Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM21015 ((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Similars | PubMed | 0.530 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Napoli Federico II Curated by ChEMBL | Assay Description Compound was evaluated for the binding affinity of Opioid receptor mu 1 by displacing the radioligand [3H]DAMGO from rat brain membrane | Bioorg Med Chem Lett 10: 1185-8 (2000) BindingDB Entry DOI: 10.7270/Q2S46SG6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Rattus norvegicus (rat)) | BDBM20462 ((5Z,8Z,11Z,14Z)-N-[2-(3,4-dihydroxyphenyl)ethyl]ic...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Patents Similars | PubMed | 380 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Bioorganic Chemistry RAS Curated by ChEMBL | Assay Description Concentration required to displace 0.4 nM [3H]-SR-141,716A from CB1 receptor in rat brain preparations in the presence of 0.1 mM phenylmethyl sulphon... | Bioorg Med Chem Lett 11: 447-9 (2001) BindingDB Entry DOI: 10.7270/Q2VT1RBM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Rattus norvegicus (rat)) | BDBM50096883 ((5Z,8Z,11Z,14Z,17Z)-Icosa-5,8,11,14,17-pentaenoic ...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 620 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Bioorganic Chemistry RAS Curated by ChEMBL | Assay Description Concentration required to displace 0.4 nM [3H]-SR-141,716A from CB1 receptor in rat brain preparations in the presence of 0.1 mM phenylmethyl sulphon... | Bioorg Med Chem Lett 11: 447-9 (2001) BindingDB Entry DOI: 10.7270/Q2VT1RBM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50089073 (({1-[3-({1-[2-Amino-3-(4-hydroxy-phenyl)-propionyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 720 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Napoli Federico II Curated by ChEMBL | Assay Description Compound was evaluated for the binding affinity of Opioid receptor mu 1 by displacing the radioligand [3H]DAMGO from rat brain membrane | Bioorg Med Chem Lett 10: 1185-8 (2000) BindingDB Entry DOI: 10.7270/Q2S46SG6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Rattus norvegicus (rat)) | BDBM22988 ((5Z,8Z,11Z,14Z)-N-(2-hydroxyethyl)icosa-5,8,11,14-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL KEGG PC cid PC sid PDB UniChem Patents Similars | PubMed | 800 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Bioorganic Chemistry RAS Curated by ChEMBL | Assay Description Concentration required to displace 0.4 nM [3H]-SR-141,716A from CB1 receptor in rat brain preparations in the presence of 0.1 mM phenylmethyl sulphon... | Bioorg Med Chem Lett 11: 447-9 (2001) BindingDB Entry DOI: 10.7270/Q2VT1RBM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Rattus norvegicus (rat)) | BDBM50096881 ((10Z,13Z,16Z,19Z)-Docosa-7,10,13,16,19-pentaenoic ...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 1.37E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Bioorganic Chemistry RAS Curated by ChEMBL | Assay Description Concentration required to displace 0.4 nM [3H]-SR-141,716A from CB1 receptor in rat brain preparations in the presence of 0.1 mM phenylmethyl sulphon... | Bioorg Med Chem Lett 11: 447-9 (2001) BindingDB Entry DOI: 10.7270/Q2VT1RBM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50089075 (2-({1-[2-({1-[3-({1-[2-Amino-3-(4-hydroxy-phenyl)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.44E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Napoli Federico II Curated by ChEMBL | Assay Description Compound was evaluated for the binding affinity of Opioid receptor mu 1 by displacing the radioligand [3H]DAMGO from rat brain membrane | Bioorg Med Chem Lett 10: 1185-8 (2000) BindingDB Entry DOI: 10.7270/Q2S46SG6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50089071 (({1-[2-({1-[2-Amino-3-(4-hydroxy-phenyl)-propionyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | PubMed | 1.62E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Napoli Federico II Curated by ChEMBL | Assay Description Compound was evaluated for the binding affinity of Opioid receptor mu 1 by displacing the radioligand [3H]DAMGO from rat brain membrane | Bioorg Med Chem Lett 10: 1185-8 (2000) BindingDB Entry DOI: 10.7270/Q2S46SG6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Rattus norvegicus (rat)) | BDBM50096882 ((5Z,9Z,12Z)-Octadeca-5,9,12-trienoic acid [2-(3,4-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 1.72E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Bioorganic Chemistry RAS Curated by ChEMBL | Assay Description Concentration required to displace 0.4 nM [3H]-SR-141,716A from CB1 receptor in rat brain preparations in the presence of 0.1 mM phenylmethyl sulphon... | Bioorg Med Chem Lett 11: 447-9 (2001) BindingDB Entry DOI: 10.7270/Q2VT1RBM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Rattus norvegicus (rat)) | BDBM50096885 ((6Z,9Z,12Z,15Z)-Octadeca-6,9,12,15-tetraenoic acid...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 2.43E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Bioorganic Chemistry RAS Curated by ChEMBL | Assay Description Concentration required to displace 0.4 nM [3H]-SR-141,716A from CB1 receptor in rat brain preparations in the presence of 0.1 mM phenylmethyl sulphon... | Bioorg Med Chem Lett 11: 447-9 (2001) BindingDB Entry DOI: 10.7270/Q2VT1RBM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Rattus norvegicus (rat)) | BDBM50096884 ((9Z,12Z,15Z)-Octadeca-9,12,15-trienoic acid [2-(3,...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 3.13E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Bioorganic Chemistry RAS Curated by ChEMBL | Assay Description Concentration required to displace 0.4 nM [3H]-SR-141,716A from CB1 receptor in rat brain preparations in the presence of 0.1 mM phenylmethyl sulphon... | Bioorg Med Chem Lett 11: 447-9 (2001) BindingDB Entry DOI: 10.7270/Q2VT1RBM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50089072 (2-({1-[2-({1-[2-({1-[2-Amino-3-(4-hydroxy-phenyl)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | PubMed | 7.54E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Napoli Federico II Curated by ChEMBL | Assay Description Compound was evaluated for the binding affinity of Opioid receptor mu 1 by displacing the radioligand [3H]DAMGO from rat brain membrane | Bioorg Med Chem Lett 10: 1185-8 (2000) BindingDB Entry DOI: 10.7270/Q2S46SG6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50089073 (({1-[3-({1-[2-Amino-3-(4-hydroxy-phenyl)-propionyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Napoli Federico II Curated by ChEMBL | Assay Description Inhibitory concentration against [3H]DAMGO binding to Opioid receptor mu 1 in rat brain membrane | Bioorg Med Chem Lett 10: 1185-8 (2000) BindingDB Entry DOI: 10.7270/Q2S46SG6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50089075 (2-({1-[2-({1-[3-({1-[2-Amino-3-(4-hydroxy-phenyl)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 4.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Napoli Federico II Curated by ChEMBL | Assay Description Inhibitory concentration against [3H]DAMGO binding to Opioid receptor mu 1 in rat brain membrane | Bioorg Med Chem Lett 10: 1185-8 (2000) BindingDB Entry DOI: 10.7270/Q2S46SG6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50089071 (({1-[2-({1-[2-Amino-3-(4-hydroxy-phenyl)-propionyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 4.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Napoli Federico II Curated by ChEMBL | Assay Description Inhibitory concentration against [3H]DAMGO binding to Opioid receptor mu 1 in rat brain membrane | Bioorg Med Chem Lett 10: 1185-8 (2000) BindingDB Entry DOI: 10.7270/Q2S46SG6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50089072 (2-({1-[2-({1-[2-({1-[2-Amino-3-(4-hydroxy-phenyl)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Napoli Federico II Curated by ChEMBL | Assay Description Inhibitory concentration against [3H]DAMGO binding to Opioid receptor mu 1 in rat brain membrane | Bioorg Med Chem Lett 10: 1185-8 (2000) BindingDB Entry DOI: 10.7270/Q2S46SG6 | |||||||||||
More data for this Ligand-Target Pair |