Through the "gatekeeper door": exploiting the active kinase conformation

J Med Chem. 2010 Apr 8;53(7):2681-94. doi: 10.1021/jm901443h.
No abstract available

Publication types

  • Review

MeSH terms

  • Drug Design
  • Humans
  • Protein Kinase Inhibitors / chemistry
  • Protein Kinase Inhibitors / pharmacology
  • Protein Kinases / chemistry*
  • Protein Kinases / metabolism*
  • Substrate Specificity

Substances

  • Protein Kinase Inhibitors
  • Protein Kinases