BDBM82006 D-AP4::D-APB::US9212196, L-AP4
SMILES: N[C@H](CCP(O)(O)=O)C(O)=O
InChI Key: InChIKey=DDOQBQRIEWHWBT-GSVOUGTGSA-N
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
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Glutamate receptor ionotropic, NMDA 1 (RAT) | BDBM82006 (D-AP4 | D-APB | US9212196, L-AP4) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Patents Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Minnesota Curated by PDSP Ki Database | Biochemistry 24: 2401-5 (1985) Article DOI: 10.1021/bi00331a002 BindingDB Entry DOI: 10.7270/Q2W094FK | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 8 (mGlu8) (Rattus norvegicus (Rat)) | BDBM82006 (D-AP4 | D-APB | US9212196, L-AP4) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Patents Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Toronto Curated by PDSP Ki Database | Neuropharmacology 40: 170-7 (2001) Article DOI: 10.1016/s0028-3908(00)00128-3 BindingDB Entry DOI: 10.7270/Q27P8WZ1 | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 7 (mGlu7) (Rattus norvegicus (Rat)) | BDBM82006 (D-AP4 | D-APB | US9212196, L-AP4) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a |
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE US Patent | Assay Description Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ... | US Patent US9212196 (2015) BindingDB Entry DOI: 10.7270/Q28G8JJR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 6 (mGlu6) (Rattus norvegicus (Rat)) | BDBM82006 (D-AP4 | D-APB | US9212196, L-AP4) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | n/a | n/a | 1.03E+3 | n/a | n/a | n/a | n/a |
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE US Patent | Assay Description Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ... | US Patent US9212196 (2015) BindingDB Entry DOI: 10.7270/Q28G8JJR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 8 (mGlu8) (Rattus norvegicus (Rat)) | BDBM82006 (D-AP4 | D-APB | US9212196, L-AP4) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | n/a | n/a | 290 | n/a | n/a | n/a | n/a |
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE US Patent | Assay Description Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ... | US Patent US9212196 (2015) BindingDB Entry DOI: 10.7270/Q28G8JJR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 4 (mGlu4) (Rattus norvegicus (Rat)) | BDBM82006 (D-AP4 | D-APB | US9212196, L-AP4) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | n/a | n/a | 130 | n/a | n/a | n/a | n/a |
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE US Patent | Assay Description Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ... | US Patent US9212196 (2015) BindingDB Entry DOI: 10.7270/Q28G8JJR | |||||||||||
More data for this Ligand-Target Pair |