BindingDB PrimarySearch

BDBM81962 S-L-365,260

SMILES: CN1c2ccccc2C(=N[C@@H](NC(=O)Nc2cccc(C)c2)C1=O)c1ccccc1

InChI Key: InChIKey=KDFQABSFVYLGPM-QFIPXVFZSA-N

Data: 16 KI 27 IC50 1 Kd

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 44 hits for monomerid = 81962
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Cholecystokinin receptor (RAT)	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	Article PubMed	0.148	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Glaxo Wellcome Medicines Research Centre Curated by ChEMBL					Assay Description Inhibition by displacing [3H]CCK-8S against Cholecystokinin type A receptor of rat pancreatic membranes				J Med Chem 43: 3596-613 (2000) Article DOI: 10.1021/jm990967h BindingDB Entry DOI: 10.7270/Q26H4M5V
Glaxo Wellcome Medicines Research Centre Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin receptor (Homo sapiens (Human))	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	Article PubMed	1.60	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Glaxo Wellcome Medicines Research Centre Curated by ChEMBL					Assay Description Inhibition by displacing [3H]CCK-8S against human Cholecystokinin type B receptor				J Med Chem 43: 3596-613 (2000) Article DOI: 10.1021/jm990967h BindingDB Entry DOI: 10.7270/Q26H4M5V
Glaxo Wellcome Medicines Research Centre Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin receptor (Homo sapiens (Human))	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	Article	1.80	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description The compound was evaluated for the inhibition of binding of [3H]-PD 140376 to Cholecystokinin type B receptor in guinea pig cortex.				Bioorg Med Chem Lett 3: 885-888 (1993) Article DOI: 10.1016/S0960-894X(00)80686-1 BindingDB Entry DOI: 10.7270/Q2D79BWZ
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin receptor (Homo sapiens (Human))	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	Article PubMed	2	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
INSERM Curated by ChEMBL					Assay Description Compound was tested for the affinity against Cholecystokinin type B receptor on guinea pig cortex.				J Med Chem 40: 3947-56 (1998) Article DOI: 10.1021/jm970439a BindingDB Entry DOI: 10.7270/Q27H1K8Z
INSERM Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin receptor (Homo sapiens (Human))	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	PubMed	2.20	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
INSERM Curated by ChEMBL					Assay Description Displacement of [3H]pCCK-8 from cholecystokinin type B receptor in guinea pig brain membrane				J Med Chem 36: 166-72 (1993) BindingDB Entry DOI: 10.7270/Q26M37FJ
INSERM Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin B (GUINEA PIG)	BDBM81962 (S-L-365,260) Show SMILES Show InChI	Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	Article PubMed	3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Merck Sharp & Dohme Research Laboratories Curated by PDSP K_i Database									Eur J Pharmacol 162: 273-80 (1989) Article DOI: 10.1016/0014-2999(89)90290-2 BindingDB Entry DOI: 10.7270/Q2QF8RB7
					More data for this Ligand-Target Pair
Cholecystokinin receptor (Homo sapiens (Human))	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	Article PubMed	3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Glaxo Wellcome Medicines Research Centre Curated by ChEMBL					Assay Description Inhibition by displacing [3H]CCK-8S against Cholecystokinin type B receptor of guinea pig				J Med Chem 43: 3596-613 (2000) Article DOI: 10.1021/jm990967h BindingDB Entry DOI: 10.7270/Q26H4M5V
Glaxo Wellcome Medicines Research Centre Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin receptor (MOUSE)	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	Article PubMed	3.70	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
James Black Foundation Curated by ChEMBL					Assay Description Tested for its receptor affinity from competition with 20 pM [125I]BH-CCK-8S for Cholecystokinin type B receptor binding sites in mouse cortical homo...				J Med Chem 37: 3671-3 (1994) Article DOI: 10.1021/jm00048a001 BindingDB Entry DOI: 10.7270/Q28918MZ
James Black Foundation Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin receptor (MOUSE)	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	Article PubMed	4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
James Black Foundation Curated by ChEMBL					Assay Description Displacement of binding of [125I]CCK-8S to Cholecystokinin type B receptor in mouse cerebral cortex homogenates				J Med Chem 43: 3518-29 (2000) Article DOI: 10.1021/jm000960w BindingDB Entry DOI: 10.7270/Q2KS6V9G
James Black Foundation Curated by ChEMBL					More data for this Ligand-Target Pair
CCKBR (RAT)	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	PubMed	12	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
INSERM Curated by ChEMBL					Assay Description Affinity of compound on binding of [3H]pCCK-8 to the cholecystokinin type B receptor in rat brain membrane				J Med Chem 36: 166-72 (1993) BindingDB Entry DOI: 10.7270/Q26M37FJ
INSERM Curated by ChEMBL					More data for this Ligand-Target Pair
CCKBR (RAT)	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	Article PubMed	15	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
INSERM Curated by ChEMBL					Assay Description Compound was tested for binding affinity against rat brain Cholecystokinin type B receptor expressed in CHO cells.				J Med Chem 40: 3947-56 (1998) Article DOI: 10.1021/jm970439a BindingDB Entry DOI: 10.7270/Q27H1K8Z
INSERM Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin B (GUINEA PIG)	BDBM81962 (S-L-365,260) Show SMILES Show InChI	Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	Article PubMed	130	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Merck Sharp & Dohme Research Laboratories Curated by PDSP K_i Database									Eur J Pharmacol 162: 273-80 (1989) Article DOI: 10.1016/0014-2999(89)90290-2 BindingDB Entry DOI: 10.7270/Q2QF8RB7
					More data for this Ligand-Target Pair
Cholecystokinin B (GUINEA PIG)	BDBM81962 (S-L-365,260) Show SMILES Show InChI	Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	Article PubMed	151	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Merck Sharp & Dohme Research Laboratories Curated by PDSP K_i Database									Eur J Pharmacol 162: 273-80 (1989) Article DOI: 10.1016/0014-2999(89)90290-2 BindingDB Entry DOI: 10.7270/Q2QF8RB7
					More data for this Ligand-Target Pair
Cholecystokinin receptor (RAT)	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	Article PubMed	269	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Glaxo Wellcome Medicines Research Centre Curated by ChEMBL					Assay Description Inhibition by displacing [3H]CCK-8S against Cholecystokinin type B receptor of rat pancreatic membranes				J Med Chem 43: 3596-613 (2000) Article DOI: 10.1021/jm990967h BindingDB Entry DOI: 10.7270/Q26H4M5V
Glaxo Wellcome Medicines Research Centre Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin A receptor (Cavia porcellus)	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	Article PubMed	316	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
James Black Foundation Curated by ChEMBL					Assay Description Displacement of [125I]BH-CCK-8S from CC1 receptor expressed in guinea pig pancreatic cells				J Med Chem 51: 565-73 (2008) Article DOI: 10.1021/jm070880t BindingDB Entry DOI: 10.7270/Q2TF014R
James Black Foundation Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin A receptor (Cavia porcellus)	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	Article PubMed	468	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
James Black Foundation Curated by ChEMBL					Assay Description Tested for its receptor affinity from competition with 20 pM [125I]BH-CCK-8S for Cholecystokinin type A receptor binding sites on guinea pig-pancreat...				J Med Chem 37: 3671-3 (1994) Article DOI: 10.1021/jm00048a001 BindingDB Entry DOI: 10.7270/Q28918MZ
James Black Foundation Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin receptor (RAT)	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	PubMed	n/a	n/a	280	n/a	n/a	n/a	n/a	n/a	n/a
Merck Sharp& Dohme Research Laboratories Curated by ChEMBL					Assay Description Inhibition of binding of [125I]- CCK-33 to rat pancreas				J Med Chem 33: 591-5 (1990) BindingDB Entry DOI: 10.7270/Q29K4BTP
Merck Sharp& Dohme Research Laboratories Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin receptor (Homo sapiens (Human))	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	PubMed	n/a	n/a	1.10	n/a	n/a	n/a	n/a	n/a	n/a
Merck Sharp& Dohme Research Laboratories Curated by ChEMBL					Assay Description Inhibition of binding of [125I]gastrin to Cholecystokinin type B receptor from guinea pig gastric glands				J Med Chem 33: 591-5 (1990) BindingDB Entry DOI: 10.7270/Q29K4BTP
Merck Sharp& Dohme Research Laboratories Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin receptor (RAT)	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	PubMed	n/a	n/a	230	n/a	n/a	n/a	n/a	n/a	n/a
Parke-Davis Neuroscience Research Centre Curated by ChEMBL					Assay Description Evaluated for inhibition of cholecystokinin type A receptor by displacing [125I]bolton hunter CCK-8 radioligand in the rat pancreas				J Med Chem 35: 2573-81 (1992) BindingDB Entry DOI: 10.7270/Q2TT4RJ4
Parke-Davis Neuroscience Research Centre Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin receptor (MOUSE)	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	PubMed	n/a	n/a	5.10	n/a	n/a	n/a	n/a	n/a	n/a
Parke-Davis Neuroscience Research Centre Curated by ChEMBL					Assay Description Evaluated for inhibition of cholecystokinin type B receptor by displacing [125I]-Bolton hunter CCK-8 radioligand in the mouse cerebral cortex				J Med Chem 35: 2573-81 (1992) BindingDB Entry DOI: 10.7270/Q2TT4RJ4
Parke-Davis Neuroscience Research Centre Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin receptor (RAT)	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	PubMed	n/a	n/a	230	n/a	n/a	n/a	n/a	n/a	n/a
Parke-Davis Research Unit Curated by ChEMBL					Assay Description Half-maximal inhibition of specific binding of [125I]bolton hunter CCK-8 to rat pancreas cholecystokinin type A receptor				J Med Chem 34: 404-14 (1991) BindingDB Entry DOI: 10.7270/Q2RJ4K3V
Parke-Davis Research Unit Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin receptor (MOUSE)	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	PubMed	n/a	n/a	5.10	n/a	n/a	n/a	n/a	n/a	n/a
Parke-Davis Research Unit Curated by ChEMBL					Assay Description Half-maximal inhibition of specific binding of [125I]bolton hunter CCK-8 to mouse cerebral cortex cholecystokinin type B receptor				J Med Chem 34: 404-14 (1991) BindingDB Entry DOI: 10.7270/Q2RJ4K3V
Parke-Davis Research Unit Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin receptor (Homo sapiens (Human))	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	PubMed	n/a	n/a	8.5	n/a	n/a	n/a	n/a	n/a	n/a
Merck, Sharp and Dohme Research Laboratories Curated by ChEMBL					Assay Description Binding activity against Cholecystokinin type B receptor from guinea pig cortex using [125]BH CCK-8s as radioligand.				J Med Chem 37: 719-21 (1994) BindingDB Entry DOI: 10.7270/Q2QN67FP
					More data for this Ligand-Target Pair
Cholecystokinin receptor (RAT)	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	PubMed	n/a	n/a	736	n/a	n/a	n/a	n/a	n/a	n/a
Merck, Sharp and Dohme Research Laboratories Curated by ChEMBL					Assay Description Binding activity against Cholecystokinin type A receptor from rat pancreas using [125]BH CCK-8s as radioligand.				J Med Chem 37: 719-21 (1994) BindingDB Entry DOI: 10.7270/Q2QN67FP
					More data for this Ligand-Target Pair
CCKBR (RAT)	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	39	n/a	n/a	n/a	n/a	n/a	n/a
INSERM Curated by ChEMBL					Assay Description Inhibition of inositol phosphate production induced by Cholecystokinin type B receptor (0.5 nM)				J Med Chem 40: 3947-56 (1998) Article DOI: 10.1021/jm970439a BindingDB Entry DOI: 10.7270/Q27H1K8Z
INSERM Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin receptor (MOUSE)	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	PubMed	n/a	n/a	2	n/a	n/a	n/a	n/a	n/a	n/a
James Black Foundation Curated by ChEMBL					Assay Description Half maximal inhibition of specific binding of [125I]Bolton-Hunter CCK-8 to Cholecystokinin type B receptor in the mouse cerebral cortex				J Med Chem 43: 3505-17 (2000) BindingDB Entry DOI: 10.7270/Q2FQ9XBZ
James Black Foundation Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin receptor (RAT)	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	PubMed	n/a	n/a	280	n/a	n/a	n/a	n/a	n/a	n/a
James Black Foundation Curated by ChEMBL					Assay Description Half maximal inhibition of specific binding of [125I]-Bolton-Hunter CCK-8 to Cholecystokinin type A receptor in the rat pancreas				J Med Chem 43: 3505-17 (2000) BindingDB Entry DOI: 10.7270/Q2FQ9XBZ
James Black Foundation Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin receptor (Homo sapiens (Human))	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	PubMed	n/a	n/a	2	n/a	n/a	n/a	n/a	n/a	n/a
Merck Research Laboratories Curated by ChEMBL					Assay Description Inhibition of Cholecystokinin type B receptor induced guinea pig gall bladder contractions when given intravenously				J Med Chem 45: 5609-16 (2002) BindingDB Entry DOI: 10.7270/Q270825W
Merck Research Laboratories Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin receptor (RAT)	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	PubMed	n/a	n/a	280	n/a	n/a	n/a	n/a	n/a	n/a
Merck Research Laboratories Curated by ChEMBL					Assay Description Concentration required for 50% inhibition of Cholecystokinin type A receptor in rat pancreatic tissue				J Med Chem 45: 5609-16 (2002) BindingDB Entry DOI: 10.7270/Q270825W
Merck Research Laboratories Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human))	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	5.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
China Pharmaceutical University Curated by ChEMBL					Assay Description Inhibitory concentration against IKr potassium channel				Bioorg Med Chem Lett 14: 4771-7 (2004) Article DOI: 10.1016/j.bmcl.2004.06.070 BindingDB Entry DOI: 10.7270/Q208661K
China Pharmaceutical University Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin receptor (Homo sapiens (Human))	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	4	n/a	n/a	n/a	n/a	n/a	n/a
Organon Laboratories Curated by ChEMBL					Assay Description Inhibitory concentration against gastrin receptor				J Med Chem 48: 6523-43 (2005) Article DOI: 10.1021/jm058225d BindingDB Entry DOI: 10.7270/Q2SF2WZ9
Organon Laboratories Curated by ChEMBL					More data for this Ligand-Target Pair
CCKBR (RAT)	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	n/a	28.8	n/a	n/a	n/a	n/a	n/a
James Black Foundation Curated by ChEMBL					Assay Description Affinity for CCK2 receptor assessed by inhibition of pentagastrin-stimulated acid secretion in perfused rat stomach				J Med Chem 49: 2253-61 (2006) Article DOI: 10.1021/jm051219x BindingDB Entry DOI: 10.7270/Q28K7B8B
James Black Foundation Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin receptor (Homo sapiens (Human))	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	PubMed	n/a	n/a	1.10	n/a	n/a	n/a	n/a	n/a	n/a
Merck Sharp& Dohme Research Laboratories Curated by ChEMBL					Assay Description Displacement of 125 I-gastrin from gastrin receptor of guinea pig gastric glands				J Med Chem 32: 13-6 (1989) BindingDB Entry DOI: 10.7270/Q2MC90MG
Merck Sharp& Dohme Research Laboratories Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin receptor (Homo sapiens (Human))	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	PubMed	n/a	n/a	6.30	n/a	n/a	n/a	n/a	n/a	n/a
Glaxo Research Institute Curated by ChEMBL					Assay Description Displacement of CCK-8 from human Cholecystokinin type B receptor expressing CHO cell membranes				J Med Chem 38: 207-11 (1995) BindingDB Entry DOI: 10.7270/Q28C9XF9
Glaxo Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin receptor (Homo sapiens (Human))	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	PubMed	n/a	n/a	2	n/a	n/a	n/a	n/a	n/a	n/a
Merck Research Laboratories Curated by ChEMBL					Assay Description Antagonistic activity against cholecystokinin type B receptor				J Med Chem 36: 2051-8 (1993) BindingDB Entry DOI: 10.7270/Q2NP2524
Merck Research Laboratories Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin receptor (Homo sapiens (Human))	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	PubMed	n/a	n/a	2	n/a	n/a	n/a	n/a	n/a	n/a
Merck Sharp& Dohme Research Laboratories Curated by ChEMBL					Assay Description Displacement of [125 I] CCK-8 from Cholecystokinin type B receptor of guinea pig cerebral cortex				J Med Chem 32: 13-6 (1989) BindingDB Entry DOI: 10.7270/Q2MC90MG
Merck Sharp& Dohme Research Laboratories Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin receptor (RAT)	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	PubMed	n/a	n/a	230	n/a	n/a	n/a	n/a	n/a	n/a
Parke-Davis Neuroscience Research Centre Curated by ChEMBL					Assay Description Inhibition of binding of [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type A receptor in the rat pancreas.				J Med Chem 36: 552-65 (1993) BindingDB Entry DOI: 10.7270/Q2JM2B88
Parke-Davis Neuroscience Research Centre Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin receptor (MOUSE)	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	PubMed	n/a	n/a	5.10	n/a	n/a	n/a	n/a	n/a	n/a
Parke-Davis Neuroscience Research Centre Curated by ChEMBL					Assay Description Inhibition of binding of [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortex				J Med Chem 36: 552-65 (1993) BindingDB Entry DOI: 10.7270/Q2JM2B88
Parke-Davis Neuroscience Research Centre Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin receptor (RAT)	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	PubMed	n/a	n/a	740	n/a	n/a	n/a	n/a	n/a	n/a
Merck Research Laboratories Curated by ChEMBL					Assay Description Inhibition of binding of [125I]CCK-8 to cholecystokinin type A receptor in rat pancreatic tissue				J Med Chem 36: 4276-92 (1994) BindingDB Entry DOI: 10.7270/Q22J6CH9
Merck Research Laboratories Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin receptor (RAT)	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	PubMed	n/a	n/a	280	n/a	n/a	n/a	n/a	n/a	n/a
Merck Sharp& Dohme Research Laboratories Curated by ChEMBL					Assay Description Displacement of [125 I] CCK-8 from Cholecystokinin type A receptor of rat pancreas				J Med Chem 32: 13-6 (1989) BindingDB Entry DOI: 10.7270/Q2MC90MG
Merck Sharp& Dohme Research Laboratories Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin receptor (Homo sapiens (Human))	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	PubMed	n/a	n/a	8.5	n/a	n/a	n/a	n/a	n/a	n/a
Merck Research Laboratories Curated by ChEMBL					Assay Description Inhibition of binding of [125I]-CCK-8 to the cholecystokinin type B receptor				J Med Chem 36: 4276-92 (1994) BindingDB Entry DOI: 10.7270/Q22J6CH9
Merck Research Laboratories Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin A receptor (Cavia porcellus)	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	PubMed	n/a	n/a	2	n/a	n/a	n/a	n/a	n/a	n/a
Merck Sharp& Dohme Research Laboratories Curated by ChEMBL					Assay Description Inhibition of binding of [125I]- CCK-33 to guinea pig cortex				J Med Chem 33: 591-5 (1990) BindingDB Entry DOI: 10.7270/Q29K4BTP
Merck Sharp& Dohme Research Laboratories Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin receptor (Homo sapiens (Human))	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	PubMed	n/a	n/a	158	n/a	n/a	n/a	n/a	n/a	n/a
Glaxo Research Institute Curated by ChEMBL					Assay Description Displacement of CCK-8 from CHO cell membranes expressing human Cholecystokinin type A receptor				J Med Chem 38: 207-11 (1995) BindingDB Entry DOI: 10.7270/Q28C9XF9
Glaxo Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin receptor (Homo sapiens (Human))	BDBM81962 (S-L-365,260) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	29	n/a	n/a	n/a	n/a	n/a	n/a
Organon Laboratories Curated by ChEMBL					Assay Description Inhibitory concentration against Cholecystokinin B receptor				J Med Chem 48: 6523-43 (2005) Article DOI: 10.1021/jm058225d BindingDB Entry DOI: 10.7270/Q2SF2WZ9
Organon Laboratories Curated by ChEMBL					More data for this Ligand-Target Pair