPNOXACSN-UHFFFAOYSA-N
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Voltage-dependent L-type calcium channel subunit alpha-1C (RAT) | BDBM50079462 (2,6-Dimethyl-4-(3-methyl-5-phenethyl-isoxazol-4-yl...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 25 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
State University of New York Curated by ChEMBL | Assay Description Displacement of [3H](+)-PN200-110 binding from calcium channels of rat cardiac membranes. | J Med Chem 42: 3087-93 (1999) Article DOI: 10.1021/jm980439q BindingDB Entry DOI: 10.7270/Q20C4TZD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Voltage-dependent L-type calcium channel subunit alpha-1C (Homo sapiens (Human)) | BDBM50079462 (2,6-Dimethyl-4-(3-methyl-5-phenethyl-isoxazol-4-yl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 23 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
State University of New York Curated by ChEMBL | Assay Description Displacement of [3H](+)-PN200-110 binding to calcium channels in guinea pig cardiac membranes. | J Med Chem 42: 3087-93 (1999) Article DOI: 10.1021/jm980439q BindingDB Entry DOI: 10.7270/Q20C4TZD | |||||||||||
More data for this Ligand-Target Pair |