Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Peroxisome proliferator-activated receptor gamma (Homo sapiens (Human)) | BDBM50428854 (CHEMBL1236924) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Similars | MMDB PDB Article PubMed | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Displacement of [3H]rosiglitazone from human PPARgamma LBD expressed in HEK293 cells by filtration assay | J Med Chem 60: 4584-4593 (2017) Article DOI: 10.1021/acs.jmedchem.6b01727 BindingDB Entry DOI: 10.7270/Q23J3G4S | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50002903 (CHEMBL223836) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 15 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RX 821002 from human adrenergic alpha2A receptor expressed in CHO cells | J Med Chem 50: 3964-8 (2007) Checked by Author Article DOI: 10.1021/jm061487a BindingDB Entry DOI: 10.7270/Q2W095NP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2C adrenergic receptor (Homo sapiens (Human)) | BDBM50002903 (CHEMBL223836) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 17 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RX 821002 from human adrenergic Alpha-2C receptor expressed in CHO cells | J Med Chem 50: 3964-8 (2007) Checked by Author Article DOI: 10.1021/jm061487a BindingDB Entry DOI: 10.7270/Q2W095NP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2C adrenergic receptor (Homo sapiens (Human)) | BDBM50417350 (CHEMBL374584) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 18 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RX 821002 from human adrenergic Alpha-2C receptor expressed in CHO cells | J Med Chem 50: 3964-8 (2007) Checked by Author Article DOI: 10.1021/jm061487a BindingDB Entry DOI: 10.7270/Q2W095NP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50417350 (CHEMBL374584) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 28 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RX 821002 from human adrenergic alpha2A receptor expressed in CHO cells | J Med Chem 50: 3964-8 (2007) Checked by Author Article DOI: 10.1021/jm061487a BindingDB Entry DOI: 10.7270/Q2W095NP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2C adrenergic receptor (Homo sapiens (Human)) | BDBM50085683 ((+)-4-((S)-alpha,2,3-trimethylbenzyl)imidazole | 4...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | 31 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RX 821002 from human adrenergic alpha-2c receptor expressed in CHO cells in presence of GppNHp/Na | J Med Chem 50: 3964-8 (2007) Checked by Author Article DOI: 10.1021/jm061487a BindingDB Entry DOI: 10.7270/Q2W095NP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50412250 (CHEMBL128168) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 48 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RX 821002 from human adrenergic alpha2A receptor expressed in CHO cells | J Med Chem 50: 3964-8 (2007) Checked by Author Article DOI: 10.1021/jm061487a BindingDB Entry DOI: 10.7270/Q2W095NP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50002904 (CHEMBL222928) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RX 821002 from human adrenergic alpha2A receptor expressed in CHO cells | J Med Chem 50: 3964-8 (2007) Checked by Author Article DOI: 10.1021/jm061487a BindingDB Entry DOI: 10.7270/Q2W095NP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2C adrenergic receptor (Homo sapiens (Human)) | BDBM50002905 (CHEMBL373535) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 65 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RX 821002 from human adrenergic Alpha-2C receptor expressed in CHO cells | J Med Chem 50: 3964-8 (2007) Checked by Author Article DOI: 10.1021/jm061487a BindingDB Entry DOI: 10.7270/Q2W095NP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50417341 (CHEMBL397753) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 72 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RX 821002 from human adrenergic alpha2A receptor expressed in CHO cells | J Med Chem 50: 3964-8 (2007) Checked by Author Article DOI: 10.1021/jm061487a BindingDB Entry DOI: 10.7270/Q2W095NP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50218115 ((R)-2-[1-(3'-nitrobiphenyl-2-yloxy)ethyl]-4,5-dihy...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 81 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RX 821002 from human adrenergic alpha2A receptor expressed in CHO cells | J Med Chem 50: 3964-8 (2007) Checked by Author Article DOI: 10.1021/jm061487a BindingDB Entry DOI: 10.7270/Q2W095NP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50417354 (CHEMBL396013) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 91 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RX 821002 from human adrenergic alpha2A receptor expressed in CHO cells | J Med Chem 50: 3964-8 (2007) Checked by Author Article DOI: 10.1021/jm061487a BindingDB Entry DOI: 10.7270/Q2W095NP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50002905 (CHEMBL373535) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 138 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RX 821002 from human adrenergic alpha2A receptor expressed in CHO cells | J Med Chem 50: 3964-8 (2007) Checked by Author Article DOI: 10.1021/jm061487a BindingDB Entry DOI: 10.7270/Q2W095NP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2A adrenergic receptor (Homo sapiens (Human)) | BDBM50417353 (CHEMBL242265) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 186 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RX 821002 from human adrenergic alpha2A receptor expressed in CHO cells | J Med Chem 50: 3964-8 (2007) Checked by Author Article DOI: 10.1021/jm061487a BindingDB Entry DOI: 10.7270/Q2W095NP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2C adrenergic receptor (Homo sapiens (Human)) | BDBM50412250 (CHEMBL128168) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 200 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RX 821002 from human adrenergic Alpha-2C receptor expressed in CHO cells | J Med Chem 50: 3964-8 (2007) Checked by Author Article DOI: 10.1021/jm061487a BindingDB Entry DOI: 10.7270/Q2W095NP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2C adrenergic receptor (Homo sapiens (Human)) | BDBM50002904 (CHEMBL222928) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 234 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RX 821002 from human adrenergic Alpha-2C receptor expressed in CHO cells | J Med Chem 50: 3964-8 (2007) Checked by Author Article DOI: 10.1021/jm061487a BindingDB Entry DOI: 10.7270/Q2W095NP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2C adrenergic receptor (Homo sapiens (Human)) | BDBM50218115 ((R)-2-[1-(3'-nitrobiphenyl-2-yloxy)ethyl]-4,5-dihy...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 257 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RX 821002 from human adrenergic Alpha-2C receptor expressed in CHO cells | J Med Chem 50: 3964-8 (2007) Checked by Author Article DOI: 10.1021/jm061487a BindingDB Entry DOI: 10.7270/Q2W095NP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2B adrenergic receptor (Homo sapiens (Human)) | BDBM50002903 (CHEMBL223836) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 269 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RX 821002 from human adrenergic alpha-2B receptor expressed in CHO cells | J Med Chem 50: 3964-8 (2007) Checked by Author Article DOI: 10.1021/jm061487a BindingDB Entry DOI: 10.7270/Q2W095NP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2C adrenergic receptor (Homo sapiens (Human)) | BDBM50417354 (CHEMBL396013) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 302 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RX 821002 from human adrenergic Alpha-2C receptor expressed in CHO cells | J Med Chem 50: 3964-8 (2007) Checked by Author Article DOI: 10.1021/jm061487a BindingDB Entry DOI: 10.7270/Q2W095NP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2B adrenergic receptor (Homo sapiens (Human)) | BDBM50417350 (CHEMBL374584) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 355 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RX 821002 from human adrenergic alpha-2B receptor expressed in CHO cells | J Med Chem 50: 3964-8 (2007) Checked by Author Article DOI: 10.1021/jm061487a BindingDB Entry DOI: 10.7270/Q2W095NP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2C adrenergic receptor (Homo sapiens (Human)) | BDBM50218115 ((R)-2-[1-(3'-nitrobiphenyl-2-yloxy)ethyl]-4,5-dihy...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 363 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RX 821002 from human adrenergic alpha-2c receptor expressed in CHO cells in presence of GppNHp/Na | J Med Chem 50: 3964-8 (2007) Checked by Author Article DOI: 10.1021/jm061487a BindingDB Entry DOI: 10.7270/Q2W095NP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2B adrenergic receptor (Homo sapiens (Human)) | BDBM50412250 (CHEMBL128168) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 501 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RX 821002 from human adrenergic alpha-2B receptor expressed in CHO cells | J Med Chem 50: 3964-8 (2007) Checked by Author Article DOI: 10.1021/jm061487a BindingDB Entry DOI: 10.7270/Q2W095NP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2C adrenergic receptor (Homo sapiens (Human)) | BDBM50417341 (CHEMBL397753) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 537 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RX 821002 from human adrenergic Alpha-2C receptor expressed in CHO cells | J Med Chem 50: 3964-8 (2007) Checked by Author Article DOI: 10.1021/jm061487a BindingDB Entry DOI: 10.7270/Q2W095NP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2B adrenergic receptor (Homo sapiens (Human)) | BDBM50417354 (CHEMBL396013) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 589 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RX 821002 from human adrenergic alpha-2B receptor expressed in CHO cells | J Med Chem 50: 3964-8 (2007) Checked by Author Article DOI: 10.1021/jm061487a BindingDB Entry DOI: 10.7270/Q2W095NP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2B adrenergic receptor (Homo sapiens (Human)) | BDBM50002904 (CHEMBL222928) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 661 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RX 821002 from human adrenergic alpha-2B receptor expressed in CHO cells | J Med Chem 50: 3964-8 (2007) Checked by Author Article DOI: 10.1021/jm061487a BindingDB Entry DOI: 10.7270/Q2W095NP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2B adrenergic receptor (Homo sapiens (Human)) | BDBM50218115 ((R)-2-[1-(3'-nitrobiphenyl-2-yloxy)ethyl]-4,5-dihy...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 741 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RX 821002 from human adrenergic alpha-2B receptor expressed in CHO cells | J Med Chem 50: 3964-8 (2007) Checked by Author Article DOI: 10.1021/jm061487a BindingDB Entry DOI: 10.7270/Q2W095NP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2B adrenergic receptor (Homo sapiens (Human)) | BDBM50002905 (CHEMBL373535) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 933 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RX 821002 from human adrenergic alpha-2B receptor expressed in CHO cells | J Med Chem 50: 3964-8 (2007) Checked by Author Article DOI: 10.1021/jm061487a BindingDB Entry DOI: 10.7270/Q2W095NP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2C adrenergic receptor (Homo sapiens (Human)) | BDBM50417353 (CHEMBL242265) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 977 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RX 821002 from human adrenergic Alpha-2C receptor expressed in CHO cells | J Med Chem 50: 3964-8 (2007) Checked by Author Article DOI: 10.1021/jm061487a BindingDB Entry DOI: 10.7270/Q2W095NP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M2 (Homo sapiens (Human)) | BDBM50004656 ((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank KEGG MMDB PC cid PC sid PDB UniChem Similars | Article PubMed | 1.23E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cells by microplate scintillation counting | Bioorg Med Chem 17: 8174-85 (2009) Article DOI: 10.1016/j.bmc.2009.10.027 BindingDB Entry DOI: 10.7270/Q2125TW3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2B adrenergic receptor (Homo sapiens (Human)) | BDBM50417353 (CHEMBL242265) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.26E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RX 821002 from human adrenergic alpha-2B receptor expressed in CHO cells | J Med Chem 50: 3964-8 (2007) Checked by Author Article DOI: 10.1021/jm061487a BindingDB Entry DOI: 10.7270/Q2W095NP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M2 (Homo sapiens (Human)) | BDBM50385682 (CHEMBL390842) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.58E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cells by microplate scintillation counting | Bioorg Med Chem 17: 8174-85 (2009) Article DOI: 10.1016/j.bmc.2009.10.027 BindingDB Entry DOI: 10.7270/Q2125TW3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-2B adrenergic receptor (Homo sapiens (Human)) | BDBM50417341 (CHEMBL397753) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.59E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università degli Studi di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]RX 821002 from human adrenergic alpha-2B receptor expressed in CHO cells | J Med Chem 50: 3964-8 (2007) Checked by Author Article DOI: 10.1021/jm061487a BindingDB Entry DOI: 10.7270/Q2W095NP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M1 (Homo sapiens (Human)) | BDBM50006584 ((McN-A-343) [4-(3-Chloro-phenylcarbamoyloxy)-but-2...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | 1.95E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells by microplate scintillation counting | Bioorg Med Chem 17: 8174-85 (2009) Article DOI: 10.1016/j.bmc.2009.10.027 BindingDB Entry DOI: 10.7270/Q2125TW3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M3 (Homo sapiens (Human)) | BDBM50006584 ((McN-A-343) [4-(3-Chloro-phenylcarbamoyloxy)-but-2...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | 2.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO cells by microplate scintillation counting | Bioorg Med Chem 17: 8174-85 (2009) Article DOI: 10.1016/j.bmc.2009.10.027 BindingDB Entry DOI: 10.7270/Q2125TW3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M2 (Homo sapiens (Human)) | BDBM50006584 ((McN-A-343) [4-(3-Chloro-phenylcarbamoyloxy)-but-2...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | 3.24E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cells by microplate scintillation counting | Bioorg Med Chem 17: 8174-85 (2009) Article DOI: 10.1016/j.bmc.2009.10.027 BindingDB Entry DOI: 10.7270/Q2125TW3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M5 (Homo sapiens (Human)) | BDBM50006584 ((McN-A-343) [4-(3-Chloro-phenylcarbamoyloxy)-but-2...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | 3.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human muscarinic M5 receptor expressed in CHO cells by microplate scintillation counting | Bioorg Med Chem 17: 8174-85 (2009) Article DOI: 10.1016/j.bmc.2009.10.027 BindingDB Entry DOI: 10.7270/Q2125TW3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M2 (Homo sapiens (Human)) | BDBM50415218 (CHEMBL404557) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cells by microplate scintillation counting | Bioorg Med Chem 17: 8174-85 (2009) Article DOI: 10.1016/j.bmc.2009.10.027 BindingDB Entry DOI: 10.7270/Q2125TW3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M4 (Homo sapiens (Human)) | BDBM50004656 ((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank KEGG MMDB PC cid PC sid PDB UniChem Similars | Article PubMed | 6.31E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human muscarinic M4 receptor expressed in CHO cells by microplate scintillation counting | Bioorg Med Chem 17: 8174-85 (2009) Article DOI: 10.1016/j.bmc.2009.10.027 BindingDB Entry DOI: 10.7270/Q2125TW3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M3 (Homo sapiens (Human)) | BDBM50385682 (CHEMBL390842) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7.59E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO cells by microplate scintillation counting | Bioorg Med Chem 17: 8174-85 (2009) Article DOI: 10.1016/j.bmc.2009.10.027 BindingDB Entry DOI: 10.7270/Q2125TW3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M5 (Homo sapiens (Human)) | BDBM50385682 (CHEMBL390842) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7.76E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human muscarinic M5 receptor expressed in CHO cells by microplate scintillation counting | Bioorg Med Chem 17: 8174-85 (2009) Article DOI: 10.1016/j.bmc.2009.10.027 BindingDB Entry DOI: 10.7270/Q2125TW3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M4 (Homo sapiens (Human)) | BDBM50006584 ((McN-A-343) [4-(3-Chloro-phenylcarbamoyloxy)-but-2...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | 9.12E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human muscarinic M4 receptor expressed in CHO cells by microplate scintillation counting | Bioorg Med Chem 17: 8174-85 (2009) Article DOI: 10.1016/j.bmc.2009.10.027 BindingDB Entry DOI: 10.7270/Q2125TW3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M3 (Homo sapiens (Human)) | BDBM50415225 (CHEMBL593620) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.05E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO cells by microplate scintillation counting | Bioorg Med Chem 17: 8174-85 (2009) Article DOI: 10.1016/j.bmc.2009.10.027 BindingDB Entry DOI: 10.7270/Q2125TW3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M3 (Homo sapiens (Human)) | BDBM50415219 (CHEMBL595265) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO cells by microplate scintillation counting | Bioorg Med Chem 17: 8174-85 (2009) Article DOI: 10.1016/j.bmc.2009.10.027 BindingDB Entry DOI: 10.7270/Q2125TW3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M2 (Homo sapiens (Human)) | BDBM50415222 (CHEMBL594376) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.12E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cells by microplate scintillation counting | Bioorg Med Chem 17: 8174-85 (2009) Article DOI: 10.1016/j.bmc.2009.10.027 BindingDB Entry DOI: 10.7270/Q2125TW3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M4 (Homo sapiens (Human)) | BDBM50385682 (CHEMBL390842) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.15E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human muscarinic M4 receptor expressed in CHO cells by microplate scintillation counting | Bioorg Med Chem 17: 8174-85 (2009) Article DOI: 10.1016/j.bmc.2009.10.027 BindingDB Entry DOI: 10.7270/Q2125TW3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M2 (Homo sapiens (Human)) | BDBM50415219 (CHEMBL595265) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.38E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cells by microplate scintillation counting | Bioorg Med Chem 17: 8174-85 (2009) Article DOI: 10.1016/j.bmc.2009.10.027 BindingDB Entry DOI: 10.7270/Q2125TW3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M5 (Homo sapiens (Human)) | BDBM50415219 (CHEMBL595265) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.55E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human muscarinic M5 receptor expressed in CHO cells by microplate scintillation counting | Bioorg Med Chem 17: 8174-85 (2009) Article DOI: 10.1016/j.bmc.2009.10.027 BindingDB Entry DOI: 10.7270/Q2125TW3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M3 (Homo sapiens (Human)) | BDBM50415224 (CHEMBL593685) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.62E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO cells by microplate scintillation counting | Bioorg Med Chem 17: 8174-85 (2009) Article DOI: 10.1016/j.bmc.2009.10.027 BindingDB Entry DOI: 10.7270/Q2125TW3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M2 (Homo sapiens (Human)) | BDBM50415215 (CHEMBL593871) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.66E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cells by microplate scintillation counting | Bioorg Med Chem 17: 8174-85 (2009) Article DOI: 10.1016/j.bmc.2009.10.027 BindingDB Entry DOI: 10.7270/Q2125TW3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M5 (Homo sapiens (Human)) | BDBM50415225 (CHEMBL593620) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.66E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Camerino Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human muscarinic M5 receptor expressed in CHO cells by microplate scintillation counting | Bioorg Med Chem 17: 8174-85 (2009) Article DOI: 10.1016/j.bmc.2009.10.027 BindingDB Entry DOI: 10.7270/Q2125TW3 | |||||||||||
More data for this Ligand-Target Pair |
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