Bradykinin B1 receptor antagonists as potential therapeutic agents for pain

J Med Chem. 2010 Aug 12;53(15):5383-99. doi: 10.1021/jm1000776.
No abstract available

MeSH terms

  • Amides / chemistry
  • Amides / pharmacology
  • Amides / therapeutic use
  • Analgesics / chemistry*
  • Analgesics / pharmacology
  • Analgesics / therapeutic use
  • Animals
  • Bradykinin B1 Receptor Antagonists*
  • Clinical Trials as Topic
  • Drug Evaluation, Preclinical
  • Humans
  • Models, Molecular
  • Pain / drug therapy*
  • Receptor, Bradykinin B1 / physiology
  • Sulfonamides / chemistry
  • Sulfonamides / pharmacology
  • Sulfonamides / therapeutic use

Substances

  • Amides
  • Analgesics
  • Bradykinin B1 Receptor Antagonists
  • Receptor, Bradykinin B1
  • Sulfonamides