Novel selective thiol inhibitors of neutral endopeptidase containing heterocycles at P'2 position

J Enzyme Inhib. 1997 Jun;12(2):155-60. doi: 10.3109/14756369709035816.
No abstract available

MeSH terms

  • Atrial Natriuretic Factor / metabolism
  • Models, Chemical
  • Neprilysin / antagonists & inhibitors*
  • Neprilysin / chemistry
  • Peptidyl-Dipeptidase A / metabolism
  • Protease Inhibitors / pharmacology*
  • Structure-Activity Relationship
  • Thiorphan / analogs & derivatives*
  • Thiorphan / pharmacology

Substances

  • Protease Inhibitors
  • Atrial Natriuretic Factor
  • Thiorphan
  • Peptidyl-Dipeptidase A
  • Neprilysin