Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50442630 (CHEMBL2441638) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.390 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from rhesus monkey histamine H3 receptor expressed in CHO cells | Bioorg Med Chem Lett 23: 6141-5 (2013) Article DOI: 10.1016/j.bmcl.2013.09.006 BindingDB Entry DOI: 10.7270/Q24T6KT6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50443217 (CHEMBL3087669) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 0.400 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from recombinant rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation... | Bioorg Med Chem Lett 23: 6269-73 (2013) Article DOI: 10.1016/j.bmcl.2013.09.081 BindingDB Entry DOI: 10.7270/Q27D2WK2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50442628 (CHEMBL2441640) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from rhesus monkey histamine H3 receptor expressed in CHO cells | Bioorg Med Chem Lett 23: 6141-5 (2013) Article DOI: 10.1016/j.bmcl.2013.09.006 BindingDB Entry DOI: 10.7270/Q24T6KT6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(4) dopamine receptor (Homo sapiens (Human)) | BDBM84440 (Isoindoline, 7 | Isoindoline, 8 | Isoindoline, 9) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 0.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Aventis Pharmaceuticals | Assay Description Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp. | Chembiochem 3: 999-1009 (2002) Article DOI: 10.1002/1439-7633(20021004)3:10 BindingDB Entry DOI: 10.7270/Q27D2SP5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(4) dopamine receptor (Homo sapiens (Human)) | BDBM84445 (Isoindoline, 12) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 0.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Aventis Pharmaceuticals | Assay Description Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp. | Chembiochem 3: 999-1009 (2002) Article DOI: 10.1002/1439-7633(20021004)3:10 BindingDB Entry DOI: 10.7270/Q27D2SP5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50442627 (CHEMBL2441641) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.550 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from rhesus monkey histamine H3 receptor expressed in CHO cells | Bioorg Med Chem Lett 23: 6141-5 (2013) Article DOI: 10.1016/j.bmcl.2013.09.006 BindingDB Entry DOI: 10.7270/Q24T6KT6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50442629 (CHEMBL2441639) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.550 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from rhesus monkey histamine H3 receptor expressed in CHO cells | Bioorg Med Chem Lett 23: 6141-5 (2013) Article DOI: 10.1016/j.bmcl.2013.09.006 BindingDB Entry DOI: 10.7270/Q24T6KT6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(4) dopamine receptor (Homo sapiens (Human)) | BDBM84451 (Isoindoline, 18 | Isoindoline, 19) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 0.600 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Aventis Pharmaceuticals | Assay Description Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp. | Chembiochem 3: 999-1009 (2002) Article DOI: 10.1002/1439-7633(20021004)3:10 BindingDB Entry DOI: 10.7270/Q27D2SP5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50442626 (CHEMBL2441642) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.850 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from rhesus monkey histamine H3 receptor expressed in CHO cells | Bioorg Med Chem Lett 23: 6141-5 (2013) Article DOI: 10.1016/j.bmcl.2013.09.006 BindingDB Entry DOI: 10.7270/Q24T6KT6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM50443217 (CHEMBL3087669) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 0.900 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]-methylhistamine from rat histamine H3 receptor (445 amino acid residues) transfected in human 293 cells after 1 hr by scintillat... | Bioorg Med Chem Lett 23: 6269-73 (2013) Article DOI: 10.1016/j.bmcl.2013.09.081 BindingDB Entry DOI: 10.7270/Q27D2WK2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50442632 (CHEMBL2441636) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.970 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from rhesus monkey histamine H3 receptor expressed in CHO cells | Bioorg Med Chem Lett 23: 6141-5 (2013) Article DOI: 10.1016/j.bmcl.2013.09.006 BindingDB Entry DOI: 10.7270/Q24T6KT6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(4) dopamine receptor (Homo sapiens (Human)) | BDBM84440 (Isoindoline, 7 | Isoindoline, 8 | Isoindoline, 9) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 1 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Aventis Pharmaceuticals | Assay Description Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp. | Chembiochem 3: 999-1009 (2002) Article DOI: 10.1002/1439-7633(20021004)3:10 BindingDB Entry DOI: 10.7270/Q27D2SP5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50443216 (CHEMBL3087667) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 1.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from recombinant rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation... | Bioorg Med Chem Lett 23: 6269-73 (2013) Article DOI: 10.1016/j.bmcl.2013.09.081 BindingDB Entry DOI: 10.7270/Q27D2WK2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(4) dopamine receptor (Homo sapiens (Human)) | BDBM84446 (Isoindoline, 13) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 1.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Aventis Pharmaceuticals | Assay Description Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp. | Chembiochem 3: 999-1009 (2002) Article DOI: 10.1002/1439-7633(20021004)3:10 BindingDB Entry DOI: 10.7270/Q27D2SP5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(4) dopamine receptor (Homo sapiens (Human)) | BDBM84443 (Isoindoline, 10 | Isoindoline, 11) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 1.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Aventis Pharmaceuticals | Assay Description Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp. | Chembiochem 3: 999-1009 (2002) Article DOI: 10.1002/1439-7633(20021004)3:10 BindingDB Entry DOI: 10.7270/Q27D2SP5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(4) dopamine receptor (Homo sapiens (Human)) | BDBM84453 (Isoindoline, 20) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 1.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Aventis Pharmaceuticals | Assay Description Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp. | Chembiochem 3: 999-1009 (2002) Article DOI: 10.1002/1439-7633(20021004)3:10 BindingDB Entry DOI: 10.7270/Q27D2SP5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50443227 (CHEMBL3087356) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 1.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from recombinant rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation... | Bioorg Med Chem Lett 23: 6269-73 (2013) Article DOI: 10.1016/j.bmcl.2013.09.081 BindingDB Entry DOI: 10.7270/Q27D2WK2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50443226 (CHEMBL3087357) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 1.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from recombinant rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation... | Bioorg Med Chem Lett 23: 6269-73 (2013) Article DOI: 10.1016/j.bmcl.2013.09.081 BindingDB Entry DOI: 10.7270/Q27D2WK2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50434389 (CHEMBL2387288) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun... | Bioorg Med Chem Lett 23: 3416-20 (2013) Article DOI: 10.1016/j.bmcl.2013.03.080 BindingDB Entry DOI: 10.7270/Q2RB75Z5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50437067 (CHEMBL2403550) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from recombinant rhesus monkey histamine H3 receptor transfected in CHO cell membranes after 1 hr by scin... | Bioorg Med Chem Lett 23: 4044-7 (2013) Article DOI: 10.1016/j.bmcl.2013.05.068 BindingDB Entry DOI: 10.7270/Q28C9XN0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50437067 (CHEMBL2403550) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from recombinant rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation... | Bioorg Med Chem Lett 23: 6269-73 (2013) Article DOI: 10.1016/j.bmcl.2013.09.081 BindingDB Entry DOI: 10.7270/Q27D2WK2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50443225 (CHEMBL3087671) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 2.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from recombinant rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation... | Bioorg Med Chem Lett 23: 6269-73 (2013) Article DOI: 10.1016/j.bmcl.2013.09.081 BindingDB Entry DOI: 10.7270/Q27D2WK2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50443224 (CHEMBL3087670) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from recombinant rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation... | Bioorg Med Chem Lett 23: 6269-73 (2013) Article DOI: 10.1016/j.bmcl.2013.09.081 BindingDB Entry DOI: 10.7270/Q27D2WK2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM50437067 (CHEMBL2403550) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from recombinant rat histamine H3 receptor transfected in CHO cell membranes after 1 hr by scintillation ... | Bioorg Med Chem Lett 23: 4044-7 (2013) Article DOI: 10.1016/j.bmcl.2013.05.068 BindingDB Entry DOI: 10.7270/Q28C9XN0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50442640 (CHEMBL2441653) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from rhesus monkey histamine H3 receptor expressed in CHO cells | Bioorg Med Chem Lett 23: 6141-5 (2013) Article DOI: 10.1016/j.bmcl.2013.09.006 BindingDB Entry DOI: 10.7270/Q24T6KT6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50434405 (CHEMBL2387306) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun... | Bioorg Med Chem Lett 23: 3416-20 (2013) Article DOI: 10.1016/j.bmcl.2013.03.080 BindingDB Entry DOI: 10.7270/Q2RB75Z5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50434382 (CHEMBL2387309) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 3.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun... | Bioorg Med Chem Lett 23: 3416-20 (2013) Article DOI: 10.1016/j.bmcl.2013.03.080 BindingDB Entry DOI: 10.7270/Q2RB75Z5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(4) dopamine receptor (Homo sapiens (Human)) | BDBM84459 (Isoindoline, 26) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 3.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Aventis Pharmaceuticals | Assay Description Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp. | Chembiochem 3: 999-1009 (2002) Article DOI: 10.1002/1439-7633(20021004)3:10 BindingDB Entry DOI: 10.7270/Q27D2SP5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(4) dopamine receptor (Homo sapiens (Human)) | BDBM84449 (Isoindoline, 16) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 3.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Aventis Pharmaceuticals | Assay Description Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp. | Chembiochem 3: 999-1009 (2002) Article DOI: 10.1002/1439-7633(20021004)3:10 BindingDB Entry DOI: 10.7270/Q27D2SP5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50442631 (CHEMBL2441637) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from rhesus monkey histamine H3 receptor expressed in CHO cells | Bioorg Med Chem Lett 23: 6141-5 (2013) Article DOI: 10.1016/j.bmcl.2013.09.006 BindingDB Entry DOI: 10.7270/Q24T6KT6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50443223 (CHEMBL3087358) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 3.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from recombinant rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation... | Bioorg Med Chem Lett 23: 6269-73 (2013) Article DOI: 10.1016/j.bmcl.2013.09.081 BindingDB Entry DOI: 10.7270/Q27D2WK2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1B adrenergic receptor (Rattus norvegicus (rat)) | BDBM84456 (Isoindoline, 23) | Reactome pathway UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 4.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Aventis Pharmaceuticals | Assay Description All rat alpha-1 adrenoceptor binding was performed by Hugo M. vargas, Karen M. Brooks and Lynn Laws-Ricker. | Chembiochem 3: 999-1009 (2002) Article DOI: 10.1002/1439-7633(20021004)3:10 BindingDB Entry DOI: 10.7270/Q27D2SP5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50434401 (CHEMBL2387314) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun... | Bioorg Med Chem Lett 23: 3416-20 (2013) Article DOI: 10.1016/j.bmcl.2013.03.080 BindingDB Entry DOI: 10.7270/Q2RB75Z5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50443222 (CHEMBL3087673) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from recombinant rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation... | Bioorg Med Chem Lett 23: 6269-73 (2013) Article DOI: 10.1016/j.bmcl.2013.09.081 BindingDB Entry DOI: 10.7270/Q27D2WK2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(4) dopamine receptor (Homo sapiens (Human)) | BDBM84448 (Isoindoline, 15) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 4.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Aventis Pharmaceuticals | Assay Description Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp. | Chembiochem 3: 999-1009 (2002) Article DOI: 10.1002/1439-7633(20021004)3:10 BindingDB Entry DOI: 10.7270/Q27D2SP5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50434400 (CHEMBL2387315) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun... | Bioorg Med Chem Lett 23: 3416-20 (2013) Article DOI: 10.1016/j.bmcl.2013.03.080 BindingDB Entry DOI: 10.7270/Q2RB75Z5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50443221 (CHEMBL3087668) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 4.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from recombinant rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation... | Bioorg Med Chem Lett 23: 6269-73 (2013) Article DOI: 10.1016/j.bmcl.2013.09.081 BindingDB Entry DOI: 10.7270/Q27D2WK2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50443220 (CHEMBL3087359) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from recombinant rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation... | Bioorg Med Chem Lett 23: 6269-73 (2013) Article DOI: 10.1016/j.bmcl.2013.09.081 BindingDB Entry DOI: 10.7270/Q27D2WK2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50443219 (CHEMBL3087672) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 4.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from recombinant rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation... | Bioorg Med Chem Lett 23: 6269-73 (2013) Article DOI: 10.1016/j.bmcl.2013.09.081 BindingDB Entry DOI: 10.7270/Q27D2WK2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(4) dopamine receptor (Homo sapiens (Human)) | BDBM84456 (Isoindoline, 23) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 5.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Aventis Pharmaceuticals | Assay Description Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp. | Chembiochem 3: 999-1009 (2002) Article DOI: 10.1002/1439-7633(20021004)3:10 BindingDB Entry DOI: 10.7270/Q27D2SP5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50434392 (CHEMBL2387285) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun... | Bioorg Med Chem Lett 23: 3416-20 (2013) Article DOI: 10.1016/j.bmcl.2013.03.080 BindingDB Entry DOI: 10.7270/Q2RB75Z5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50442631 (CHEMBL2441637) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 6.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from rhesus monkey histamine H3 receptor expressed in CHO cells | Bioorg Med Chem Lett 23: 6141-5 (2013) Article DOI: 10.1016/j.bmcl.2013.09.006 BindingDB Entry DOI: 10.7270/Q24T6KT6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50434387 (CHEMBL2387290) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun... | Bioorg Med Chem Lett 23: 3416-20 (2013) Article DOI: 10.1016/j.bmcl.2013.03.080 BindingDB Entry DOI: 10.7270/Q2RB75Z5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50442624 (CHEMBL2441635) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from rhesus monkey histamine H3 receptor expressed in CHO cells | Bioorg Med Chem Lett 23: 6141-5 (2013) Article DOI: 10.1016/j.bmcl.2013.09.006 BindingDB Entry DOI: 10.7270/Q24T6KT6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50442625 (CHEMBL2441643) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from rhesus monkey histamine H3 receptor expressed in CHO cells | Bioorg Med Chem Lett 23: 6141-5 (2013) Article DOI: 10.1016/j.bmcl.2013.09.006 BindingDB Entry DOI: 10.7270/Q24T6KT6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50437068 (CHEMBL2403549) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from recombinant rhesus monkey histamine H3 receptor transfected in CHO cell membranes after 1 hr by scin... | Bioorg Med Chem Lett 23: 4044-7 (2013) Article DOI: 10.1016/j.bmcl.2013.05.068 BindingDB Entry DOI: 10.7270/Q28C9XN0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50434388 (CHEMBL2387289) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 8.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun... | Bioorg Med Chem Lett 23: 3416-20 (2013) Article DOI: 10.1016/j.bmcl.2013.03.080 BindingDB Entry DOI: 10.7270/Q2RB75Z5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50442626 (CHEMBL2441642) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 8.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from rhesus monkey histamine H3 receptor expressed in CHO cells | Bioorg Med Chem Lett 23: 6141-5 (2013) Article DOI: 10.1016/j.bmcl.2013.09.006 BindingDB Entry DOI: 10.7270/Q24T6KT6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50442637 (CHEMBL2441658) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 8.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from rhesus monkey histamine H3 receptor expressed in CHO cells | Bioorg Med Chem Lett 23: 6141-5 (2013) Article DOI: 10.1016/j.bmcl.2013.09.006 BindingDB Entry DOI: 10.7270/Q24T6KT6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine receptor H3 (Macaca mulatta (Rhesus macaque)) | BDBM50442630 (CHEMBL2441638) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 9 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Curated by ChEMBL | Assay Description Displacement of [3H]N-alpha-methylhistamine from rhesus monkey histamine H3 receptor expressed in CHO cells | Bioorg Med Chem Lett 23: 6141-5 (2013) Article DOI: 10.1016/j.bmcl.2013.09.006 BindingDB Entry DOI: 10.7270/Q24T6KT6 | |||||||||||
More data for this Ligand-Target Pair |
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