BindingDB PrimarySearch

Found 501 hits with Last Name = 'macchiarulo' and Initial = 'a'
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Mineralocorticoid receptor (Homo sapiens (Human))	BDBM21725 ((1S,2R,10R,11S,14Z,15S)-14-ethylidene-2,15-dimethy...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase PC cid PC sid UniChem Similars	Article PubMed	37	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Perugia Curated by ChEMBL					Assay Description Inhibitory concentration against Mineralocorticoid receptor				J Med Chem 48: 6948-55 (2005) Article DOI: 10.1021/jm0505056 BindingDB Entry DOI: 10.7270/Q20V8DKV
Universit£ di Perugia Curated by ChEMBL					More data for this Ligand-Target Pair
Mineralocorticoid receptor (Homo sapiens (Human))	BDBM50226465 (CHEMBL402063 \| E-guggulsterone \| pregna-4,17(20)-c...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	39	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Perugia Curated by ChEMBL					Assay Description Inhibitory concentration against Mineralocorticoid receptor				J Med Chem 48: 6948-55 (2005) Article DOI: 10.1021/jm0505056 BindingDB Entry DOI: 10.7270/Q20V8DKV
Universit£ di Perugia Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 2 (Homo sapiens (Human))	BDBM50107108 ((1S,2S,3R)-2-(Amino-carboxy-methyl)-3-[2-(9H-xanth...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	85	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Perugia Curated by ChEMBL					Assay Description Antagonistic activity against stimulation of GTP (gamma) 35 S binding by glutamate in membranes from CHO cells expressing human Metabotropic glutamat...				Bioorg Med Chem Lett 11: 3179-82 (2001) BindingDB Entry DOI: 10.7270/Q27M08H1
Universit£ di Perugia Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50007548 ((S)-2-Amino-4-phosphono-butyric acid \| (S)-2-amino...) Show SMILES N[C@@H](CCP(O)(O)=O)C(O)=O \|r\| Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars	Article PubMed	160	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Salerno Curated by ChEMBL					Assay Description Displacement of [3H]Quisqualate from human mGluR4 receptor expressed in BHK cells				Bioorg Med Chem 17: 242-50 (2008) Article DOI: 10.1016/j.bmc.2008.11.015 BindingDB Entry DOI: 10.7270/Q2HD7WKF
Universit£ di Salerno Curated by ChEMBL					More data for this Ligand-Target Pair
Progesterone receptor (Homo sapiens (Human))	BDBM50226465 (CHEMBL402063 \| E-guggulsterone \| pregna-4,17(20)-c...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	201	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Perugia Curated by ChEMBL					Assay Description Inhibitory concentration against Progesterone receptor				J Med Chem 48: 6948-55 (2005) Article DOI: 10.1021/jm0505056 BindingDB Entry DOI: 10.7270/Q20V8DKV
Universit£ di Perugia Curated by ChEMBL					More data for this Ligand-Target Pair
Progesterone receptor (Homo sapiens (Human))	BDBM21725 ((1S,2R,10R,11S,14Z,15S)-14-ethylidene-2,15-dimethy...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase PC cid PC sid UniChem Similars	Article PubMed	224	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Perugia Curated by ChEMBL					Assay Description Inhibitory concentration against Progesterone receptor				J Med Chem 48: 6948-55 (2005) Article DOI: 10.1021/jm0505056 BindingDB Entry DOI: 10.7270/Q20V8DKV
Universit£ di Perugia Curated by ChEMBL					More data for this Ligand-Target Pair
Glucocorticoid receptor (Homo sapiens (Human))	BDBM50226465 (CHEMBL402063 \| E-guggulsterone \| pregna-4,17(20)-c...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	224	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Perugia Curated by ChEMBL					Assay Description Inhibitory concentration against Glucorticoid receptor				J Med Chem 48: 6948-55 (2005) Article DOI: 10.1021/jm0505056 BindingDB Entry DOI: 10.7270/Q20V8DKV
Universit£ di Perugia Curated by ChEMBL					More data for this Ligand-Target Pair
Androgen receptor (Homo sapiens (Human))	BDBM50226465 (CHEMBL402063 \| E-guggulsterone \| pregna-4,17(20)-c...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	240	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Perugia Curated by ChEMBL					Assay Description Inhibitory concentration against Androgen receptor				J Med Chem 48: 6948-55 (2005) Article DOI: 10.1021/jm0505056 BindingDB Entry DOI: 10.7270/Q20V8DKV
Universit£ di Perugia Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 1 (Homo sapiens (Human))	BDBM17657 ((2S)-2-aminopentanedioic acid \| (S)-Glu \| D-Glutam...) Show SMILES N[C@@H](CCC(O)=O)C(O)=O Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars	Article PubMed	250	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Perugia Curated by ChEMBL					Assay Description Displacement of [3H]quisqualate from mGluR1 receptor expressed in BHK cells				J Med Chem 50: 4630-41 (2007) Article DOI: 10.1021/jm070322e BindingDB Entry DOI: 10.7270/Q2DF6S12
Universit£ di Perugia Curated by ChEMBL					More data for this Ligand-Target Pair
Glucocorticoid receptor (Homo sapiens (Human))	BDBM21725 ((1S,2R,10R,11S,14Z,15S)-14-ethylidene-2,15-dimethy...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase PC cid PC sid UniChem Similars	Article PubMed	252	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Perugia Curated by ChEMBL					Assay Description Inhibitory concentration against Glucorticoid receptor				J Med Chem 48: 6948-55 (2005) Article DOI: 10.1021/jm0505056 BindingDB Entry DOI: 10.7270/Q20V8DKV
Universit£ di Perugia Curated by ChEMBL					More data for this Ligand-Target Pair
Androgen receptor (Homo sapiens (Human))	BDBM21725 ((1S,2R,10R,11S,14Z,15S)-14-ethylidene-2,15-dimethy...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase PC cid PC sid UniChem Similars	Article PubMed	315	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Perugia Curated by ChEMBL					Assay Description Inhibitory concentration against Androgen receptor				J Med Chem 48: 6948-55 (2005) Article DOI: 10.1021/jm0505056 BindingDB Entry DOI: 10.7270/Q20V8DKV
Universit£ di Perugia Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 5 (Homo sapiens (Human))	BDBM17657 ((2S)-2-aminopentanedioic acid \| (S)-Glu \| D-Glutam...) Show SMILES N[C@@H](CCC(O)=O)C(O)=O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars	Article PubMed	390	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Perugia Curated by ChEMBL					Assay Description Binding affinity to mGluR5 receptor expressed in BHK cells				J Med Chem 50: 4630-41 (2007) Article DOI: 10.1021/jm070322e BindingDB Entry DOI: 10.7270/Q2DF6S12
Universit£ di Perugia Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 1 (Homo sapiens (Human))	BDBM17657 ((2S)-2-aminopentanedioic acid \| (S)-Glu \| D-Glutam...) Show SMILES N[C@@H](CCC(O)=O)C(O)=O Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars	Article PubMed	570	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Salerno Curated by ChEMBL					Assay Description Displacement of [3H]Quisqualate from human mGluR1A receptor expressed in BHK cells				Bioorg Med Chem 17: 242-50 (2008) Article DOI: 10.1016/j.bmc.2008.11.015 BindingDB Entry DOI: 10.7270/Q2HD7WKF
Universit£ di Salerno Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 5 (Homo sapiens (Human))	BDBM17657 ((2S)-2-aminopentanedioic acid \| (S)-Glu \| D-Glutam...) Show SMILES N[C@@H](CCC(O)=O)C(O)=O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars	Article PubMed	1.16E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Salerno Curated by ChEMBL					Assay Description Displacement of [3H]Quisqualate from human mGluR5 receptor expressed in BHK cells				Bioorg Med Chem 17: 242-50 (2008) Article DOI: 10.1016/j.bmc.2008.11.015 BindingDB Entry DOI: 10.7270/Q2HD7WKF
Universit£ di Salerno Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM17657 ((2S)-2-aminopentanedioic acid \| (S)-Glu \| D-Glutam...) Show SMILES N[C@@H](CCC(O)=O)C(O)=O Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars	Article PubMed	1.40E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Salerno Curated by ChEMBL					Assay Description Displacement of [3H]Quisqualate from human mGluR4 receptor expressed in BHK cells				Bioorg Med Chem 17: 242-50 (2008) Article DOI: 10.1016/j.bmc.2008.11.015 BindingDB Entry DOI: 10.7270/Q2HD7WKF
Universit£ di Salerno Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM17657 ((2S)-2-aminopentanedioic acid \| (S)-Glu \| D-Glutam...) Show SMILES N[C@@H](CCC(O)=O)C(O)=O Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars	Article PubMed	2.40E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Perugia Curated by ChEMBL					Assay Description Displacement of [3H]LAP4 from mGluR4 receptor expressed in BHK cells				J Med Chem 50: 4630-41 (2007) Article DOI: 10.1021/jm070322e BindingDB Entry DOI: 10.7270/Q2DF6S12
Universit£ di Perugia Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 2 (Homo sapiens (Human))	BDBM50107109 ((1S,2S,3R)-2-(Amino-carboxy-methyl)-3-(9H-xanthen-...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	2.70E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Perugia Curated by ChEMBL					Assay Description Antagonistic activity against stimulation of GTP (gamma) 35 S binding by glutamate in membranes from CHO cells expressing human Metabotropic glutamat...				Bioorg Med Chem Lett 11: 3179-82 (2001) BindingDB Entry DOI: 10.7270/Q27M08H1
Universit£ di Perugia Curated by ChEMBL					More data for this Ligand-Target Pair
Bile acid receptor (Homo sapiens (Human))	BDBM21725 ((1S,2R,10R,11S,14Z,15S)-14-ethylidene-2,15-dimethy...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase PC cid PC sid UniChem Similars	Article PubMed	>5.00E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Perugia Curated by ChEMBL					Assay Description Inhibitory concentration against Farnesoid X receptor				J Med Chem 48: 6948-55 (2005) Article DOI: 10.1021/jm0505056 BindingDB Entry DOI: 10.7270/Q20V8DKV
Universit£ di Perugia Curated by ChEMBL					More data for this Ligand-Target Pair
Bile acid receptor (Homo sapiens (Human))	BDBM50226465 (CHEMBL402063 \| E-guggulsterone \| pregna-4,17(20)-c...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	>5.00E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Perugia Curated by ChEMBL					Assay Description Inhibitory concentration against Farnesoid X receptor				J Med Chem 48: 6948-55 (2005) Article DOI: 10.1021/jm0505056 BindingDB Entry DOI: 10.7270/Q20V8DKV
Universit£ di Perugia Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 2 (Homo sapiens (Human))	BDBM17657 ((2S)-2-aminopentanedioic acid \| (S)-Glu \| D-Glutam...) Show SMILES N[C@@H](CCC(O)=O)C(O)=O Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars	Article PubMed	6.40E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Salerno Curated by ChEMBL					Assay Description Displacement of [3H]Quisqualate from human mGluR2 receptor expressed in BHK cells				Bioorg Med Chem 17: 242-50 (2008) Article DOI: 10.1016/j.bmc.2008.11.015 BindingDB Entry DOI: 10.7270/Q2HD7WKF
Universit£ di Salerno Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 2 (Homo sapiens (Human))	BDBM17657 ((2S)-2-aminopentanedioic acid \| (S)-Glu \| D-Glutam...) Show SMILES N[C@@H](CCC(O)=O)C(O)=O Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars	Article PubMed	1.10E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Perugia Curated by ChEMBL					Assay Description Displacement of [3H]LY341495 from mGluR2 receptor expressed in BHK cells				J Med Chem 50: 4630-41 (2007) Article DOI: 10.1021/jm070322e BindingDB Entry DOI: 10.7270/Q2DF6S12
Universit£ di Perugia Curated by ChEMBL					More data for this Ligand-Target Pair
Aryl hydrocarbon receptor (Homo sapiens (Human))	BDBM50506041 (CHEBI:16946 \| L-kynurenine) Show SMILES N[C@@H](CC(=O)c1ccccc1N)C(O)=O Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase MCE KEGG PC cid PC sid UniChem	Article PubMed	2.16E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
University of Perugia Curated by ChEMBL					Assay Description Inhibition of AhR (unknown origin)				Eur J Med Chem 185: (2020) Article DOI: 10.1016/j.ejmech.2019.111842 BindingDB Entry DOI: 10.7270/Q2N019SX
University of Perugia Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 1 (Homo sapiens (Human))	BDBM50220148 ((2S,1'R,2'S)-2-(2'-sulfonocyclopropyl)glycine \| CH...) Show SMILES N[C@@H]([C@H]1C[C@@H]1S(O)(=O)=O)C(O)=O Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	3.40E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Perugia Curated by ChEMBL					Assay Description Displacement of [3H]quisqualate from mGluR1 receptor expressed in BHK cells				J Med Chem 50: 4630-41 (2007) Article DOI: 10.1021/jm070322e BindingDB Entry DOI: 10.7270/Q2DF6S12
Universit£ di Perugia Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 5 (Homo sapiens (Human))	BDBM50220148 ((2S,1'R,2'S)-2-(2'-sulfonocyclopropyl)glycine \| CH...) Show SMILES N[C@@H]([C@H]1C[C@@H]1S(O)(=O)=O)C(O)=O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	4.90E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Perugia Curated by ChEMBL					Assay Description Binding affinity to mGluR5 receptor expressed in BHK cells				J Med Chem 50: 4630-41 (2007) Article DOI: 10.1021/jm070322e BindingDB Entry DOI: 10.7270/Q2DF6S12
Universit£ di Perugia Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50220147 ((S)-2-amino-4-sulfobutanoic acid \| CHEMBL230951 \| ...) Show SMILES N[C@@H](CCS(O)(=O)=O)C(O)=O \|r\| Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE KEGG PC cid PC sid PDB UniChem Patents Similars	Article PubMed	5.30E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Perugia Curated by ChEMBL					Assay Description Displacement of [3H]LAP4 from mGluR4 receptor expressed in BHK cells				J Med Chem 50: 4630-41 (2007) Article DOI: 10.1021/jm070322e BindingDB Entry DOI: 10.7270/Q2DF6S12
Universit£ di Perugia Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 5 (Homo sapiens (Human))	BDBM50220147 ((S)-2-amino-4-sulfobutanoic acid \| CHEMBL230951 \| ...) Show SMILES N[C@@H](CCS(O)(=O)=O)C(O)=O \|r\| Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE KEGG PC cid PC sid PDB UniChem Patents Similars	Article PubMed	5.40E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Perugia Curated by ChEMBL					Assay Description Binding affinity to mGluR5 receptor expressed in BHK cells				J Med Chem 50: 4630-41 (2007) Article DOI: 10.1021/jm070322e BindingDB Entry DOI: 10.7270/Q2DF6S12
Universit£ di Perugia Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 5 (Homo sapiens (Human))	BDBM50220154 ((2R,1'R,2'R)-2-(2'-sulfonocyclopropyl)glycine \| CH...) Show SMILES N[C@H]([C@H]1C[C@H]1S(O)(=O)=O)C(O)=O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	5.50E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Perugia Curated by ChEMBL					Assay Description Binding affinity to mGluR5 receptor expressed in BHK cells				J Med Chem 50: 4630-41 (2007) Article DOI: 10.1021/jm070322e BindingDB Entry DOI: 10.7270/Q2DF6S12
Universit£ di Perugia Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 1 (Homo sapiens (Human))	BDBM50254389 ((2S)-2-(3'-Carboxymethylbicyclo[1.1.1]pentyl)glyci...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	5.90E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Salerno Curated by ChEMBL					Assay Description Displacement of [3H]Quisqualate from human mGluR1A receptor expressed in BHK cells				Bioorg Med Chem 17: 242-50 (2008) Article DOI: 10.1016/j.bmc.2008.11.015 BindingDB Entry DOI: 10.7270/Q2HD7WKF
Universit£ di Salerno Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 5 (Homo sapiens (Human))	BDBM50220150 ((2R,1'S,2'R)-2-(2'-sulfonocyclopropyl)glycine \| CH...) Show SMILES N[C@H]([C@@H]1C[C@H]1S(O)(=O)=O)C(O)=O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	6.70E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Perugia Curated by ChEMBL					Assay Description Binding affinity to mGluR5 receptor expressed in BHK cells				J Med Chem 50: 4630-41 (2007) Article DOI: 10.1021/jm070322e BindingDB Entry DOI: 10.7270/Q2DF6S12
Universit£ di Perugia Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 1 (Homo sapiens (Human))	BDBM50220149 ((2S,1'S,2'R)-2-(2'-sulfonocyclopropyl)glycine \| CH...) Show SMILES N[C@@H]([C@@H]1C[C@H]1S(O)(=O)=O)C(O)=O Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	7.70E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Perugia Curated by ChEMBL					Assay Description Displacement of [3H]quisqualate from mGluR1 receptor expressed in BHK cells				J Med Chem 50: 4630-41 (2007) Article DOI: 10.1021/jm070322e BindingDB Entry DOI: 10.7270/Q2DF6S12
Universit£ di Perugia Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 5 (Homo sapiens (Human))	BDBM50220149 ((2S,1'S,2'R)-2-(2'-sulfonocyclopropyl)glycine \| CH...) Show SMILES N[C@@H]([C@@H]1C[C@H]1S(O)(=O)=O)C(O)=O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	8.10E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Perugia Curated by ChEMBL					Assay Description Binding affinity to mGluR5 receptor expressed in BHK cells				J Med Chem 50: 4630-41 (2007) Article DOI: 10.1021/jm070322e BindingDB Entry DOI: 10.7270/Q2DF6S12
Universit£ di Perugia Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 1 (Homo sapiens (Human))	BDBM50220147 ((S)-2-amino-4-sulfobutanoic acid \| CHEMBL230951 \| ...) Show SMILES N[C@@H](CCS(O)(=O)=O)C(O)=O \|r\| Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE KEGG PC cid PC sid PDB UniChem Patents Similars	Article PubMed	8.70E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Perugia Curated by ChEMBL					Assay Description Displacement of [3H]quisqualate from mGluR1 receptor expressed in BHK cells				J Med Chem 50: 4630-41 (2007) Article DOI: 10.1021/jm070322e BindingDB Entry DOI: 10.7270/Q2DF6S12
Universit£ di Perugia Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 1 (Homo sapiens (Human))	BDBM50254338 ((2R)-3-(3'-Carboxybicyclo[1.1.1]pentyl)alanine \| C...) Show SMILES N[C@H](CC12CC(C1)(C2)C(O)=O)C(O)=O \|r\| Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	2.10E+5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Salerno Curated by ChEMBL					Assay Description Displacement of [3H]Quisqualate from human mGluR1A receptor expressed in BHK cells				Bioorg Med Chem 17: 242-50 (2008) Article DOI: 10.1016/j.bmc.2008.11.015 BindingDB Entry DOI: 10.7270/Q2HD7WKF
Universit£ di Salerno Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 2 (Homo sapiens (Human))	BDBM50220148 ((2S,1'R,2'S)-2-(2'-sulfonocyclopropyl)glycine \| CH...) Show SMILES N[C@@H]([C@H]1C[C@@H]1S(O)(=O)=O)C(O)=O Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	2.35E+5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Perugia Curated by ChEMBL					Assay Description Displacement of [3H]LY341495 from mGluR2 receptor expressed in BHK cells				J Med Chem 50: 4630-41 (2007) Article DOI: 10.1021/jm070322e BindingDB Entry DOI: 10.7270/Q2DF6S12
Universit£ di Perugia Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 1 (Homo sapiens (Human))	BDBM50220150 ((2R,1'S,2'R)-2-(2'-sulfonocyclopropyl)glycine \| CH...) Show SMILES N[C@H]([C@@H]1C[C@H]1S(O)(=O)=O)C(O)=O Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	2.54E+5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Perugia Curated by ChEMBL					Assay Description Displacement of [3H]quisqualate from mGluR1 receptor expressed in BHK cells				J Med Chem 50: 4630-41 (2007) Article DOI: 10.1021/jm070322e BindingDB Entry DOI: 10.7270/Q2DF6S12
Universit£ di Perugia Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 5 (Homo sapiens (Human))	BDBM50254389 ((2S)-2-(3'-Carboxymethylbicyclo[1.1.1]pentyl)glyci...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	2.93E+5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Salerno Curated by ChEMBL					Assay Description Displacement of [3H]Quisqualate from human mGluR5 receptor expressed in BHK cells				Bioorg Med Chem 17: 242-50 (2008) Article DOI: 10.1016/j.bmc.2008.11.015 BindingDB Entry DOI: 10.7270/Q2HD7WKF
Universit£ di Salerno Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50220145 ((2S,1'R,2'R)-2-(2'-sulfonocyclopropyl)glycine \| CH...) Show SMILES N[C@@H]([C@H]1C[C@H]1S(O)(=O)=O)C(O)=O Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	>3.00E+5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Perugia Curated by ChEMBL					Assay Description Displacement of [3H]LAP4 from mGluR4 receptor expressed in BHK cells				J Med Chem 50: 4630-41 (2007) Article DOI: 10.1021/jm070322e BindingDB Entry DOI: 10.7270/Q2DF6S12
Universit£ di Perugia Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 5 (Homo sapiens (Human))	BDBM50254391 ((2S)-(3'-Phosphonomethylbicyclo[1.1.1]pentyl)glyci...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	>3.00E+5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Salerno Curated by ChEMBL					Assay Description Displacement of [3H]Quisqualate from human mGluR5 receptor expressed in BHK cells				Bioorg Med Chem 17: 242-50 (2008) Article DOI: 10.1016/j.bmc.2008.11.015 BindingDB Entry DOI: 10.7270/Q2HD7WKF
Universit£ di Salerno Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 1 (Homo sapiens (Human))	BDBM50254391 ((2S)-(3'-Phosphonomethylbicyclo[1.1.1]pentyl)glyci...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	>3.00E+5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Salerno Curated by ChEMBL					Assay Description Displacement of [3H]Quisqualate from human mGluR1A receptor expressed in BHK cells				Bioorg Med Chem 17: 242-50 (2008) Article DOI: 10.1016/j.bmc.2008.11.015 BindingDB Entry DOI: 10.7270/Q2HD7WKF
Universit£ di Salerno Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 1 (Homo sapiens (Human))	BDBM50220145 ((2S,1'R,2'R)-2-(2'-sulfonocyclopropyl)glycine \| CH...) Show SMILES N[C@@H]([C@H]1C[C@H]1S(O)(=O)=O)C(O)=O Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	>3.00E+5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Perugia Curated by ChEMBL					Assay Description Displacement of [3H]quisqualate from mGluR1 receptor expressed in BHK cells				J Med Chem 50: 4630-41 (2007) Article DOI: 10.1021/jm070322e BindingDB Entry DOI: 10.7270/Q2DF6S12
Universit£ di Perugia Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 5 (Homo sapiens (Human))	BDBM50220146 ((2S,1'S,2'S)-2-(2'-sulfonocyclopropyl)glycine \| CH...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	>3.00E+5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Perugia Curated by ChEMBL					Assay Description Binding affinity to mGluR5 receptor expressed in BHK cells				J Med Chem 50: 4630-41 (2007) Article DOI: 10.1021/jm070322e BindingDB Entry DOI: 10.7270/Q2DF6S12
Universit£ di Perugia Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 2 (Homo sapiens (Human))	BDBM50220147 ((S)-2-amino-4-sulfobutanoic acid \| CHEMBL230951 \| ...) Show SMILES N[C@@H](CCS(O)(=O)=O)C(O)=O \|r\| Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE KEGG PC cid PC sid PDB UniChem Patents Similars	Article PubMed	>3.00E+5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Perugia Curated by ChEMBL					Assay Description Displacement of [3H]LY341495 from mGluR2 receptor expressed in BHK cells				J Med Chem 50: 4630-41 (2007) Article DOI: 10.1021/jm070322e BindingDB Entry DOI: 10.7270/Q2DF6S12
Universit£ di Perugia Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50220153 ((2R,1'R,2'S)-2-(2'-sulfonocyclopropyl)glycine \| CH...) Show SMILES N[C@H]([C@H]1C[C@@H]1S(O)(=O)=O)C(O)=O Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	>3.00E+5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Perugia Curated by ChEMBL					Assay Description Displacement of [3H]LAP4 from mGluR4 receptor expressed in BHK cells				J Med Chem 50: 4630-41 (2007) Article DOI: 10.1021/jm070322e BindingDB Entry DOI: 10.7270/Q2DF6S12
Universit£ di Perugia Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50220150 ((2R,1'S,2'R)-2-(2'-sulfonocyclopropyl)glycine \| CH...) Show SMILES N[C@H]([C@@H]1C[C@H]1S(O)(=O)=O)C(O)=O Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	>3.00E+5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Perugia Curated by ChEMBL					Assay Description Displacement of [3H]LAP4 from mGluR4 receptor expressed in BHK cells				J Med Chem 50: 4630-41 (2007) Article DOI: 10.1021/jm070322e BindingDB Entry DOI: 10.7270/Q2DF6S12
Universit£ di Perugia Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 5 (Homo sapiens (Human))	BDBM50254337 ((2S)-3-(3'-Carboxybicyclo[1.1.1]pentyl)alanine \| C...) Show SMILES N[C@@H](CC12CC(C1)(C2)C(O)=O)C(O)=O \|r\| Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	>3.00E+5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Salerno Curated by ChEMBL					Assay Description Displacement of [3H]Quisqualate from human mGluR5 receptor expressed in BHK cells				Bioorg Med Chem 17: 242-50 (2008) Article DOI: 10.1016/j.bmc.2008.11.015 BindingDB Entry DOI: 10.7270/Q2HD7WKF
Universit£ di Salerno Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50220149 ((2S,1'S,2'R)-2-(2'-sulfonocyclopropyl)glycine \| CH...) Show SMILES N[C@@H]([C@@H]1C[C@H]1S(O)(=O)=O)C(O)=O Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	>3.00E+5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Perugia Curated by ChEMBL					Assay Description Displacement of [3H]LAP4 from mGluR4 receptor expressed in BHK cells				J Med Chem 50: 4630-41 (2007) Article DOI: 10.1021/jm070322e BindingDB Entry DOI: 10.7270/Q2DF6S12
Universit£ di Perugia Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50220151 ((2R,1'S,2'S)-2-(2'-sulfonocyclopropyl)glycine \| CH...) Show SMILES N[C@H]([C@@H]1C[C@@H]1S(O)(=O)=O)C(O)=O Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	>3.00E+5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Perugia Curated by ChEMBL					Assay Description Displacement of [3H]LAP4 from mGluR4 receptor expressed in BHK cells				J Med Chem 50: 4630-41 (2007) Article DOI: 10.1021/jm070322e BindingDB Entry DOI: 10.7270/Q2DF6S12
Universit£ di Perugia Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 5 (Homo sapiens (Human))	BDBM50254390 ((2R)-2-(3'-Carboxymethylbicyclo[1.1.1]pentyl)glyci...) Show SMILES N[C@H](CC12CC(CC(O)=O)(C1)C2)C(O)=O \|r\| Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	>3.00E+5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Salerno Curated by ChEMBL					Assay Description Displacement of [3H]Quisqualate from human mGluR5 receptor expressed in BHK cells				Bioorg Med Chem 17: 242-50 (2008) Article DOI: 10.1016/j.bmc.2008.11.015 BindingDB Entry DOI: 10.7270/Q2HD7WKF
Universit£ di Salerno Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 2 (Homo sapiens (Human))	BDBM50220154 ((2R,1'R,2'R)-2-(2'-sulfonocyclopropyl)glycine \| CH...) Show SMILES N[C@H]([C@H]1C[C@H]1S(O)(=O)=O)C(O)=O Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	>3.00E+5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Perugia Curated by ChEMBL					Assay Description Displacement of [3H]LY341495 from mGluR2 receptor expressed in BHK cells				J Med Chem 50: 4630-41 (2007) Article DOI: 10.1021/jm070322e BindingDB Entry DOI: 10.7270/Q2DF6S12
Universit£ di Perugia Curated by ChEMBL					More data for this Ligand-Target Pair
Metabotropic glutamate receptor 4 (Homo sapiens (Human))	BDBM50220154 ((2R,1'R,2'R)-2-(2'-sulfonocyclopropyl)glycine \| CH...) Show SMILES N[C@H]([C@H]1C[C@H]1S(O)(=O)=O)C(O)=O Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	>3.00E+5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Perugia Curated by ChEMBL					Assay Description Displacement of [3H]LAP4 from mGluR4 receptor expressed in BHK cells				J Med Chem 50: 4630-41 (2007) Article DOI: 10.1021/jm070322e BindingDB Entry DOI: 10.7270/Q2DF6S12
Universit£ di Perugia Curated by ChEMBL					More data for this Ligand-Target Pair

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