Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Heterogeneous nuclear ribonucleoprotein A1 (Homo sapiens (Human)) | BDBM50008923 ((S)-4-ethyl-4-hydroxy-1,12-dihydro-4H-2-oxa-6,12a-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | 82.7 | n/a | n/a | n/a | n/a | n/a |
Tokyo University of Science Curated by ChEMBL | Assay Description Binding affinity to recombinant GST-tagged human hnRNP A1 expressed in Escherichia coli using QCM biosensor by Scatchard plot analysis | Bioorg Med Chem 19: 7690-7 (2011) Article DOI: 10.1016/j.bmc.2011.09.059 BindingDB Entry DOI: 10.7270/Q2WW7J55 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
GRB10-interacting GYF protein 2 (Homo sapiens (Human)) | BDBM50428560 (CHEMBL2337520) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 186 | n/a | n/a | n/a | n/a | n/a |
Tokyo University of Science Curated by ChEMBL | Assay Description Binding affinity to recombinant His-tagged Grb10 interacting GYF protein 2 (745-1030 amino acids) (unknown origin) by surface plasmon resonance analy... | Bioorg Med Chem 21: 311-20 (2012) Article DOI: 10.1016/j.bmc.2012.10.037 BindingDB Entry DOI: 10.7270/Q2KK9D5C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fanconi anemia group F protein (Homo sapiens (Human)) | BDBM50394323 (CHEMBL2159398) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 530 | n/a | n/a | n/a | n/a | n/a |
Tokyo University of Science Curated by ChEMBL | Assay Description Binding affinity to human thymus flag-tagged full-length FANCF expressed in HEK293T cells assessed as dissociation constant by surface plasmon resona... | Bioorg Med Chem 20: 6248-55 (2012) Article DOI: 10.1016/j.bmc.2012.09.015 BindingDB Entry DOI: 10.7270/Q2NK3G43 | |||||||||||
More data for this Ligand-Target Pair |