Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Kallikrein-2 (Homo sapiens (Human)) | BDBM50292533 (CHEMBL446790 | Fukugetin) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Campus Inc Curated by ChEMBL | Assay Description Mixed-type inhibition of human tissue kallikrein-2 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate preincubated fo... | Bioorg Med Chem Lett 26: 1485-9 (2016) Article DOI: 10.1016/j.bmcl.2016.01.039 BindingDB Entry DOI: 10.7270/Q2862J9K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-7 (Homo sapiens (Human)) | BDBM50391075 (CHEMBL2087343) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Tri£ngulo Mineiro Curated by ChEMBL | Assay Description Competitive inhibition of recombinant human KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysis | Bioorg Med Chem Lett 22: 6072-5 (2012) Article DOI: 10.1016/j.bmcl.2012.08.047 BindingDB Entry DOI: 10.7270/Q2SF2X8R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-7 (Homo sapiens (Human)) | BDBM50391078 (CHEMBL2087346) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Tri£ngulo Mineiro Curated by ChEMBL | Assay Description Competitive inhibition of recombinant human KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysis | Bioorg Med Chem Lett 22: 6072-5 (2012) Article DOI: 10.1016/j.bmcl.2012.08.047 BindingDB Entry DOI: 10.7270/Q2SF2X8R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-1 (Homo sapiens (Human)) | BDBM50292533 (CHEMBL446790 | Fukugetin) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Campus Inc Curated by ChEMBL | Assay Description Mixed-type inhibition of human tissue kallikrein-1 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate preincubated fo... | Bioorg Med Chem Lett 26: 1485-9 (2016) Article DOI: 10.1016/j.bmcl.2016.01.039 BindingDB Entry DOI: 10.7270/Q2862J9K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-7 (Homo sapiens (Human)) | BDBM50355086 (CHEMBL1834753) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.22E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Tri£ngulo Mineiro Curated by ChEMBL | Assay Description Inhibition of human kallikrein 7 using Abz-KLYSSKQ-EDDnp as substrate by Lineweaver-Burk plot analysis | Bioorg Med Chem Lett 21: 6112-5 (2011) Article DOI: 10.1016/j.bmcl.2011.08.044 BindingDB Entry DOI: 10.7270/Q24M94ZP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-5 [D153N] (Homo sapiens (Human)) | BDBM50355088 (CHEMBL1834754) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.29E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Tri£ngulo Mineiro Curated by ChEMBL | Assay Description Inhibition of human kallikrein 5 using Abz-KLRSSKQ-EDDnp as substrate by Lineweaver-Burk plot analysis | Bioorg Med Chem Lett 21: 6112-5 (2011) Article DOI: 10.1016/j.bmcl.2011.08.044 BindingDB Entry DOI: 10.7270/Q24M94ZP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-5 [D153N] (Homo sapiens (Human)) | BDBM50355086 (CHEMBL1834753) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.44E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Tri£ngulo Mineiro Curated by ChEMBL | Assay Description Inhibition of human kallikrein 5 using Abz-KLRSSKQ-EDDnp as substrate by Lineweaver-Burk plot analysis | Bioorg Med Chem Lett 21: 6112-5 (2011) Article DOI: 10.1016/j.bmcl.2011.08.044 BindingDB Entry DOI: 10.7270/Q24M94ZP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-7 (Homo sapiens (Human)) | BDBM50355088 (CHEMBL1834754) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.72E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Tri£ngulo Mineiro Curated by ChEMBL | Assay Description Inhibition of human kallikrein 7 using Abz-KLYSSKQ-EDDnp as substrate by Lineweaver-Burk plot analysis | Bioorg Med Chem Lett 21: 6112-5 (2011) Article DOI: 10.1016/j.bmcl.2011.08.044 BindingDB Entry DOI: 10.7270/Q24M94ZP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-5 [D153N] (Homo sapiens (Human)) | BDBM50355087 (CHEMBL1833982) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.75E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Tri£ngulo Mineiro Curated by ChEMBL | Assay Description Inhibition of human kallikrein 5 using Abz-KLRSSKQ-EDDnp as substrate by Lineweaver-Burk plot analysis | Bioorg Med Chem Lett 21: 6112-5 (2011) Article DOI: 10.1016/j.bmcl.2011.08.044 BindingDB Entry DOI: 10.7270/Q24M94ZP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-5 [D153N] (Homo sapiens (Human)) | BDBM50391078 (CHEMBL2087346) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 7.04E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Tri£ngulo Mineiro Curated by ChEMBL | Assay Description Competitive inhibition of human KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysis | Bioorg Med Chem Lett 22: 6072-5 (2012) Article DOI: 10.1016/j.bmcl.2012.08.047 BindingDB Entry DOI: 10.7270/Q2SF2X8R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-5 [D153N] (Homo sapiens (Human)) | BDBM50391075 (CHEMBL2087343) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7.07E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Tri£ngulo Mineiro Curated by ChEMBL | Assay Description Competitive inhibition of human KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysis | Bioorg Med Chem Lett 22: 6072-5 (2012) Article DOI: 10.1016/j.bmcl.2012.08.047 BindingDB Entry DOI: 10.7270/Q2SF2X8R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-7 (Homo sapiens (Human)) | BDBM50355087 (CHEMBL1833982) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7.07E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Tri£ngulo Mineiro Curated by ChEMBL | Assay Description Inhibition of human kallikrein 7 using Abz-KLYSSKQ-EDDnp as substrate by Lineweaver-Burk plot analysis | Bioorg Med Chem Lett 21: 6112-5 (2011) Article DOI: 10.1016/j.bmcl.2011.08.044 BindingDB Entry DOI: 10.7270/Q24M94ZP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-5 [D153N] (Homo sapiens (Human)) | BDBM50391079 (CHEMBL2087347) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7.19E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Tri£ngulo Mineiro Curated by ChEMBL | Assay Description Competitive inhibition of human KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysis | Bioorg Med Chem Lett 22: 6072-5 (2012) Article DOI: 10.1016/j.bmcl.2012.08.047 BindingDB Entry DOI: 10.7270/Q2SF2X8R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-7 (Homo sapiens (Human)) | BDBM50391077 (CHEMBL2087345) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 7.51E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Tri£ngulo Mineiro Curated by ChEMBL | Assay Description Competitive inhibition of recombinant human KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysis | Bioorg Med Chem Lett 22: 6072-5 (2012) Article DOI: 10.1016/j.bmcl.2012.08.047 BindingDB Entry DOI: 10.7270/Q2SF2X8R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-7 (Homo sapiens (Human)) | BDBM50391079 (CHEMBL2087347) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7.74E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Tri£ngulo Mineiro Curated by ChEMBL | Assay Description Competitive inhibition of recombinant human KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysis | Bioorg Med Chem Lett 22: 6072-5 (2012) Article DOI: 10.1016/j.bmcl.2012.08.047 BindingDB Entry DOI: 10.7270/Q2SF2X8R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-7 (Homo sapiens (Human)) | BDBM50391076 (CHEMBL2087344) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 8.03E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Tri£ngulo Mineiro Curated by ChEMBL | Assay Description Competitive inhibition of recombinant human KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysis | Bioorg Med Chem Lett 22: 6072-5 (2012) Article DOI: 10.1016/j.bmcl.2012.08.047 BindingDB Entry DOI: 10.7270/Q2SF2X8R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-5 [D153N] (Homo sapiens (Human)) | BDBM50391077 (CHEMBL2087345) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 2.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Tri£ngulo Mineiro Curated by ChEMBL | Assay Description Competitive inhibition of human KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysis | Bioorg Med Chem Lett 22: 6072-5 (2012) Article DOI: 10.1016/j.bmcl.2012.08.047 BindingDB Entry DOI: 10.7270/Q2SF2X8R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-5 [D153N] (Homo sapiens (Human)) | BDBM50391076 (CHEMBL2087344) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 3.57E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Tri£ngulo Mineiro Curated by ChEMBL | Assay Description Competitive inhibition of human KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysis | Bioorg Med Chem Lett 22: 6072-5 (2012) Article DOI: 10.1016/j.bmcl.2012.08.047 BindingDB Entry DOI: 10.7270/Q2SF2X8R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-2 (Homo sapiens (Human)) | BDBM50292533 (CHEMBL446790 | Fukugetin) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Campus Inc Curated by ChEMBL | Assay Description Inhibition of human tissue kallikrein-2 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate preincubated for 10 mins f... | Bioorg Med Chem Lett 26: 1485-9 (2016) Article DOI: 10.1016/j.bmcl.2016.01.039 BindingDB Entry DOI: 10.7270/Q2862J9K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-1 (Homo sapiens (Human)) | BDBM50292533 (CHEMBL446790 | Fukugetin) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Campus Inc Curated by ChEMBL | Assay Description Inhibition of human tissue kallikrein-1 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate preincubated for 10 mins f... | Bioorg Med Chem Lett 26: 1485-9 (2016) Article DOI: 10.1016/j.bmcl.2016.01.039 BindingDB Entry DOI: 10.7270/Q2862J9K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-5 [D153N] (Homo sapiens (Human)) | BDBM50292533 (CHEMBL446790 | Fukugetin) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.25E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Campus Inc Curated by ChEMBL | Assay Description Inhibition of human tissue kallikrein-5 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate preincubated for 10 mins f... | Bioorg Med Chem Lett 26: 1485-9 (2016) Article DOI: 10.1016/j.bmcl.2016.01.039 BindingDB Entry DOI: 10.7270/Q2862J9K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostate-specific antigen (Homo sapiens (Human)) | BDBM50292533 (CHEMBL446790 | Fukugetin) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Campus Inc Curated by ChEMBL | Assay Description Inhibition of human tissue kallikrein-3 expressed in baculovirus infected insect cells using Abz-KLYSSQ-EDDnp as substrate preincubated for 10 mins f... | Bioorg Med Chem Lett 26: 1485-9 (2016) Article DOI: 10.1016/j.bmcl.2016.01.039 BindingDB Entry DOI: 10.7270/Q2862J9K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-7 (Homo sapiens (Human)) | BDBM50391075 (CHEMBL2087343) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.33E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Tri£ngulo Mineiro Curated by ChEMBL | Assay Description Inhibition of human recombinant KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysis | Bioorg Med Chem Lett 22: 6072-5 (2012) Article DOI: 10.1016/j.bmcl.2012.08.047 BindingDB Entry DOI: 10.7270/Q2SF2X8R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-6 (Homo sapiens (Human)) | BDBM50292533 (CHEMBL446790 | Fukugetin) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.35E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Campus Inc Curated by ChEMBL | Assay Description Inhibition of human tissue kallikrein-6 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate preincubated for 10 mins f... | Bioorg Med Chem Lett 26: 1485-9 (2016) Article DOI: 10.1016/j.bmcl.2016.01.039 BindingDB Entry DOI: 10.7270/Q2862J9K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-7 (Homo sapiens (Human)) | BDBM50292533 (CHEMBL446790 | Fukugetin) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Campus Inc Curated by ChEMBL | Assay Description Inhibition of human tissue kallikrein-7 expressed in baculovirus infected insect cells using Abz-KLYSSQ-EDDnp as substrate preincubated for 10 mins f... | Bioorg Med Chem Lett 26: 1485-9 (2016) Article DOI: 10.1016/j.bmcl.2016.01.039 BindingDB Entry DOI: 10.7270/Q2862J9K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-7 (Homo sapiens (Human)) | BDBM50391078 (CHEMBL2087346) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.63E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Tri£ngulo Mineiro Curated by ChEMBL | Assay Description Inhibition of human recombinant KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysis | Bioorg Med Chem Lett 22: 6072-5 (2012) Article DOI: 10.1016/j.bmcl.2012.08.047 BindingDB Entry DOI: 10.7270/Q2SF2X8R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-5 [D153N] (Homo sapiens (Human)) | BDBM50355088 (CHEMBL1834754) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.37E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Tri£ngulo Mineiro Curated by ChEMBL | Assay Description Inhibition of human kallikrein 5 using Abz-KLRSSKQ-EDDnp as substrate by spectrofluorimetric assay | Bioorg Med Chem Lett 21: 6112-5 (2011) Article DOI: 10.1016/j.bmcl.2011.08.044 BindingDB Entry DOI: 10.7270/Q24M94ZP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-5 [D153N] (Homo sapiens (Human)) | BDBM50355086 (CHEMBL1834753) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.29E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Tri£ngulo Mineiro Curated by ChEMBL | Assay Description Inhibition of human kallikrein 5 using Abz-KLRSSKQ-EDDnp as substrate by spectrofluorimetric assay | Bioorg Med Chem Lett 21: 6112-5 (2011) Article DOI: 10.1016/j.bmcl.2011.08.044 BindingDB Entry DOI: 10.7270/Q24M94ZP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-5 [D153N] (Homo sapiens (Human)) | BDBM50391078 (CHEMBL2087346) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 9.91E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Tri£ngulo Mineiro Curated by ChEMBL | Assay Description Inhibition of human recombinant KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysis | Bioorg Med Chem Lett 22: 6072-5 (2012) Article DOI: 10.1016/j.bmcl.2012.08.047 BindingDB Entry DOI: 10.7270/Q2SF2X8R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-5 [D153N] (Homo sapiens (Human)) | BDBM50391075 (CHEMBL2087343) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.92E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Tri£ngulo Mineiro Curated by ChEMBL | Assay Description Inhibition of human recombinant KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysis | Bioorg Med Chem Lett 22: 6072-5 (2012) Article DOI: 10.1016/j.bmcl.2012.08.047 BindingDB Entry DOI: 10.7270/Q2SF2X8R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-5 [D153N] (Homo sapiens (Human)) | BDBM50391079 (CHEMBL2087347) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.01E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Tri£ngulo Mineiro Curated by ChEMBL | Assay Description Inhibition of human recombinant KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysis | Bioorg Med Chem Lett 22: 6072-5 (2012) Article DOI: 10.1016/j.bmcl.2012.08.047 BindingDB Entry DOI: 10.7270/Q2SF2X8R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-7 (Homo sapiens (Human)) | BDBM50355086 (CHEMBL1834753) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.12E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Tri£ngulo Mineiro Curated by ChEMBL | Assay Description Inhibition of human kallikrein 7 using Abz-KLYSSKQ-EDDnp as substrate by spectrofluorimetric assay | Bioorg Med Chem Lett 21: 6112-5 (2011) Article DOI: 10.1016/j.bmcl.2011.08.044 BindingDB Entry DOI: 10.7270/Q24M94ZP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-7 (Homo sapiens (Human)) | BDBM50355088 (CHEMBL1834754) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.35E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Tri£ngulo Mineiro Curated by ChEMBL | Assay Description Inhibition of human kallikrein 7 using Abz-KLYSSKQ-EDDnp as substrate by spectrofluorimetric assay | Bioorg Med Chem Lett 21: 6112-5 (2011) Article DOI: 10.1016/j.bmcl.2011.08.044 BindingDB Entry DOI: 10.7270/Q24M94ZP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-7 (Homo sapiens (Human)) | BDBM50391079 (CHEMBL2087347) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.61E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Tri£ngulo Mineiro Curated by ChEMBL | Assay Description Inhibition of human recombinant KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysis | Bioorg Med Chem Lett 22: 6072-5 (2012) Article DOI: 10.1016/j.bmcl.2012.08.047 BindingDB Entry DOI: 10.7270/Q2SF2X8R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-7 (Homo sapiens (Human)) | BDBM50355087 (CHEMBL1833982) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.66E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Tri£ngulo Mineiro Curated by ChEMBL | Assay Description Inhibition of human kallikrein 7 using Abz-KLYSSKQ-EDDnp as substrate by spectrofluorimetric assay | Bioorg Med Chem Lett 21: 6112-5 (2011) Article DOI: 10.1016/j.bmcl.2011.08.044 BindingDB Entry DOI: 10.7270/Q24M94ZP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-7 (Homo sapiens (Human)) | BDBM50391077 (CHEMBL2087345) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.96E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Tri£ngulo Mineiro Curated by ChEMBL | Assay Description Inhibition of human recombinant KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysis | Bioorg Med Chem Lett 22: 6072-5 (2012) Article DOI: 10.1016/j.bmcl.2012.08.047 BindingDB Entry DOI: 10.7270/Q2SF2X8R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-7 (Homo sapiens (Human)) | BDBM50391076 (CHEMBL2087344) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.05E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Tri£ngulo Mineiro Curated by ChEMBL | Assay Description Inhibition of human recombinant KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysis | Bioorg Med Chem Lett 22: 6072-5 (2012) Article DOI: 10.1016/j.bmcl.2012.08.047 BindingDB Entry DOI: 10.7270/Q2SF2X8R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-5 [D153N] (Homo sapiens (Human)) | BDBM50391077 (CHEMBL2087345) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.24E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Tri£ngulo Mineiro Curated by ChEMBL | Assay Description Inhibition of human recombinant KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysis | Bioorg Med Chem Lett 22: 6072-5 (2012) Article DOI: 10.1016/j.bmcl.2012.08.047 BindingDB Entry DOI: 10.7270/Q2SF2X8R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-5 [D153N] (Homo sapiens (Human)) | BDBM50355087 (CHEMBL1833982) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.67E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Tri£ngulo Mineiro Curated by ChEMBL | Assay Description Inhibition of human kallikrein 5 using Abz-KLRSSKQ-EDDnp as substrate by spectrofluorimetric assay | Bioorg Med Chem Lett 21: 6112-5 (2011) Article DOI: 10.1016/j.bmcl.2011.08.044 BindingDB Entry DOI: 10.7270/Q24M94ZP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-5 [D153N] (Homo sapiens (Human)) | BDBM50391076 (CHEMBL2087344) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Tri£ngulo Mineiro Curated by ChEMBL | Assay Description Inhibition of human recombinant KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysis | Bioorg Med Chem Lett 22: 6072-5 (2012) Article DOI: 10.1016/j.bmcl.2012.08.047 BindingDB Entry DOI: 10.7270/Q2SF2X8R | |||||||||||
More data for this Ligand-Target Pair |