BDBM50128926 CHEMBL304896::N-(5-Ethyl-6-oxo-5,6-dihydro-phenanthridin-9-yl)-2-pyridin-4-yl-acetamide
SMILES: CCn1c2ccccc2c2cc(NC(=O)Cc3ccncc3)ccc2c1=O
InChI Key: InChIKey=AVGCFTCKHIHCOQ-UHFFFAOYSA-N
Data: 1 KI
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Neuropeptide Y receptor type 5 ( NPY Y5) (Homo sapiens (Human)) | BDBM50128926 (CHEMBL304896 | N-(5-Ethyl-6-oxo-5,6-dihydro-phenan...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 12 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Binding affinity towards human neuropeptide Y receptor type 5 using 125[I]-PYY as radioligand | Bioorg Med Chem Lett 13: 1989-92 (2003) BindingDB Entry DOI: 10.7270/Q2057F9D | |||||||||||
More data for this Ligand-Target Pair |