Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Melatonin receptor type 1A (Homo sapiens (Human)) | BDBM50118470 (CHEMBL1218 | N-[2-(1,6,7,8-Tetrahydro-2H-3-oxa-as-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid PDB UniChem Patents Similars | DrugBank PDB PubMed | 0.0138 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Chemical Industries, Ltd. Curated by ChEMBL | Assay Description Binding affinity against human Melatonin receptor type 1A (MT1) | J Med Chem 45: 4222-39 (2002) BindingDB Entry DOI: 10.7270/Q2D799S6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Melatonin receptor type 1B (Homo sapiens (Human)) | BDBM50118470 (CHEMBL1218 | N-[2-(1,6,7,8-Tetrahydro-2H-3-oxa-as-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid PDB UniChem Patents Similars | DrugBank PDB PubMed | 0.0450 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Chemical Industries, Ltd. Curated by ChEMBL | Assay Description Binding affinity against human Melatonin receptor type 1B (MT2) | J Med Chem 45: 4222-39 (2002) BindingDB Entry DOI: 10.7270/Q2D799S6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Melatonin receptor type 1A (Homo sapiens (Human)) | BDBM9019 (CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | DrugBank PubMed | 0.0823 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Chemical Industries, Ltd. Curated by ChEMBL | Assay Description Binding affinity against human Melatonin receptor type 1A (MT1) | J Med Chem 45: 4222-39 (2002) BindingDB Entry DOI: 10.7270/Q2D799S6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (GUINEA PIG) | BDBM50474150 (CHEMBL58362) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid PDB UniChem | Article PubMed | 0.0871 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Chiba University Curated by ChEMBL | Assay Description Binding affinity using guinea pig brain membrane preparations, towards Opioid receptor mu 1 using [3H]- DAMGO as radioligand | J Med Chem 45: 1949-56 (2002) Article DOI: 10.1021/jm010576e BindingDB Entry DOI: 10.7270/Q2WS8X0T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent serotonin transporter (Homo sapiens (Human)) | BDBM22416 ((3S,4R)-3-[(1,3-benzodioxol-5-yloxy)methyl]-4-(4-f...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | DrugBank PDB Article PubMed | 0.110 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd. Curated by ChEMBL | Assay Description Displacement of [3H]citalopram from human SERT expressed in HEK293 cell membranes after 1 hr by liquid scintillation counting method | Bioorg Med Chem 25: 293-304 (2017) Article DOI: 10.1016/j.bmc.2016.10.034 BindingDB Entry DOI: 10.7270/Q2571F0B | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Enteropeptidase (Homo sapiens (Human)) | BDBM158073 (US9024044, 1 | US9227949, 1 | US9655879, 1) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | US Patent | 0.140 | n/a | n/a | n/a | n/a | n/a | n/a | 8.0 | n/a |
AJINOMOTO CO., INC. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 uL), 400 mM Tris-HCl buffer (pH 8.0, 25 uL) and 0.5 mg/mL, fluorescence enzyme substrate (... | US Patent US9227949 (2016) BindingDB Entry DOI: 10.7270/Q2959GBT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Enteropeptidase (Homo sapiens (Human)) | BDBM158073 (US9024044, 1 | US9227949, 1 | US9655879, 1) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | US Patent | 0.140 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
EA Pharma Co., Ltd. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 μL) was mixed with 20 μM fluorescence enzyme substrate (Boc-Phe-Ser-Arg-AMC, 50 ... | US Patent US9655879 (2017) BindingDB Entry DOI: 10.7270/Q22Z17KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Homo sapiens (Human)) | BDBM50160807 (4-(4-Fluoro-phenyl)-2-(4-propyl-piperazin-1-yl)-5,...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid UniChem Patents Similars | Article PubMed | 0.140 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Dainippon Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description In vitro binding affinity of the compound against recombinant human dopamine receptor D2L in human liver microsomes | Bioorg Med Chem Lett 15: 1055-9 (2005) Article DOI: 10.1016/j.bmcl.2004.12.028 BindingDB Entry DOI: 10.7270/Q2Z60NKV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Enteropeptidase (Homo sapiens (Human)) | BDBM158073 (US9024044, 1 | US9227949, 1 | US9655879, 1) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | US Patent | 0.140 | n/a | n/a | n/a | n/a | n/a | n/a | 8.0 | n/a |
Ajinomoto Co., Inc. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 μL), 400 mM Tris-HCl buffer (pH 8.0, 25 μL) and 0.5 mg/mL fluorescence enzyme su... | US Patent US9024044 (2015) BindingDB Entry DOI: 10.7270/Q2F47MVB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine protease 1 (Homo sapiens (Human)) | BDBM158146 (US9024044, 74 | US9227949, 74 | US9655879, 74) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 0.180 | n/a | n/a | n/a | n/a | n/a | n/a | 8.0 | n/a |
Ajinomoto Co., Inc. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 μL) was mixed with 20 μM fluorescence enzyme substrate (Boc-Phe-Ser-Arg-AMC, 50 ... | US Patent US9024044 (2015) BindingDB Entry DOI: 10.7270/Q2F47MVB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine protease 1 (Homo sapiens (Human)) | BDBM158146 (US9024044, 74 | US9227949, 74 | US9655879, 74) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 0.180 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
EA Pharma Co., Ltd. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 μL), 400 mM Tris-HCl buffer (pH 8.0, 25 μL) and 0.5 mg/mL fluorescence enzyme su... | US Patent US9655879 (2017) BindingDB Entry DOI: 10.7270/Q22Z17KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine protease 1 (Homo sapiens (Human)) | BDBM158146 (US9024044, 74 | US9227949, 74 | US9655879, 74) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 0.180 | n/a | n/a | n/a | n/a | n/a | n/a | 8.0 | n/a |
AJINOMOTO CO., INC. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 uL) was mixed with 20 uM fluorescence enzyme substrate (Boc-Phe-Ser-Arg-AMC, 50 uL) mixed ... | US Patent US9227949 (2016) BindingDB Entry DOI: 10.7270/Q2959GBT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melatonin receptor type 1B (Homo sapiens (Human)) | BDBM9019 (CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | DrugBank PubMed | 0.195 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Chemical Industries, Ltd. Curated by ChEMBL | Assay Description Binding affinity against human Melatonin receptor type 1B (MT2) | J Med Chem 45: 4222-39 (2002) BindingDB Entry DOI: 10.7270/Q2D799S6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine protease 1 (Homo sapiens (Human)) | BDBM158140 (US9024044, 68 | US9227949, 68 | US9655879, 68) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 0.210 | n/a | n/a | n/a | n/a | n/a | n/a | 8.0 | n/a |
Ajinomoto Co., Inc. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 μL) was mixed with 20 μM fluorescence enzyme substrate (Boc-Phe-Ser-Arg-AMC, 50 ... | US Patent US9024044 (2015) BindingDB Entry DOI: 10.7270/Q2F47MVB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine protease 1 (Homo sapiens (Human)) | BDBM158140 (US9024044, 68 | US9227949, 68 | US9655879, 68) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 0.210 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
EA Pharma Co., Ltd. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 μL), 400 mM Tris-HCl buffer (pH 8.0, 25 μL) and 0.5 mg/mL fluorescence enzyme su... | US Patent US9655879 (2017) BindingDB Entry DOI: 10.7270/Q22Z17KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine protease 1 (Homo sapiens (Human)) | BDBM158140 (US9024044, 68 | US9227949, 68 | US9655879, 68) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 0.210 | n/a | n/a | n/a | n/a | n/a | n/a | 8.0 | n/a |
AJINOMOTO CO., INC. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 uL) was mixed with 20 uM fluorescence enzyme substrate (Boc-Phe-Ser-Arg-AMC, 50 uL) mixed ... | US Patent US9227949 (2016) BindingDB Entry DOI: 10.7270/Q2959GBT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Enteropeptidase (Homo sapiens (Human)) | BDBM158077 (US9024044, 5 | US9227949, 5 | US9655879, 5) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 0.240 | n/a | n/a | n/a | n/a | n/a | n/a | 8.0 | n/a |
AJINOMOTO CO., INC. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 uL), 400 mM Tris-HCl buffer (pH 8.0, 25 uL) and 0.5 mg/mL, fluorescence enzyme substrate (... | US Patent US9227949 (2016) BindingDB Entry DOI: 10.7270/Q2959GBT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Enteropeptidase (Homo sapiens (Human)) | BDBM158140 (US9024044, 68 | US9227949, 68 | US9655879, 68) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 0.240 | n/a | n/a | n/a | n/a | n/a | n/a | 8.0 | n/a |
Ajinomoto Co., Inc. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 μL), 400 mM Tris-HCl buffer (pH 8.0, 25 μL) and 0.5 mg/mL fluorescence enzyme su... | US Patent US9024044 (2015) BindingDB Entry DOI: 10.7270/Q2F47MVB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Enteropeptidase (Homo sapiens (Human)) | BDBM158077 (US9024044, 5 | US9227949, 5 | US9655879, 5) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 0.240 | n/a | n/a | n/a | n/a | n/a | n/a | 8.0 | n/a |
Ajinomoto Co., Inc. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 μL), 400 mM Tris-HCl buffer (pH 8.0, 25 μL) and 0.5 mg/mL fluorescence enzyme su... | US Patent US9024044 (2015) BindingDB Entry DOI: 10.7270/Q2F47MVB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Enteropeptidase (Homo sapiens (Human)) | BDBM158077 (US9024044, 5 | US9227949, 5 | US9655879, 5) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 0.240 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
EA Pharma Co., Ltd. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 μL) was mixed with 20 μM fluorescence enzyme substrate (Boc-Phe-Ser-Arg-AMC, 50 ... | US Patent US9655879 (2017) BindingDB Entry DOI: 10.7270/Q22Z17KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Enteropeptidase (Homo sapiens (Human)) | BDBM199976 (US9227949, 86) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 0.240 | n/a | n/a | n/a | n/a | n/a | n/a | 8.0 | n/a |
AJINOMOTO CO., INC. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 uL), 400 mM Tris-HCl buffer (pH 8.0, 25 uL) and 0.5 mg/mL, fluorescence enzyme substrate (... | US Patent US9227949 (2016) BindingDB Entry DOI: 10.7270/Q2959GBT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Enteropeptidase (Homo sapiens (Human)) | BDBM308550 (US9655879, 86) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 0.240 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
EA Pharma Co., Ltd. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 μL) was mixed with 20 μM fluorescence enzyme substrate (Boc-Phe-Ser-Arg-AMC, 50 ... | US Patent US9655879 (2017) BindingDB Entry DOI: 10.7270/Q22Z17KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Enteropeptidase (Homo sapiens (Human)) | BDBM158140 (US9024044, 68 | US9227949, 68 | US9655879, 68) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 0.240 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
EA Pharma Co., Ltd. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 μL) was mixed with 20 μM fluorescence enzyme substrate (Boc-Phe-Ser-Arg-AMC, 50 ... | US Patent US9655879 (2017) BindingDB Entry DOI: 10.7270/Q22Z17KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Enteropeptidase (Homo sapiens (Human)) | BDBM158140 (US9024044, 68 | US9227949, 68 | US9655879, 68) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 0.240 | n/a | n/a | n/a | n/a | n/a | n/a | 8.0 | n/a |
AJINOMOTO CO., INC. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 uL), 400 mM Tris-HCl buffer (pH 8.0, 25 uL) and 0.5 mg/mL, fluorescence enzyme substrate (... | US Patent US9227949 (2016) BindingDB Entry DOI: 10.7270/Q2959GBT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Enteropeptidase (Homo sapiens (Human)) | BDBM158097 (US9024044, 25 | US9227949, 25) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | US Patent | 0.260 | n/a | n/a | n/a | n/a | n/a | n/a | 8.0 | n/a |
AJINOMOTO CO., INC. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 uL), 400 mM Tris-HCl buffer (pH 8.0, 25 uL) and 0.5 mg/mL, fluorescence enzyme substrate (... | US Patent US9227949 (2016) BindingDB Entry DOI: 10.7270/Q2959GBT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Enteropeptidase (Homo sapiens (Human)) | BDBM308429 (US9655879, 25) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 0.260 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
EA Pharma Co., Ltd. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 μL) was mixed with 20 μM fluorescence enzyme substrate (Boc-Phe-Ser-Arg-AMC, 50 ... | US Patent US9655879 (2017) BindingDB Entry DOI: 10.7270/Q22Z17KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Enteropeptidase (Homo sapiens (Human)) | BDBM158097 (US9024044, 25 | US9227949, 25) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | US Patent | 0.260 | n/a | n/a | n/a | n/a | n/a | n/a | 8.0 | n/a |
Ajinomoto Co., Inc. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 μL), 400 mM Tris-HCl buffer (pH 8.0, 25 μL) and 0.5 mg/mL fluorescence enzyme su... | US Patent US9024044 (2015) BindingDB Entry DOI: 10.7270/Q2F47MVB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Enteropeptidase (Homo sapiens (Human)) | BDBM158096 (US9024044, 24 | US9227949, 24) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 0.270 | n/a | n/a | n/a | n/a | n/a | n/a | 8.0 | n/a |
AJINOMOTO CO., INC. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 uL), 400 mM Tris-HCl buffer (pH 8.0, 25 uL) and 0.5 mg/mL, fluorescence enzyme substrate (... | US Patent US9227949 (2016) BindingDB Entry DOI: 10.7270/Q2959GBT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Enteropeptidase (Homo sapiens (Human)) | BDBM308428 (US9655879, 24) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 0.270 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
EA Pharma Co., Ltd. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 μL) was mixed with 20 μM fluorescence enzyme substrate (Boc-Phe-Ser-Arg-AMC, 50 ... | US Patent US9655879 (2017) BindingDB Entry DOI: 10.7270/Q22Z17KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Enteropeptidase (Homo sapiens (Human)) | BDBM158096 (US9024044, 24 | US9227949, 24) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 0.270 | n/a | n/a | n/a | n/a | n/a | n/a | 8.0 | n/a |
Ajinomoto Co., Inc. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 μL), 400 mM Tris-HCl buffer (pH 8.0, 25 μL) and 0.5 mg/mL fluorescence enzyme su... | US Patent US9024044 (2015) BindingDB Entry DOI: 10.7270/Q2F47MVB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Enteropeptidase (Homo sapiens (Human)) | BDBM158075 (US9024044, 3 | US9227949, 3) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 0.290 | n/a | n/a | n/a | n/a | n/a | n/a | 8.0 | n/a |
AJINOMOTO CO., INC. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 uL), 400 mM Tris-HCl buffer (pH 8.0, 25 uL) and 0.5 mg/mL, fluorescence enzyme substrate (... | US Patent US9227949 (2016) BindingDB Entry DOI: 10.7270/Q2959GBT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Enteropeptidase (Homo sapiens (Human)) | BDBM308123 (US9655879, 3) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 0.290 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
EA Pharma Co., Ltd. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 μL) was mixed with 20 μM fluorescence enzyme substrate (Boc-Phe-Ser-Arg-AMC, 50 ... | US Patent US9655879 (2017) BindingDB Entry DOI: 10.7270/Q22Z17KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Enteropeptidase (Homo sapiens (Human)) | BDBM158075 (US9024044, 3 | US9227949, 3) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 0.290 | n/a | n/a | n/a | n/a | n/a | n/a | 8.0 | n/a |
Ajinomoto Co., Inc. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 μL), 400 mM Tris-HCl buffer (pH 8.0, 25 μL) and 0.5 mg/mL fluorescence enzyme su... | US Patent US9024044 (2015) BindingDB Entry DOI: 10.7270/Q2F47MVB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Enteropeptidase (Homo sapiens (Human)) | BDBM308557 (US9655879, 93) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 0.300 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
EA Pharma Co., Ltd. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 μL) was mixed with 20 μM fluorescence enzyme substrate (Boc-Phe-Ser-Arg-AMC, 50 ... | US Patent US9655879 (2017) BindingDB Entry DOI: 10.7270/Q22Z17KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Enteropeptidase (Homo sapiens (Human)) | BDBM199983 (US9227949, 93) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 0.300 | n/a | n/a | n/a | n/a | n/a | n/a | 8.0 | n/a |
AJINOMOTO CO., INC. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 uL), 400 mM Tris-HCl buffer (pH 8.0, 25 uL) and 0.5 mg/mL, fluorescence enzyme substrate (... | US Patent US9227949 (2016) BindingDB Entry DOI: 10.7270/Q2959GBT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Enteropeptidase (Homo sapiens (Human)) | BDBM158131 (US9024044, 59 | US9227949, 59 | US9655879, 59) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 0.310 | n/a | n/a | n/a | n/a | n/a | n/a | 8.0 | n/a |
Ajinomoto Co., Inc. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 μL), 400 mM Tris-HCl buffer (pH 8.0, 25 μL) and 0.5 mg/mL fluorescence enzyme su... | US Patent US9024044 (2015) BindingDB Entry DOI: 10.7270/Q2F47MVB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Enteropeptidase (Homo sapiens (Human)) | BDBM158131 (US9024044, 59 | US9227949, 59 | US9655879, 59) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 0.310 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
EA Pharma Co., Ltd. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 μL) was mixed with 20 μM fluorescence enzyme substrate (Boc-Phe-Ser-Arg-AMC, 50 ... | US Patent US9655879 (2017) BindingDB Entry DOI: 10.7270/Q22Z17KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Enteropeptidase (Homo sapiens (Human)) | BDBM158131 (US9024044, 59 | US9227949, 59 | US9655879, 59) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 0.310 | n/a | n/a | n/a | n/a | n/a | n/a | 8.0 | n/a |
AJINOMOTO CO., INC. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 uL), 400 mM Tris-HCl buffer (pH 8.0, 25 uL) and 0.5 mg/mL, fluorescence enzyme substrate (... | US Patent US9227949 (2016) BindingDB Entry DOI: 10.7270/Q2959GBT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Enteropeptidase (Homo sapiens (Human)) | BDBM158091 (US9024044, 19 | US9227949, 19) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | US Patent | 0.330 | n/a | n/a | n/a | n/a | n/a | n/a | 8.0 | n/a |
AJINOMOTO CO., INC. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 uL), 400 mM Tris-HCl buffer (pH 8.0, 25 uL) and 0.5 mg/mL, fluorescence enzyme substrate (... | US Patent US9227949 (2016) BindingDB Entry DOI: 10.7270/Q2959GBT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Enteropeptidase (Homo sapiens (Human)) | BDBM308401 (US9655879, 19) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 0.330 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
EA Pharma Co., Ltd. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 μL) was mixed with 20 μM fluorescence enzyme substrate (Boc-Phe-Ser-Arg-AMC, 50 ... | US Patent US9655879 (2017) BindingDB Entry DOI: 10.7270/Q22Z17KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Enteropeptidase (Homo sapiens (Human)) | BDBM158091 (US9024044, 19 | US9227949, 19) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | US Patent | 0.330 | n/a | n/a | n/a | n/a | n/a | n/a | 8.0 | n/a |
Ajinomoto Co., Inc. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 μL), 400 mM Tris-HCl buffer (pH 8.0, 25 μL) and 0.5 mg/mL fluorescence enzyme su... | US Patent US9024044 (2015) BindingDB Entry DOI: 10.7270/Q2F47MVB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Homo sapiens (Human)) | BDBM50206761 (CHEMBL3958278) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.360 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd. Curated by ChEMBL | Assay Description Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in CHOK1 cells after 30 mins by liquid scintillation counting analysis | Bioorg Med Chem 25: 293-304 (2017) Article DOI: 10.1016/j.bmc.2016.10.034 BindingDB Entry DOI: 10.7270/Q2571F0B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Enteropeptidase (Homo sapiens (Human)) | BDBM158147 (US9024044, 75 | US9227949, 75 | US9655879, 75) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 0.390 | n/a | n/a | n/a | n/a | n/a | n/a | 8.0 | n/a |
Ajinomoto Co., Inc. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 μL), 400 mM Tris-HCl buffer (pH 8.0, 25 μL) and 0.5 mg/mL fluorescence enzyme su... | US Patent US9024044 (2015) BindingDB Entry DOI: 10.7270/Q2F47MVB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Enteropeptidase (Homo sapiens (Human)) | BDBM158147 (US9024044, 75 | US9227949, 75 | US9655879, 75) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 0.390 | n/a | n/a | n/a | n/a | n/a | n/a | 8.0 | n/a |
AJINOMOTO CO., INC. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 uL), 400 mM Tris-HCl buffer (pH 8.0, 25 uL) and 0.5 mg/mL, fluorescence enzyme substrate (... | US Patent US9227949 (2016) BindingDB Entry DOI: 10.7270/Q2959GBT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Enteropeptidase (Homo sapiens (Human)) | BDBM158147 (US9024044, 75 | US9227949, 75 | US9655879, 75) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 0.390 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
EA Pharma Co., Ltd. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 μL) was mixed with 20 μM fluorescence enzyme substrate (Boc-Phe-Ser-Arg-AMC, 50 ... | US Patent US9655879 (2017) BindingDB Entry DOI: 10.7270/Q22Z17KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Enteropeptidase (Homo sapiens (Human)) | BDBM199977 (US9227949, 87 | US9655879, 87) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 0.390 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
EA Pharma Co., Ltd. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 μL) was mixed with 20 μM fluorescence enzyme substrate (Boc-Phe-Ser-Arg-AMC, 50 ... | US Patent US9655879 (2017) BindingDB Entry DOI: 10.7270/Q22Z17KS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Enteropeptidase (Homo sapiens (Human)) | BDBM199977 (US9227949, 87 | US9655879, 87) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 0.390 | n/a | n/a | n/a | n/a | n/a | n/a | 8.0 | n/a |
AJINOMOTO CO., INC. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 uL), 400 mM Tris-HCl buffer (pH 8.0, 25 uL) and 0.5 mg/mL, fluorescence enzyme substrate (... | US Patent US9227949 (2016) BindingDB Entry DOI: 10.7270/Q2959GBT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Enteropeptidase (Homo sapiens (Human)) | BDBM158079 (US9024044, 7 | US9227949, 7 | US9655879, 7) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 0.410 | n/a | n/a | n/a | n/a | n/a | n/a | 8.0 | n/a |
AJINOMOTO CO., INC. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 uL), 400 mM Tris-HCl buffer (pH 8.0, 25 uL) and 0.5 mg/mL, fluorescence enzyme substrate (... | US Patent US9227949 (2016) BindingDB Entry DOI: 10.7270/Q2959GBT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Enteropeptidase (Homo sapiens (Human)) | BDBM158083 (US9024044, 11 | US9227949, 11) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 0.410 | n/a | n/a | n/a | n/a | n/a | n/a | 8.0 | n/a |
AJINOMOTO CO., INC. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 uL), 400 mM Tris-HCl buffer (pH 8.0, 25 uL) and 0.5 mg/mL, fluorescence enzyme substrate (... | US Patent US9227949 (2016) BindingDB Entry DOI: 10.7270/Q2959GBT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Enteropeptidase (Homo sapiens (Human)) | BDBM158079 (US9024044, 7 | US9227949, 7 | US9655879, 7) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 0.410 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
EA Pharma Co., Ltd. US Patent | Assay Description Using a 96 well plate (#3915, Costar), a test compound (25 μL) was mixed with 20 μM fluorescence enzyme substrate (Boc-Phe-Ser-Arg-AMC, 50 ... | US Patent US9655879 (2017) BindingDB Entry DOI: 10.7270/Q22Z17KS | |||||||||||
More data for this Ligand-Target Pair |
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