Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50011635 (1-{3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,8...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 0.200 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description PAF-antagonist activity determined in dog platelets by PAF-binding assay | J Med Chem 34: 1209-21 (1991) BindingDB Entry DOI: 10.7270/Q23X85M1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50011650 (1-{3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,8...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 0.300 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description PAF-antagonist activity determined in dog platelets by PAF-binding assay | J Med Chem 34: 1209-21 (1991) BindingDB Entry DOI: 10.7270/Q23X85M1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50011611 (1-{3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,8...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 0.600 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description PAF-antagonist activity determined in dog platelets by PAF-binding assay | J Med Chem 34: 1209-21 (1991) BindingDB Entry DOI: 10.7270/Q23X85M1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50011623 (2a-{3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 0.700 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description PAF-antagonist activity determined in dog platelets by PAF-binding assay | J Med Chem 34: 1209-21 (1991) BindingDB Entry DOI: 10.7270/Q23X85M1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50011634 (4-{3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,8...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 0.700 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description PAF-antagonist activity determined in dog platelets by PAF-binding assay | J Med Chem 34: 1209-21 (1991) BindingDB Entry DOI: 10.7270/Q23X85M1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50011603 (1-{3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,8...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description PAF-antagonist activity determined in dog platelets by PAF-binding assay | J Med Chem 34: 1209-21 (1991) BindingDB Entry DOI: 10.7270/Q23X85M1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50011640 (4-(2-Chloro-phenyl)-2-(3-indazol-1-yl-prop-1-ynyl)...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description PAF-antagonist activity determined in dog platelets by PAF-binding assay | J Med Chem 34: 1209-21 (1991) BindingDB Entry DOI: 10.7270/Q23X85M1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50011653 (2-{3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,8...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description PAF-antagonist activity determined in dog platelets by PAF-binding assay | J Med Chem 34: 1209-21 (1991) BindingDB Entry DOI: 10.7270/Q23X85M1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50013923 (3-(1-Butyl-4-methoxy-naphthalen-2-yl)-N-(1-methyl-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. Curated by ChEMBL | Assay Description Inhibition of [3H]-PAF binding to platelet activating factor receptor citrate-treated dog blood | J Med Chem 33: 2856-64 (1990) BindingDB Entry DOI: 10.7270/Q21V5CZJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018350 (5-(4-Methoxy-phenyl)-5-phenyl-penta-2,4-dienoic ac...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand | J Med Chem 32: 1820-35 (1989) BindingDB Entry DOI: 10.7270/Q2NZ86MR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018388 (5,5-Bis-(3-methoxy-phenyl)-penta-2,4-dienoic acid ...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand | J Med Chem 32: 1820-35 (1989) BindingDB Entry DOI: 10.7270/Q2NZ86MR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50011669 (1-{3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,8...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description PAF-antagonist activity determined in dog platelets by PAF-binding assay | J Med Chem 34: 1209-21 (1991) BindingDB Entry DOI: 10.7270/Q23X85M1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50013924 (3-(1-Butyl-4,7-dimethoxy-naphthalen-2-yl)-N-(1-met...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. Curated by ChEMBL | Assay Description Inhibition of [3H]-PAF binding to platelet activating factor receptor citrate-treated dog blood | J Med Chem 33: 2856-64 (1990) BindingDB Entry DOI: 10.7270/Q21V5CZJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50011673 (4-(2-Chloro-phenyl)-9-methyl-2-(3-phenoxy-prop-1-y...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description PAF-antagonist activity determined in dog platelets by PAF-binding assay | J Med Chem 34: 1209-21 (1991) BindingDB Entry DOI: 10.7270/Q23X85M1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50011663 (1-{3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,8...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description PAF-antagonist activity determined in dog platelets by PAF-binding assay | J Med Chem 34: 1209-21 (1991) BindingDB Entry DOI: 10.7270/Q23X85M1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50011602 (2-{3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,8...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description PAF-antagonist activity determined in dog platelets by PAF-binding assay | J Med Chem 34: 1209-21 (1991) BindingDB Entry DOI: 10.7270/Q23X85M1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018392 (5-(4-Methoxy-phenyl)-5-phenyl-penta-2,4-dienoic ac...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of [3H]-PAF binding to dog platelets. | J Med Chem 32: 1820-35 (1989) BindingDB Entry DOI: 10.7270/Q2NZ86MR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50011646 (1-{3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,8...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description PAF-antagonist activity determined in dog platelets by PAF-binding assay | J Med Chem 34: 1209-21 (1991) BindingDB Entry DOI: 10.7270/Q23X85M1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50011649 (4-{3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,8...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description PAF-antagonist activity determined in dog platelets by PAF-binding assay | J Med Chem 34: 1209-21 (1991) BindingDB Entry DOI: 10.7270/Q23X85M1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50011627 (4-(2-Chloro-phenyl)-9-methyl-2-[3-(pyridin-3-yloxy...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description PAF-antagonist activity determined in dog platelets by PAF-binding assay | J Med Chem 34: 1209-21 (1991) BindingDB Entry DOI: 10.7270/Q23X85M1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018341 (2-Ethyl-3',4'-dimethoxy-biphenyl-4-carboxylic acid...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand. | J Med Chem 32: 1814-20 (1989) BindingDB Entry DOI: 10.7270/Q2SQ8ZCJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018316 (2-Butyl-3',4'-dimethoxy-biphenyl-4-carboxylic acid...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand. | J Med Chem 32: 1814-20 (1989) BindingDB Entry DOI: 10.7270/Q2SQ8ZCJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018325 (CHEMBL53584 | [1,1';2',1'']Terphenyl-4'-carboxylic...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand. | J Med Chem 32: 1814-20 (1989) BindingDB Entry DOI: 10.7270/Q2SQ8ZCJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018315 (2-Ethynyl-3',4'-dimethoxy-biphenyl-4-carboxylic ac...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand. | J Med Chem 32: 1814-20 (1989) BindingDB Entry DOI: 10.7270/Q2SQ8ZCJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018390 (5-(4-Methoxy-phenyl)-trideca-2,4-dienoic acid (1-m...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of [3H]-PAF binding to dog platelets. | J Med Chem 32: 1820-35 (1989) BindingDB Entry DOI: 10.7270/Q2NZ86MR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50011632 (4-{3-[6-(2-Fluoro-phenyl)-1-methyl-4H-2,3,5,10b-te...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description PAF-antagonist activity determined in dog platelets by PAF-binding assay | J Med Chem 34: 1209-21 (1991) BindingDB Entry DOI: 10.7270/Q23X85M1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50011666 (1-{3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,8...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description PAF-antagonist activity determined in dog platelets by PAF-binding assay | J Med Chem 34: 1209-21 (1991) BindingDB Entry DOI: 10.7270/Q23X85M1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50011661 (2-{3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,8...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description PAF-antagonist activity determined in dog platelets by PAF-binding assay | J Med Chem 34: 1209-21 (1991) BindingDB Entry DOI: 10.7270/Q23X85M1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50011655 (6-Chloro-4-{3-[4-(2-chloro-phenyl)-9-methyl-6H-1-t...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description PAF-antagonist activity determined in dog platelets by PAF-binding assay | J Med Chem 34: 1209-21 (1991) BindingDB Entry DOI: 10.7270/Q23X85M1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50011631 (2-{3-[6-(2-Fluoro-phenyl)-1-trifluoromethyl-4H-2,3...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description PAF-antagonist activity determined in dog platelets by PAF-binding assay | J Med Chem 34: 1209-21 (1991) BindingDB Entry DOI: 10.7270/Q23X85M1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50011624 (2-(3-Benzoimidazol-1-yl-prop-1-ynyl)-4-(2-chloro-p...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description PAF-antagonist activity determined in dog platelets by PAF-binding assay | J Med Chem 34: 1209-21 (1991) BindingDB Entry DOI: 10.7270/Q23X85M1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50011660 (1-{3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,8...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description PAF-antagonist activity determined in dog platelets by PAF-binding assay | J Med Chem 34: 1209-21 (1991) BindingDB Entry DOI: 10.7270/Q23X85M1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50011612 (1-{3-[6-(2-Fluoro-phenyl)-1,4-dimethyl-4H-2,3,5,10...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description PAF-antagonist activity determined in dog platelets by PAF-binding assay | J Med Chem 34: 1209-21 (1991) BindingDB Entry DOI: 10.7270/Q23X85M1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50011625 (5-{3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,8...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description PAF-antagonist activity determined in dog platelets by PAF-binding assay | J Med Chem 34: 1209-21 (1991) BindingDB Entry DOI: 10.7270/Q23X85M1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50013921 (3-(1-Butyl-5-methoxy-naphthalen-2-yl)-N-(1-methyl-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. Curated by ChEMBL | Assay Description Inhibition of [3H]-PAF binding to platelet activating factor receptor citrate-treated dog blood | J Med Chem 33: 2856-64 (1990) BindingDB Entry DOI: 10.7270/Q21V5CZJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50011648 (1-{3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,8...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description PAF-antagonist activity determined in dog platelets by PAF-binding assay | J Med Chem 34: 1209-21 (1991) BindingDB Entry DOI: 10.7270/Q23X85M1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50011609 (7-Chloro-1-{3-[4-(2-chloro-phenyl)-9-methyl-6H-1-t...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 7 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description PAF-antagonist activity determined in dog platelets by PAF-binding assay | J Med Chem 34: 1209-21 (1991) BindingDB Entry DOI: 10.7270/Q23X85M1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50011605 (4-(2-Chloro-phenyl)-9-methyl-2-[3-(1,2,3,4-tetrahy...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 7 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description PAF-antagonist activity determined in dog platelets by PAF-binding assay | J Med Chem 34: 1209-21 (1991) BindingDB Entry DOI: 10.7270/Q23X85M1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50011626 (4-{3-[6-(2-Fluoro-phenyl)-1-methyl-4H-2,3,5,10b-te...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | PubMed | n/a | n/a | 7 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description PAF-antagonist activity determined in dog platelets by PAF-binding assay | J Med Chem 34: 1209-21 (1991) BindingDB Entry DOI: 10.7270/Q23X85M1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50011607 (1-{3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,8...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 7 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description PAF-antagonist activity determined in dog platelets by PAF-binding assay | J Med Chem 34: 1209-21 (1991) BindingDB Entry DOI: 10.7270/Q23X85M1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50013925 (3-(1-Butyl-6-methoxy-naphthalen-2-yl)-N-(1-methyl-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 7 | n/a | n/a | n/a | n/a | n/a | n/a |
Hoffmann-La Roche Inc. Curated by ChEMBL | Assay Description Inhibition of [3H]-PAF binding to platelet activating factor receptor citrate-treated dog blood | J Med Chem 33: 2856-64 (1990) BindingDB Entry DOI: 10.7270/Q21V5CZJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50011872 (4-(2-Chloro-phenyl)-9-methyl-2-[2-(5-pyridin-2-yl-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 8 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets. | J Med Chem 34: 1440-6 (1991) BindingDB Entry DOI: 10.7270/Q2BG2MZ9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50011613 (1-{3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,8...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 9 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description PAF-antagonist activity determined in dog platelets by PAF-binding assay | J Med Chem 34: 1209-21 (1991) BindingDB Entry DOI: 10.7270/Q23X85M1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50011651 (6,8-Dichloro-1-{3-[4-(2-chloro-phenyl)-9-methyl-6H...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 9 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description PAF-antagonist activity determined in dog platelets by PAF-binding assay | J Med Chem 34: 1209-21 (1991) BindingDB Entry DOI: 10.7270/Q23X85M1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018361 (5-(4-Methoxy-phenyl)-undeca-2,4-dienoic acid (1-me...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 9 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of [3H]-PAF binding to dog platelets. | J Med Chem 32: 1820-35 (1989) BindingDB Entry DOI: 10.7270/Q2NZ86MR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50011866 (2-[2-(4-Butyl-phenyl)-ethyl]-4-(2-chloro-phenyl)-9...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets. | J Med Chem 34: 1440-6 (1991) BindingDB Entry DOI: 10.7270/Q2BG2MZ9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018349 (5-(4-Methoxy-phenyl)-deca-2,4-dienoic acid (1-meth...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand | J Med Chem 32: 1820-35 (1989) BindingDB Entry DOI: 10.7270/Q2NZ86MR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50011665 (2-{3-[6-(2-Fluoro-phenyl)-1-methyl-4H-2,3,5,10b-te...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description PAF-antagonist activity determined in dog platelets by PAF-binding assay | J Med Chem 34: 1209-21 (1991) BindingDB Entry DOI: 10.7270/Q23X85M1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50011876 (4-(2-Chloro-phenyl)-2-ethynyl-9-methyl-6H-1-thia-5...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets. | J Med Chem 34: 1440-6 (1991) BindingDB Entry DOI: 10.7270/Q2BG2MZ9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018347 (5,5-Bis-(4-methoxy-phenyl)-penta-2,4-dienoic acid ...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand | J Med Chem 32: 1820-35 (1989) BindingDB Entry DOI: 10.7270/Q2NZ86MR | |||||||||||
More data for this Ligand-Target Pair |
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