BDBM50214774 CHEMBL3392230
SMILES: CCOC(=O)C1=C(C)NC(C)=C(C#N)[C@@H]1c1cnccc1-c1ccc2ccccc2c1
InChI Key: InChIKey=DRAFQLUUZHHPFJ-RUZDIDTESA-N
Data: 1 IC50
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
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Voltage-dependent L-type calcium channel subunit alpha-1C (Homo sapiens (Human)) | BDBM50214774 (CHEMBL3392230) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding affinity for DHP(Dihydropyridine) site of L-type calcium channel of calf heart in the resting state | Bioorg Med Chem Lett 7: 2519-2522 (1997) Article DOI: 10.1016/S0960-894X(97)10006-3 BindingDB Entry DOI: 10.7270/Q24T6JDD | |||||||||||
More data for this Ligand-Target Pair |