Found 4 hits for monomerid = 50433356 Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
Histamine H4 Receptor
(Mus musculus (mouse)) | BDBM50433356
(CHEMBL2376801)Show InChI InChI=1S/C14H20N6/c1-3-9-6-11-12(17-7-9)13(19-14(15)18-11)20-5-4-10(8-20)16-2/h6-7,10,16H,3-5,8H2,1-2H3,(H2,15,18,19)/t10-/m1/s1 | Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| 85 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Griffin Discoveries BV
Curated by ChEMBL
| Assay Description Binding affinity to mouse histamine H4 receptor |
Bioorg Med Chem Lett 23: 2663-70 (2013)
Article DOI: 10.1016/j.bmcl.2013.02.091 BindingDB Entry DOI: 10.7270/Q2K35W11 |
More data for this Ligand-Target Pair | |
Histamine H4 Receptor
(Rattus norvegicus (rat)) | BDBM50433356
(CHEMBL2376801)Show InChI InChI=1S/C14H20N6/c1-3-9-6-11-12(17-7-9)13(19-14(15)18-11)20-5-4-10(8-20)16-2/h6-7,10,16H,3-5,8H2,1-2H3,(H2,15,18,19)/t10-/m1/s1 | KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| 138 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Griffin Discoveries BV
Curated by ChEMBL
| Assay Description Binding affinity to rat histamine H4 receptor |
Bioorg Med Chem Lett 23: 2663-70 (2013)
Article DOI: 10.1016/j.bmcl.2013.02.091 BindingDB Entry DOI: 10.7270/Q2K35W11 |
More data for this Ligand-Target Pair | |
Histamine H2 Receptor
(Homo sapiens (Human)) | BDBM50433356
(CHEMBL2376801)Show InChI InChI=1S/C14H20N6/c1-3-9-6-11-12(17-7-9)13(19-14(15)18-11)20-5-4-10(8-20)16-2/h6-7,10,16H,3-5,8H2,1-2H3,(H2,15,18,19)/t10-/m1/s1 | Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| 3.16E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Griffin Discoveries BV
Curated by ChEMBL
| Assay Description Displacement of [3H]histamine from human histamine H2 receptor expressed in HEK cells |
Bioorg Med Chem Lett 23: 2663-70 (2013)
Article DOI: 10.1016/j.bmcl.2013.02.091 BindingDB Entry DOI: 10.7270/Q2K35W11 |
More data for this Ligand-Target Pair | |
Histamine H1 receptor
(Homo sapiens (Human)) | BDBM50433356
(CHEMBL2376801)Show InChI InChI=1S/C14H20N6/c1-3-9-6-11-12(17-7-9)13(19-14(15)18-11)20-5-4-10(8-20)16-2/h6-7,10,16H,3-5,8H2,1-2H3,(H2,15,18,19)/t10-/m1/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| 1.12E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Griffin Discoveries BV
Curated by ChEMBL
| Assay Description Displacement of [3H]histamine from human histamine H1 receptor expressed in HEK cells |
Bioorg Med Chem Lett 23: 2663-70 (2013)
Article DOI: 10.1016/j.bmcl.2013.02.091 BindingDB Entry DOI: 10.7270/Q2K35W11 |
More data for this Ligand-Target Pair | |