BDBM50251001 CHEMBL457677::Kazinol F
SMILES: [#6]\[#6](-[#6])=[#6]\[#6]-c1c(-[#6]-[#6]-[#6]-c2ccc(-[#8])cc2-[#8])cc(-[#8])c(-[#8])c1-[#6]\[#6]=[#6](/[#6])-[#6]
InChI Key: InChIKey=PNQQDEFGJPUAGZ-UHFFFAOYSA-N
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Tyrosinase (Agaricus bisporus (Common mushroom)) | BDBM50251001 (CHEMBL457677 | Kazinol F) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 181 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Graduate School of Gyeongsang National University Curated by ChEMBL | Assay Description Inhibition of mushroom tyrosinase by kinetic based assay | Bioorg Med Chem 17: 35-41 (2008) Article DOI: 10.1016/j.bmc.2008.11.022 BindingDB Entry DOI: 10.7270/Q2GH9HTH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tyrosinase (Agaricus bisporus (Common mushroom)) | BDBM50251001 (CHEMBL457677 | Kazinol F) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 410 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Graduate School of Gyeongsang National University Curated by ChEMBL | Assay Description Inhibition of monophenolase activity of mushroom tyrosinase using as L-tyrosine substrate by Lineweaver-Burk plot based kinetic assay | Bioorg Med Chem 17: 35-41 (2008) Article DOI: 10.1016/j.bmc.2008.11.022 BindingDB Entry DOI: 10.7270/Q2GH9HTH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tyrosinase (Agaricus bisporus (Common mushroom)) | BDBM50251001 (CHEMBL457677 | Kazinol F) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 770 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Graduate School of Gyeongsang National University Curated by ChEMBL | Assay Description Inhibition of diphenolase activity of mushroom tyrosinase using as L-DOPA substrate by Lineweaver-Burk plot based kinetic assay | Bioorg Med Chem 17: 35-41 (2008) Article DOI: 10.1016/j.bmc.2008.11.022 BindingDB Entry DOI: 10.7270/Q2GH9HTH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tyrosinase (Agaricus bisporus (Common mushroom)) | BDBM50251001 (CHEMBL457677 | Kazinol F) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 960 | n/a | n/a | n/a | n/a | n/a | n/a |
Graduate School of Gyeongsang National University Curated by ChEMBL | Assay Description Inhibition of monophenolase activity of mushroom tyrosinase using as L-tyrosine substrate | Bioorg Med Chem 17: 35-41 (2008) Article DOI: 10.1016/j.bmc.2008.11.022 BindingDB Entry DOI: 10.7270/Q2GH9HTH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tyrosinase (Agaricus bisporus (Common mushroom)) | BDBM50251001 (CHEMBL457677 | Kazinol F) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Graduate School of Gyeongsang National University Curated by ChEMBL | Assay Description Inhibition of diphenolase activity of mushroom tyrosinase using as L-DOPA substrate | Bioorg Med Chem 17: 35-41 (2008) Article DOI: 10.1016/j.bmc.2008.11.022 BindingDB Entry DOI: 10.7270/Q2GH9HTH | |||||||||||
More data for this Ligand-Target Pair |