Found 6 hits for monomerid = 50299910 Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kcal/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Casein kinase I isoform delta
(Homo sapiens (Human)) | BDBM50299910
(4-(pyridin-3-ylmethylene)-2-styryloxazol-5(4H)-one...)Show SMILES O=C1OC(\C=C\c2ccccc2)=N/C/1=C\c1cccnc1 |c:12| Show InChI InChI=1S/C17H12N2O2/c20-17-15(11-14-7-4-10-18-12-14)19-16(21-17)9-8-13-5-2-1-3-6-13/h1-12H/b9-8+,15-11- | PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet 
| Purchase
CHEMBL
PC cid
PC sid
UniChem
Patents
| Article
PubMed
| n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
PharmaDesign, Inc.
Curated by ChEMBL
| Assay Description
Inhibition of CK1delta |
J Med Chem 52: 7323-7 (2009)
Article DOI: 10.1021/jm901191q
BindingDB Entry DOI: 10.7270/Q2639PTZ |
More data for this
Ligand-Target Pair | |
Fibroblast growth factor receptor 1
(Homo sapiens (Human)) | BDBM50299910
(4-(pyridin-3-ylmethylene)-2-styryloxazol-5(4H)-one...)Show SMILES O=C1OC(\C=C\c2ccccc2)=N/C/1=C\c1cccnc1 |c:12| Show InChI InChI=1S/C17H12N2O2/c20-17-15(11-14-7-4-10-18-12-14)19-16(21-17)9-8-13-5-2-1-3-6-13/h1-12H/b9-8+,15-11- | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| Purchase
CHEMBL
PC cid
PC sid
UniChem
Patents
| Article
PubMed
| n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
PharmaDesign, Inc.
Curated by ChEMBL
| Assay Description
Inhibition of FGFR1 |
J Med Chem 52: 7323-7 (2009)
Article DOI: 10.1021/jm901191q
BindingDB Entry DOI: 10.7270/Q2639PTZ |
More data for this
Ligand-Target Pair | |
Serine/threonine-protein kinase Sgk1
(Homo sapiens (Human)) | BDBM50299910
(4-(pyridin-3-ylmethylene)-2-styryloxazol-5(4H)-one...)Show SMILES O=C1OC(\C=C\c2ccccc2)=N/C/1=C\c1cccnc1 |c:12| Show InChI InChI=1S/C17H12N2O2/c20-17-15(11-14-7-4-10-18-12-14)19-16(21-17)9-8-13-5-2-1-3-6-13/h1-12H/b9-8+,15-11- | PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| Purchase
CHEMBL
PC cid
PC sid
UniChem
Patents
| Article
PubMed
| n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
PharmaDesign, Inc.
Curated by ChEMBL
| Assay Description
Inhibition of SGK1 |
J Med Chem 52: 7323-7 (2009)
Article DOI: 10.1021/jm901191q
BindingDB Entry DOI: 10.7270/Q2639PTZ |
More data for this
Ligand-Target Pair | |
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human)) | BDBM50299910
(4-(pyridin-3-ylmethylene)-2-styryloxazol-5(4H)-one...)Show SMILES O=C1OC(\C=C\c2ccccc2)=N/C/1=C\c1cccnc1 |c:12| Show InChI InChI=1S/C17H12N2O2/c20-17-15(11-14-7-4-10-18-12-14)19-16(21-17)9-8-13-5-2-1-3-6-13/h1-12H/b9-8+,15-11- | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| Purchase
CHEMBL
PC cid
PC sid
UniChem
Patents
| Article
PubMed
| n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
PharmaDesign, Inc.
Curated by ChEMBL
| Assay Description
Inhibition of KDR |
J Med Chem 52: 7323-7 (2009)
Article DOI: 10.1021/jm901191q
BindingDB Entry DOI: 10.7270/Q2639PTZ |
More data for this
Ligand-Target Pair | |
Mitogen-activated protein kinase 1
(Homo sapiens (Human)) | BDBM50299910
(4-(pyridin-3-ylmethylene)-2-styryloxazol-5(4H)-one...)Show SMILES O=C1OC(\C=C\c2ccccc2)=N/C/1=C\c1cccnc1 |c:12| Show InChI InChI=1S/C17H12N2O2/c20-17-15(11-14-7-4-10-18-12-14)19-16(21-17)9-8-13-5-2-1-3-6-13/h1-12H/b9-8+,15-11- | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| Purchase
CHEMBL
PC cid
PC sid
UniChem
Patents
| Article
PubMed
| n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
PharmaDesign, Inc.
Curated by ChEMBL
| Assay Description
Inhibition of Erk2 |
J Med Chem 52: 7323-7 (2009)
Article DOI: 10.1021/jm901191q
BindingDB Entry DOI: 10.7270/Q2639PTZ |
More data for this
Ligand-Target Pair | |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(Homo sapiens (Human)) | BDBM50299910
(4-(pyridin-3-ylmethylene)-2-styryloxazol-5(4H)-one...)Show SMILES O=C1OC(\C=C\c2ccccc2)=N/C/1=C\c1cccnc1 |c:12| Show InChI InChI=1S/C17H12N2O2/c20-17-15(11-14-7-4-10-18-12-14)19-16(21-17)9-8-13-5-2-1-3-6-13/h1-12H/b9-8+,15-11- | PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet
| Purchase
CHEMBL
PC cid
PC sid
UniChem
Patents
| Article
PubMed
| n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
PharmaDesign, Inc.
Curated by ChEMBL
| Assay Description
Inhibition of DYRK1R |
J Med Chem 52: 7323-7 (2009)
Article DOI: 10.1021/jm901191q
BindingDB Entry DOI: 10.7270/Q2639PTZ |
More data for this
Ligand-Target Pair | |
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