null
SMILES: CN1Cc2ccccc2[C@H](N=C1OCc1ccc(NS(C)(=O)=O)cc1)c1ccccc1
InChI Key: InChIKey=VFUWIUMIQOHXBB-HSZRJFAPSA-N
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50369030 (CHEMBL1788206) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 3.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Sterling Winthrop Research Curated by ChEMBL | Assay Description Blockade of the delayed rectifier K+ current (IKr) of guinea pig myocytes | J Med Chem 38: 2551-6 (1995) BindingDB Entry DOI: 10.7270/Q2H132N3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium channel protein type 5 subunit alpha (Homo sapiens (Human)) | BDBM50369030 (CHEMBL1788206) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.26E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Sterling Winthrop Research Curated by ChEMBL | Assay Description Blockade of Na+ current in frog oocytes expressing human cardiac sodium channel (HH1) | J Med Chem 38: 2551-6 (1995) BindingDB Entry DOI: 10.7270/Q2H132N3 | |||||||||||
More data for this Ligand-Target Pair |