null
SMILES: CCCC(=O)c1ccc(OCCCCOc2ccc(cc2)-c2nnn[nH]2)c(C)c1O
InChI Key: InChIKey=GRXBQBZQNCYJFJ-UHFFFAOYSA-N
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Metabotropic glutamate receptor 2 (Homo sapiens (Human)) | BDBM50153750 (1-(2-Hydroxy-3-methyl-4-{4-[4-(2H-tetrazol-5-yl)-p...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 304 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Effective concentration for binding to human metabotropic glutamate receptor 2 as determined by GTPgammaS assay | Bioorg Med Chem Lett 14: 5329-32 (2004) Article DOI: 10.1016/j.bmcl.2004.08.020 BindingDB Entry DOI: 10.7270/Q21Z43W0 | |||||||||||
More data for this Ligand-Target Pair |