Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122077 (CHEMBL153017 | N-[1-[5-(6-Amino-hexylamino)-pentyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 3.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-80 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122093 (CHEMBL152879 | N-[1-[4-(7-Amino-heptylamino)-butyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 38 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-80 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122084 (CHEMBL153996 | N-[1-[8-(3-Amino-propylamino)-octyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 64 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-80 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122090 (CHEMBL147182 | N-[1-[8-(3-Amino-propylamino)-octyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 65 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-80 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122096 (CHEMBL152410 | Hexanoic acid [1-[8-(3-amino-propyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 68 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-80 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122087 (CHEMBL153995 | Cyclohexanecarboxylic acid [1-[8-(3...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 78 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-80 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122085 (CHEMBL152425 | N-[1-[8-(3-Amino-propylamino)-octyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 88 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-80 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122086 (CHEMBL269192 | N-[1-[8-(3-Amino-propylamino)-octyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-80 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122095 (CHEMBL355977 | N-[8-(3-Amino-propylamino)-octyl]-3...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-80 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122091 (CHEMBL152736 | N-[1-[8-(3-Amino-propylamino)-octyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 110 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-80 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122092 (CHEMBL350228 | N-[8-(3-Amino-propylamino)-octyl]-3...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 110 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-80 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122094 (CHEMBL345521 | Pyridine-2-carboxylic acid [1-[8-(3...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 130 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-80 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122089 (CHEMBL352030 | N-[1-[8-(3-Amino-propylamino)-octyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 130 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-80 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122093 (CHEMBL152879 | N-[1-[4-(7-Amino-heptylamino)-butyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 135 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-40 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122086 (CHEMBL269192 | N-[1-[8-(3-Amino-propylamino)-octyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 140 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-40 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122078 (CHEMBL422515 | N-[1-[7-(4-Amino-butylamino)-heptyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | 168 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-80 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122091 (CHEMBL152736 | N-[1-[8-(3-Amino-propylamino)-octyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 170 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-40 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122094 (CHEMBL345521 | Pyridine-2-carboxylic acid [1-[8-(3...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 170 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-40 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122085 (CHEMBL152425 | N-[1-[8-(3-Amino-propylamino)-octyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 210 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-40 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122081 (2-Acetylamino-N-[8-(3-amino-propylamino)-octyl]-3-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 220 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-80 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122087 (CHEMBL153995 | Cyclohexanecarboxylic acid [1-[8-(3...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 240 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-40 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122083 (CHEMBL154012 | N-[1-[8-(3-Amino-propylamino)-octyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 250 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-80 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122089 (CHEMBL352030 | N-[1-[8-(3-Amino-propylamino)-octyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 250 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-40 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122092 (CHEMBL350228 | N-[8-(3-Amino-propylamino)-octyl]-3...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 250 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-40 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122083 (CHEMBL154012 | N-[1-[8-(3-Amino-propylamino)-octyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 254 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-40 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122095 (CHEMBL355977 | N-[8-(3-Amino-propylamino)-octyl]-3...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 280 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-40 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122077 (CHEMBL153017 | N-[1-[5-(6-Amino-hexylamino)-pentyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 287 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-40 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122081 (2-Acetylamino-N-[8-(3-amino-propylamino)-octyl]-3-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 300 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-40 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122084 (CHEMBL153996 | N-[1-[8-(3-Amino-propylamino)-octyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 330 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-40 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122079 (CHEMBL154184 | N-[2-[3-(8-Amino-octylamino)-propyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 350 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-80 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122082 (CHEMBL434273 | N-[1-[9-(2-Amino-ethylamino)-nonylc...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 410 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-80 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122080 (CHEMBL152153 | N-[1-[6-(5-Amino-pentylamino)-hexyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 468 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-80 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122096 (CHEMBL152410 | Hexanoic acid [1-[8-(3-amino-propyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-40 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122078 (CHEMBL422515 | N-[1-[7-(4-Amino-butylamino)-heptyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | 3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-40 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122082 (CHEMBL434273 | N-[1-[9-(2-Amino-ethylamino)-nonylc...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 6.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-40 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122090 (CHEMBL147182 | N-[1-[8-(3-Amino-propylamino)-octyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 8.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-40 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122079 (CHEMBL154184 | N-[2-[3-(8-Amino-octylamino)-propyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 8.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-40 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122080 (CHEMBL152153 | N-[1-[6-(5-Amino-pentylamino)-hexyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-40 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122088 (CHEMBL55975 | N-[1-{3-[4-(3-Amino-propylamino)-but...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 2.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-80 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor 1 (Homo sapiens (Human)) | BDBM50122088 (CHEMBL55975 | N-[1-{3-[4-(3-Amino-propylamino)-but...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 1.70E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Inhibition of the (-40 mV) current elicited by 100 microM glutamate by simultaneous co-application in xenopus oocytes injected with GluR1 flop RNA. | J Med Chem 45: 5745-54 (2002) BindingDB Entry DOI: 10.7270/Q2BP025P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 1 (Homo sapiens (Human)) | BDBM50329474 ((S)-N-(1-(3-(4-(3-aminopropylamino)butylamino)prop...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Antagonist activity at GluR1 expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced current at -60mV holding potential by tw... | J Med Chem 53: 7441-51 (2010) Article DOI: 10.1021/jm100886h BindingDB Entry DOI: 10.7270/Q2125SX4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 1 (Homo sapiens (Human)) | BDBM50329475 ((S)-N-(1-(3-(4-(3-aminopropylamino)butylamino)prop...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 21 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Antagonist activity at GluR1 expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced current at -60mV holding potential by tw... | J Med Chem 53: 7441-51 (2010) Article DOI: 10.1021/jm100886h BindingDB Entry DOI: 10.7270/Q2125SX4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 1 (Homo sapiens (Human)) | BDBM50094298 (CHEMBL16117 | N-[(S)-1-{3-[4-(3-Amino-propylamino)...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 23 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Antagonist activity at GluR1 expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced current at -60mV holding potential by tw... | J Med Chem 53: 7441-51 (2010) Article DOI: 10.1021/jm100886h BindingDB Entry DOI: 10.7270/Q2125SX4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 1 (Homo sapiens (Human)) | BDBM50329473 ((S)-N-(1-(3-(4-(3-aminopropylamino)butylamino)prop...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 32 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Antagonist activity at GluR1 expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced current at -60mV holding potential by tw... | J Med Chem 53: 7441-51 (2010) Article DOI: 10.1021/jm100886h BindingDB Entry DOI: 10.7270/Q2125SX4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 1 (Homo sapiens (Human)) | BDBM50329477 ((S)-N-(3-(4-(3-aminopropylamino)butylamino)propyl)...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 41 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Antagonist activity at GluR1 expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced current at -60mV holding potential by tw... | J Med Chem 53: 7441-51 (2010) Article DOI: 10.1021/jm100886h BindingDB Entry DOI: 10.7270/Q2125SX4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2A (Homo sapiens (Human)) | BDBM50329477 ((S)-N-(3-(4-(3-aminopropylamino)butylamino)propyl)...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 47 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Antagonist activity at NR1-1a/NR2A receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate/glycine-induced current at -60mV ... | J Med Chem 53: 7441-51 (2010) Article DOI: 10.1021/jm100886h BindingDB Entry DOI: 10.7270/Q2125SX4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 1 (Homo sapiens (Human)) | BDBM50329476 ((S)-N-(1-(3-(4-(3-aminopropylamino)butylamino)prop...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 87 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Antagonist activity at GluR1 expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced current at -60mV holding potential by tw... | J Med Chem 53: 7441-51 (2010) Article DOI: 10.1021/jm100886h BindingDB Entry DOI: 10.7270/Q2125SX4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 1 (Homo sapiens (Human)) | BDBM50329478 ((S)-2-(2-Adamantan-1-yl-acetylamino)-N-{3-[4-(3-am...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 105 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Antagonist activity at GluR1 expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced current at -60mV holding potential by tw... | J Med Chem 53: 7441-51 (2010) Article DOI: 10.1021/jm100886h BindingDB Entry DOI: 10.7270/Q2125SX4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2A (Homo sapiens (Human)) | BDBM50329480 ((S)-N-(20-amino-2,7-dioxo-1-phenyl-3,8,12,17-tetra...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 106 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Antagonist activity at NR1-1a/NR2A receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate/glycine-induced current at -60mV ... | J Med Chem 53: 7441-51 (2010) Article DOI: 10.1021/jm100886h BindingDB Entry DOI: 10.7270/Q2125SX4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine receptor subunit delta (Homo sapiens (Human)) | BDBM50111638 (CHEMBL16044 | N-[(S)-1-(11-Amino-undecylcarbamoyl)...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 460 | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Compound was evaluated for inhibitory activity against human embryonic muscle type Nicotinic acetylcholine receptor specifically delta-subunit expres... | Bioorg Med Chem Lett 12: 1159-62 (2002) BindingDB Entry DOI: 10.7270/Q2BC3XWG | |||||||||||
More data for this Ligand-Target Pair |
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