Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50010698 ((-)6-Methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]qu...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 0.380 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Debrecen Curated by ChEMBL | Assay Description Displacement of [3H]raclopride from dopamine D2 receptor in rat striatal membrane | Bioorg Med Chem 16: 4563-8 (2008) Article DOI: 10.1016/j.bmc.2008.02.038 BindingDB Entry DOI: 10.7270/Q24J0DW0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50016786 ((R)-2-Fluoro-6-methyl-5,6,6a,7-tetrahydro-4H-diben...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.430 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Debrecen Curated by ChEMBL | Assay Description Displacement of [3H]raclopride from dopamine D2 receptor in rat striatal membrane | Bioorg Med Chem 16: 4563-8 (2008) Article DOI: 10.1016/j.bmc.2008.02.038 BindingDB Entry DOI: 10.7270/Q24J0DW0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50010697 ((R)-(-)-2-methoxyapomorphine | (R)-2-Methoxy-6-met...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.12 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Debrecen Curated by ChEMBL | Assay Description Displacement of [3H]raclopride from dopamine D2 receptor in rat striatal membrane | Bioorg Med Chem 16: 4563-8 (2008) Article DOI: 10.1016/j.bmc.2008.02.038 BindingDB Entry DOI: 10.7270/Q24J0DW0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50295863 (CHEMBL562935 | N-Ethyl-2-(4-hydroxyphenyl)-norapom...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tartu Curated by ChEMBL | Assay Description Displacement of [3H]raclopride from rat dopamine D2short receptor expressed in CHO-K1 cells by liquid scintillation counting | Bioorg Med Chem 17: 4756-62 (2009) Article DOI: 10.1016/j.bmc.2009.04.047 BindingDB Entry DOI: 10.7270/Q2KD1XZ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(3) dopamine receptor (Rattus norvegicus (Rat)) | BDBM50251027 ((R)-(-)-2-(4-Hydroxyphenyl)-apomorphine hydrochlor...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Debrecen Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in SF9 cells | Bioorg Med Chem 16: 3773-9 (2008) Article DOI: 10.1016/j.bmc.2008.01.057 BindingDB Entry DOI: 10.7270/Q2959HB7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50295866 (CHEMBL560721 | N-Propyl-2-(4-hydroxyphenyl)-norapo...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tartu Curated by ChEMBL | Assay Description Displacement of [3H]raclopride from rat dopamine D2short receptor expressed in CHO-K1 cells by liquid scintillation counting | Bioorg Med Chem 17: 4756-62 (2009) Article DOI: 10.1016/j.bmc.2009.04.047 BindingDB Entry DOI: 10.7270/Q2KD1XZ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Homo sapiens (Human)) | BDBM50251027 ((R)-(-)-2-(4-Hydroxyphenyl)-apomorphine hydrochlor...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Debrecen Curated by ChEMBL | Assay Description Displacement of [3H]raclopride from human cloned dopamine D2 receptor expressed in CHO cell membrane | Bioorg Med Chem 16: 4563-8 (2008) Article DOI: 10.1016/j.bmc.2008.02.038 BindingDB Entry DOI: 10.7270/Q24J0DW0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50251027 ((R)-(-)-2-(4-Hydroxyphenyl)-apomorphine hydrochlor...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Debrecen Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat dopamine D2 receptor in brain striatal membrane | Bioorg Med Chem 16: 3773-9 (2008) Article DOI: 10.1016/j.bmc.2008.01.057 BindingDB Entry DOI: 10.7270/Q2959HB7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50251027 ((R)-(-)-2-(4-Hydroxyphenyl)-apomorphine hydrochlor...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Debrecen Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat dopamine D2 receptor in brain striatal membrane | Bioorg Med Chem 16: 3773-9 (2008) Article DOI: 10.1016/j.bmc.2008.01.057 BindingDB Entry DOI: 10.7270/Q2959HB7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50251027 ((R)-(-)-2-(4-Hydroxyphenyl)-apomorphine hydrochlor...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.14 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tartu Curated by ChEMBL | Assay Description Displacement of [3H]raclopride from rat dopamine D2short receptor expressed in CHO-K1 cells by liquid scintillation counting | Bioorg Med Chem 17: 4756-62 (2009) Article DOI: 10.1016/j.bmc.2009.04.047 BindingDB Entry DOI: 10.7270/Q2KD1XZ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(3) dopamine receptor (Rattus norvegicus (Rat)) | BDBM50251026 ((R)-(-)-2-Phenyl-apomorphine hydrochloride | CHEMB...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Debrecen Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in SF9 cells | Bioorg Med Chem 16: 3773-9 (2008) Article DOI: 10.1016/j.bmc.2008.01.057 BindingDB Entry DOI: 10.7270/Q2959HB7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50295864 (CHEMBL550180 | N-Propyl-2-methylnorapomorphine hyd...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 9.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tartu Curated by ChEMBL | Assay Description Displacement of [3H]raclopride from rat dopamine D2short receptor expressed in CHO-K1 cells by liquid scintillation counting | Bioorg Med Chem 17: 4756-62 (2009) Article DOI: 10.1016/j.bmc.2009.04.047 BindingDB Entry DOI: 10.7270/Q2KD1XZ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50347558 (CHEMBL1802233) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 9.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tartu Curated by ChEMBL | Assay Description Displacement of [3H]raclopride from rat D2 dopamine receptor expressed in CHOK1 cells after 90 mins by liquid scintillation counter scintillation cou... | Eur J Med Chem 46: 2992-9 (2011) Article DOI: 10.1016/j.ejmech.2011.04.028 BindingDB Entry DOI: 10.7270/Q2X34XTG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50347560 (CHEMBL1802235) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tartu Curated by ChEMBL | Assay Description Displacement of [3H]raclopride from rat D2 dopamine receptor expressed in CHOK1 cells after 90 mins by liquid scintillation counter scintillation cou... | Eur J Med Chem 46: 2992-9 (2011) Article DOI: 10.1016/j.ejmech.2011.04.028 BindingDB Entry DOI: 10.7270/Q2X34XTG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50001955 ((-)6-Methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]qu...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 11.1 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Debrecen Curated by ChEMBL | Assay Description Displacement of [3H]raclopride from dopamine D2 receptor in rat striatal membrane | Bioorg Med Chem 16: 4563-8 (2008) Article DOI: 10.1016/j.bmc.2008.02.038 BindingDB Entry DOI: 10.7270/Q24J0DW0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50001955 ((-)6-Methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]qu...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 11.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tartu Curated by ChEMBL | Assay Description Displacement of [3H]raclopride from rat D2 dopamine receptor expressed in CHOK1 cells after 90 mins by liquid scintillation counter scintillation cou... | Eur J Med Chem 46: 2992-9 (2011) Article DOI: 10.1016/j.ejmech.2011.04.028 BindingDB Entry DOI: 10.7270/Q2X34XTG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50001955 ((-)6-Methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]qu...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 11.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tartu Curated by ChEMBL | Assay Description Displacement of [3H]raclopride from rat dopamine D2short receptor expressed in CHO-K1 cells by liquid scintillation counting | Bioorg Med Chem 17: 4756-62 (2009) Article DOI: 10.1016/j.bmc.2009.04.047 BindingDB Entry DOI: 10.7270/Q2KD1XZ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50251026 ((R)-(-)-2-Phenyl-apomorphine hydrochloride | CHEMB...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 11.7 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tartu Curated by ChEMBL | Assay Description Displacement of [3H]raclopride from rat dopamine D2short receptor expressed in CHO-K1 cells by liquid scintillation counting | Bioorg Med Chem 17: 4756-62 (2009) Article DOI: 10.1016/j.bmc.2009.04.047 BindingDB Entry DOI: 10.7270/Q2KD1XZ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50251026 ((R)-(-)-2-Phenyl-apomorphine hydrochloride | CHEMB...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 12 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Debrecen Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat dopamine D2 receptor in brain striatal membrane | Bioorg Med Chem 16: 3773-9 (2008) Article DOI: 10.1016/j.bmc.2008.01.057 BindingDB Entry DOI: 10.7270/Q2959HB7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50295862 (CHEMBL564909 | N-Ethyl-2-phenylnorapomorphine hydr...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 14 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tartu Curated by ChEMBL | Assay Description Displacement of [3H]raclopride from rat dopamine D2short receptor expressed in CHO-K1 cells by liquid scintillation counting | Bioorg Med Chem 17: 4756-62 (2009) Article DOI: 10.1016/j.bmc.2009.04.047 BindingDB Entry DOI: 10.7270/Q2KD1XZ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50010696 ((R)-2-Bromo-6-methyl-5,6,6a,7-tetrahydro-4H-dibenz...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 17.7 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Debrecen Curated by ChEMBL | Assay Description Displacement of [3H]raclopride from dopamine D2 receptor in rat striatal membrane | Bioorg Med Chem 16: 4563-8 (2008) Article DOI: 10.1016/j.bmc.2008.02.038 BindingDB Entry DOI: 10.7270/Q24J0DW0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50016785 ((R)-2-Amino-6-methyl-5,6,6a,7-tetrahydro-4H-dibenz...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 19.9 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Debrecen Curated by ChEMBL | Assay Description Displacement of [3H]raclopride from dopamine D2 receptor in rat striatal membrane | Bioorg Med Chem 16: 4563-8 (2008) Article DOI: 10.1016/j.bmc.2008.02.038 BindingDB Entry DOI: 10.7270/Q24J0DW0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50251028 ((R)-(-)-2-Methyl-apomorphine hydrochloride | CHEMB...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 20.7 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tartu Curated by ChEMBL | Assay Description Displacement of [3H]raclopride from rat dopamine D2short receptor expressed in CHO-K1 cells by liquid scintillation counting | Bioorg Med Chem 17: 4756-62 (2009) Article DOI: 10.1016/j.bmc.2009.04.047 BindingDB Entry DOI: 10.7270/Q2KD1XZ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50251028 ((R)-(-)-2-Methyl-apomorphine hydrochloride | CHEMB...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 21 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Debrecen Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat dopamine D2 receptor in brain striatal membrane | Bioorg Med Chem 16: 3773-9 (2008) Article DOI: 10.1016/j.bmc.2008.01.057 BindingDB Entry DOI: 10.7270/Q2959HB7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(3) dopamine receptor (Rattus norvegicus (Rat)) | BDBM50251034 ((R)-(-)-2-(4-dibenzo-furanyl)-apomorphine hydrochl...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 22 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Debrecen Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in SF9 cells | Bioorg Med Chem 16: 3773-9 (2008) Article DOI: 10.1016/j.bmc.2008.01.057 BindingDB Entry DOI: 10.7270/Q2959HB7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(3) dopamine receptor (Rattus norvegicus (Rat)) | BDBM50251034 ((R)-(-)-2-(4-dibenzo-furanyl)-apomorphine hydrochl...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 22 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Debrecen Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in SF9 cells | Bioorg Med Chem 16: 3773-9 (2008) Article DOI: 10.1016/j.bmc.2008.01.057 BindingDB Entry DOI: 10.7270/Q2959HB7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(1A) dopamine receptor (Homo sapiens (Human)) | BDBM50295862 (CHEMBL564909 | N-Ethyl-2-phenylnorapomorphine hydr...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 31 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tartu Curated by ChEMBL | Assay Description Displacement of [3H]SCH23390 from dopamine D1 receptor expressed in Ltk deficient fibroblast cells by liquid scintillation counting | Bioorg Med Chem 17: 4756-62 (2009) Article DOI: 10.1016/j.bmc.2009.04.047 BindingDB Entry DOI: 10.7270/Q2KD1XZ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50001955 ((-)6-Methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]qu...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 32 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Debrecen Curated by ChEMBL | Assay Description Displacement of [3H]raclopride from rat dopamine D2(short) receptor expressed in CHOK1 cells | Bioorg Med Chem 16: 4563-8 (2008) Article DOI: 10.1016/j.bmc.2008.02.038 BindingDB Entry DOI: 10.7270/Q24J0DW0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Homo sapiens (Human)) | BDBM50001955 ((-)6-Methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]qu...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank PC cid PC sid PDB UniChem Patents Similars | DrugBank Article PubMed | 32 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Debrecen Curated by ChEMBL | Assay Description Displacement of [3H]raclopride from human cloned dopamine D2 receptor expressed in CHO cell membrane | Bioorg Med Chem 16: 4563-8 (2008) Article DOI: 10.1016/j.bmc.2008.02.038 BindingDB Entry DOI: 10.7270/Q24J0DW0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(3) dopamine receptor (Rattus norvegicus (Rat)) | BDBM29644 ((6aR)-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase DrugBank PC cid PC sid PDB UniChem Similars | Article PubMed | 36 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Debrecen Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in SF9 cells | Bioorg Med Chem 16: 3773-9 (2008) Article DOI: 10.1016/j.bmc.2008.01.057 BindingDB Entry DOI: 10.7270/Q2959HB7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(3) dopamine receptor (Rattus norvegicus (Rat)) | BDBM29644 ((6aR)-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase DrugBank PC cid PC sid PDB UniChem Similars | Article PubMed | 36 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Debrecen Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in SF9 cells | Bioorg Med Chem 16: 3773-9 (2008) Article DOI: 10.1016/j.bmc.2008.01.057 BindingDB Entry DOI: 10.7270/Q2959HB7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(3) dopamine receptor (Rattus norvegicus (Rat)) | BDBM50251028 ((R)-(-)-2-Methyl-apomorphine hydrochloride | CHEMB...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Debrecen Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in SF9 cells | Bioorg Med Chem 16: 3773-9 (2008) Article DOI: 10.1016/j.bmc.2008.01.057 BindingDB Entry DOI: 10.7270/Q2959HB7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(3) dopamine receptor (Rattus norvegicus (Rat)) | BDBM50251028 ((R)-(-)-2-Methyl-apomorphine hydrochloride | CHEMB...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Debrecen Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in SF9 cells | Bioorg Med Chem 16: 3773-9 (2008) Article DOI: 10.1016/j.bmc.2008.01.057 BindingDB Entry DOI: 10.7270/Q2959HB7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50251320 ((R)-2-Ethoxy-6-methyl-5,6,6a,7-tetrahydro-4H-diben...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 44 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Debrecen Curated by ChEMBL | Assay Description Displacement of [3H]raclopride from rat dopamine D2(short) receptor expressed in CHOK1 cells | Bioorg Med Chem 16: 4563-8 (2008) Article DOI: 10.1016/j.bmc.2008.02.038 BindingDB Entry DOI: 10.7270/Q24J0DW0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM29644 ((6aR)-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase DrugBank PC cid PC sid PDB UniChem Similars | Article PubMed | 48 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Debrecen Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat dopamine D2 receptor in brain striatal membrane | Bioorg Med Chem 16: 3773-9 (2008) Article DOI: 10.1016/j.bmc.2008.01.057 BindingDB Entry DOI: 10.7270/Q2959HB7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50251314 ((R)-6-Methyl-2-methylsulfanyl-5,6,6a,7-tetrahydro-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 54.7 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Debrecen Curated by ChEMBL | Assay Description Displacement of [3H]raclopride from dopamine D2 receptor in rat striatal membrane | Bioorg Med Chem 16: 4563-8 (2008) Article DOI: 10.1016/j.bmc.2008.02.038 BindingDB Entry DOI: 10.7270/Q24J0DW0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50347557 (CHEMBL1802232) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 55 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tartu Curated by ChEMBL | Assay Description Displacement of [3H]raclopride from rat D2 dopamine receptor expressed in CHOK1 cells after 90 mins by liquid scintillation counter scintillation cou... | Eur J Med Chem 46: 2992-9 (2011) Article DOI: 10.1016/j.ejmech.2011.04.028 BindingDB Entry DOI: 10.7270/Q2X34XTG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50251327 ((R)-2-Butoxy-6-methyl-5,6,6a,7-tetrahydro-4H-diben...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Debrecen Curated by ChEMBL | Assay Description Displacement of [3H]raclopride from rat dopamine D2(short) receptor expressed in CHOK1 cells | Bioorg Med Chem 16: 4563-8 (2008) Article DOI: 10.1016/j.bmc.2008.02.038 BindingDB Entry DOI: 10.7270/Q24J0DW0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(1A) dopamine receptor (Homo sapiens (Human)) | BDBM50001955 ((-)6-Methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]qu...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank PC cid PC sid PDB UniChem Patents Similars | DrugBank PDB Article PubMed | 72 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tartu Curated by ChEMBL | Assay Description Displacement of [3H]SCH23390 from human D1 dopamine receptor expressed in Ltk fibroblast cells after 60 mins by liquid scintillation counter | Eur J Med Chem 46: 2992-9 (2011) Article DOI: 10.1016/j.ejmech.2011.04.028 BindingDB Entry DOI: 10.7270/Q2X34XTG | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
D(1A) dopamine receptor (Homo sapiens (Human)) | BDBM50001955 ((-)6-Methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]qu...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank PC cid PC sid PDB UniChem Patents Similars | DrugBank PDB Article PubMed | 72 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tartu Curated by ChEMBL | Assay Description Displacement of [3H]SCH23390 from dopamine D1 receptor expressed in Ltk deficient fibroblast cells by liquid scintillation counting | Bioorg Med Chem 17: 4756-62 (2009) Article DOI: 10.1016/j.bmc.2009.04.047 BindingDB Entry DOI: 10.7270/Q2KD1XZ4 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50251321 ((R)-6-Methyl-2-propoxy-5,6,6a,7-tetrahydro-4H-dibe...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 75 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Debrecen Curated by ChEMBL | Assay Description Displacement of [3H]raclopride from rat dopamine D2(short) receptor expressed in CHOK1 cells | Bioorg Med Chem 16: 4563-8 (2008) Article DOI: 10.1016/j.bmc.2008.02.038 BindingDB Entry DOI: 10.7270/Q24J0DW0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(3) dopamine receptor (Rattus norvegicus (Rat)) | BDBM50251029 ((R)-(-)-2-(4-N,N-Dimethylaminophenyl)-apomorphine ...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 78 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Debrecen Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in SF9 cells | Bioorg Med Chem 16: 3773-9 (2008) Article DOI: 10.1016/j.bmc.2008.01.057 BindingDB Entry DOI: 10.7270/Q2959HB7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(3) dopamine receptor (Rattus norvegicus (Rat)) | BDBM50251029 ((R)-(-)-2-(4-N,N-Dimethylaminophenyl)-apomorphine ...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 78 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Debrecen Curated by ChEMBL | Assay Description Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in SF9 cells | Bioorg Med Chem 16: 3773-9 (2008) Article DOI: 10.1016/j.bmc.2008.01.057 BindingDB Entry DOI: 10.7270/Q2959HB7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Homo sapiens (Human)) | BDBM50251026 ((R)-(-)-2-Phenyl-apomorphine hydrochloride | CHEMB...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 88 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Debrecen Curated by ChEMBL | Assay Description Displacement of [3H]raclopride from human cloned dopamine D2 receptor expressed in CHO cell membrane | Bioorg Med Chem 16: 4563-8 (2008) Article DOI: 10.1016/j.bmc.2008.02.038 BindingDB Entry DOI: 10.7270/Q24J0DW0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(1A) dopamine receptor (Homo sapiens (Human)) | BDBM50251026 ((R)-(-)-2-Phenyl-apomorphine hydrochloride | CHEMB...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 88 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tartu Curated by ChEMBL | Assay Description Displacement of [3H]SCH23390 from dopamine D1 receptor expressed in Ltk deficient fibroblast cells by liquid scintillation counting | Bioorg Med Chem 17: 4756-62 (2009) Article DOI: 10.1016/j.bmc.2009.04.047 BindingDB Entry DOI: 10.7270/Q2KD1XZ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(1A) dopamine receptor (Homo sapiens (Human)) | BDBM50295866 (CHEMBL560721 | N-Propyl-2-(4-hydroxyphenyl)-norapo...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 94 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tartu Curated by ChEMBL | Assay Description Displacement of [3H]SCH23390 from dopamine D1 receptor expressed in Ltk deficient fibroblast cells by liquid scintillation counting | Bioorg Med Chem 17: 4756-62 (2009) Article DOI: 10.1016/j.bmc.2009.04.047 BindingDB Entry DOI: 10.7270/Q2KD1XZ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(1A) dopamine receptor (Mus musculus (Mouse)) | BDBM50001955 ((-)6-Methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]qu...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank PC cid PC sid PDB UniChem Patents Similars | PDB Article PubMed | 101 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Debrecen Curated by ChEMBL | Assay Description Displacement of [3H]SCH23390 from dopamine D1 receptor in mouse Ltk- fibroblast cells | Bioorg Med Chem 16: 4563-8 (2008) Article DOI: 10.1016/j.bmc.2008.02.038 BindingDB Entry DOI: 10.7270/Q24J0DW0 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
D(2) dopamine receptor (Rattus norvegicus (rat)) | BDBM50295861 (CHEMBL562460 | N-Ethyl-2-methylnorapomorphine hydr...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 115 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tartu Curated by ChEMBL | Assay Description Displacement of [3H]raclopride from rat dopamine D2short receptor expressed in CHO-K1 cells by liquid scintillation counting | Bioorg Med Chem 17: 4756-62 (2009) Article DOI: 10.1016/j.bmc.2009.04.047 BindingDB Entry DOI: 10.7270/Q2KD1XZ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(1A) dopamine receptor (Homo sapiens (Human)) | BDBM50295863 (CHEMBL562935 | N-Ethyl-2-(4-hydroxyphenyl)-norapom...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 124 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tartu Curated by ChEMBL | Assay Description Displacement of [3H]SCH23390 from dopamine D1 receptor expressed in Ltk deficient fibroblast cells by liquid scintillation counting | Bioorg Med Chem 17: 4756-62 (2009) Article DOI: 10.1016/j.bmc.2009.04.047 BindingDB Entry DOI: 10.7270/Q2KD1XZ4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(1A) dopamine receptor (Homo sapiens (Human)) | BDBM55121 (3-HYDROXYTYRAMINE HYDROCHLORIDE | 4-(2-aminoethyl)...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase DrugBank KEGG PC cid PC sid PDB UniChem Similars | DrugBank PDB Article PubMed | 124 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Tartu Curated by ChEMBL | Assay Description Displacement of [3H]SCH23390 from dopamine D1 receptor expressed in Ltk deficient fibroblast cells by liquid scintillation counting | Bioorg Med Chem 17: 4756-62 (2009) Article DOI: 10.1016/j.bmc.2009.04.047 BindingDB Entry DOI: 10.7270/Q2KD1XZ4 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) |
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