Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
N-formyl peptide receptor 2 (Homo sapiens (Human)) | BDBM50098189 (CHEMBL3588930) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 50 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warsaw Curated by ChEMBL | Assay Description Allosteric antagonist activity against FPR2 (unknown origin) | Bioorg Med Chem 23: 4072-81 (2015) Article DOI: 10.1016/j.bmc.2015.03.062 BindingDB Entry DOI: 10.7270/Q2KD20PR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
N-formyl peptide receptor 2 (Homo sapiens (Human)) | BDBM50097999 (CHEMBL3590218) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 80 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warsaw Curated by ChEMBL | Assay Description Antagonist activity against FPR2 (unknown origin) pre-treated for 5 mins before addition of Wpep by Fluo4 florescence based intracellular Ca2+ mobili... | Bioorg Med Chem 23: 4072-81 (2015) Article DOI: 10.1016/j.bmc.2015.03.062 BindingDB Entry DOI: 10.7270/Q2KD20PR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
N-formyl peptide receptor 2 (Homo sapiens (Human)) | BDBM50098001 (CHEMBL3590217) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 90 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warsaw Curated by ChEMBL | Assay Description Antagonist activity against human FPR2 expressed in rat RBL-2H3 cells pre-treated for 15 mins before addition of WKYMVm or C1 by intracellular Ca2+ m... | Bioorg Med Chem 23: 4072-81 (2015) Article DOI: 10.1016/j.bmc.2015.03.062 BindingDB Entry DOI: 10.7270/Q2KD20PR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
N-formyl peptide receptor 2 (Homo sapiens (Human)) | BDBM50098007 (CHEMBL3590216) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 170 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warsaw Curated by ChEMBL | Assay Description Antagonist activity against human FPR2 expressed in rat RBL-2H3 cells pre-treated for 15 mins before addition of WKYMVm or C1 by intracellular Ca2+ m... | Bioorg Med Chem 23: 4072-81 (2015) Article DOI: 10.1016/j.bmc.2015.03.062 BindingDB Entry DOI: 10.7270/Q2KD20PR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
N-formyl peptide receptor 2 (Homo sapiens (Human)) | BDBM50098046 (CHEMBL3590215) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 6.65E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Warsaw Curated by ChEMBL | Assay Description Antagonist activity against human FPR2 expressed in rat RBL-2H3 cells pre-treated for 15 mins before addition of WKYMVm or C1 by intracellular Ca2+ m... | Bioorg Med Chem 23: 4072-81 (2015) Article DOI: 10.1016/j.bmc.2015.03.062 BindingDB Entry DOI: 10.7270/Q2KD20PR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
N-formyl peptide receptor 2 (Homo sapiens (Human)) | BDBM50098055 (CHEMBL3590213) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 8.00E+3 | n/a | n/a | n/a | n/a |
University of Warsaw Curated by ChEMBL | Assay Description Agonist activity against human FPR2 expressed in human HL60 cells by Fluo-4AM dye based intracellular Ca2+ mobilization assay | Bioorg Med Chem 23: 4072-81 (2015) Article DOI: 10.1016/j.bmc.2015.03.062 BindingDB Entry DOI: 10.7270/Q2KD20PR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
N-formyl peptide receptor 2 (Homo sapiens (Human)) | BDBM50098056 (CHEMBL3590212) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 7.30E+3 | n/a | n/a | n/a | n/a |
University of Warsaw Curated by ChEMBL | Assay Description Agonist activity against human FPR2 expressed in human HL60 cells by Fluo-4AM dye based intracellular Ca2+ mobilization assay | Bioorg Med Chem 23: 4072-81 (2015) Article DOI: 10.1016/j.bmc.2015.03.062 BindingDB Entry DOI: 10.7270/Q2KD20PR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
N-formyl peptide receptor 2 (Homo sapiens (Human)) | BDBM50098058 (CHEMBL3590211) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 3.20E+3 | n/a | n/a | n/a | n/a |
University of Warsaw Curated by ChEMBL | Assay Description Agonist activity against human FPR2 expressed in human HL60 cells by Fluo-4AM dye based intracellular Ca2+ mobilization assay | Bioorg Med Chem 23: 4072-81 (2015) Article DOI: 10.1016/j.bmc.2015.03.062 BindingDB Entry DOI: 10.7270/Q2KD20PR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
N-formyl peptide receptor 2 (Homo sapiens (Human)) | BDBM50098059 (CHEMBL3590210) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 6.00E+3 | n/a | n/a | n/a | n/a |
University of Warsaw Curated by ChEMBL | Assay Description Agonist activity against human FPR2 expressed in human HL60 cells by Fluo-4AM dye based intracellular Ca2+ mobilization assay | Bioorg Med Chem 23: 4072-81 (2015) Article DOI: 10.1016/j.bmc.2015.03.062 BindingDB Entry DOI: 10.7270/Q2KD20PR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
N-formyl peptide receptor 2 (Homo sapiens (Human)) | BDBM50098060 (CHEMBL3590209) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 4.03E+3 | n/a | n/a | n/a | n/a |
University of Warsaw Curated by ChEMBL | Assay Description Agonist activity against human FPR2 expressed in human HL60 cells by Fluo-4AM dye based intracellular Ca2+ mobilization assay | Bioorg Med Chem 23: 4072-81 (2015) Article DOI: 10.1016/j.bmc.2015.03.062 BindingDB Entry DOI: 10.7270/Q2KD20PR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
N-formyl peptide receptor 2 (Homo sapiens (Human)) | BDBM50098111 (CHEMBL3590208) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 250 | n/a | n/a | n/a | n/a |
University of Warsaw Curated by ChEMBL | Assay Description Agonist activity against human FPR2 expressed in human HL60 cells by Fluo-4AM dye based intracellular Ca2+ mobilization assay | Bioorg Med Chem 23: 4072-81 (2015) Article DOI: 10.1016/j.bmc.2015.03.062 BindingDB Entry DOI: 10.7270/Q2KD20PR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
N-formyl peptide receptor 2 (Homo sapiens (Human)) | BDBM50098172 (CHEMBL3590207) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 160 | n/a | n/a | n/a | n/a |
University of Warsaw Curated by ChEMBL | Assay Description Agonist activity against human FPR2 expressed in human HL60 cells by Fluo-4AM dye based intracellular Ca2+ mobilization assay | Bioorg Med Chem 23: 4072-81 (2015) Article DOI: 10.1016/j.bmc.2015.03.062 BindingDB Entry DOI: 10.7270/Q2KD20PR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
N-formyl peptide receptor 2 (Homo sapiens (Human)) | BDBM50098173 (CHEMBL3590206) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 7 | n/a | n/a | n/a | n/a |
University of Warsaw Curated by ChEMBL | Assay Description Agonist activity against human FPR2 expressed in human HL60 cells by Fluo-4AM dye based intracellular Ca2+ mobilization assay | Bioorg Med Chem 23: 4072-81 (2015) Article DOI: 10.1016/j.bmc.2015.03.062 BindingDB Entry DOI: 10.7270/Q2KD20PR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
N-formyl peptide receptor 2 (Homo sapiens (Human)) | BDBM50098174 (CHEMBL3588929) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 4 | n/a | n/a | n/a | n/a |
University of Warsaw Curated by ChEMBL | Assay Description Agonist activity against human FPR2 expressed in human HL60 cells by Fluo-4AM dye based intracellular Ca2+ mobilization assay | Bioorg Med Chem 23: 4072-81 (2015) Article DOI: 10.1016/j.bmc.2015.03.062 BindingDB Entry DOI: 10.7270/Q2KD20PR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
N-formyl peptide receptor 2 (Homo sapiens (Human)) | BDBM50098175 (CHEMBL3588928) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 300 | n/a | n/a | n/a | n/a |
University of Warsaw Curated by ChEMBL | Assay Description Agonist activity against human FPR2 expressed in human HL60 cells by Fluo-4AM dye based intracellular Ca2+ mobilization assay | Bioorg Med Chem 23: 4072-81 (2015) Article DOI: 10.1016/j.bmc.2015.03.062 BindingDB Entry DOI: 10.7270/Q2KD20PR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
N-formyl peptide receptor 2 (Homo sapiens (Human)) | BDBM50098176 (CHEMBL3588927) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 50 | n/a | n/a | n/a | n/a |
University of Warsaw Curated by ChEMBL | Assay Description Agonist activity against human FPR2 expressed in human HL60 cells by Fluo-4AM dye based intracellular Ca2+ mobilization assay | Bioorg Med Chem 23: 4072-81 (2015) Article DOI: 10.1016/j.bmc.2015.03.062 BindingDB Entry DOI: 10.7270/Q2KD20PR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
N-formyl peptide receptor 2 (Homo sapiens (Human)) | BDBM50098177 (CHEMBL3588926) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 40 | n/a | n/a | n/a | n/a |
University of Warsaw Curated by ChEMBL | Assay Description Agonist activity against human FPR2 expressed in human HL60 cells by Fluo-4AM dye based intracellular Ca2+ mobilization assay | Bioorg Med Chem 23: 4072-81 (2015) Article DOI: 10.1016/j.bmc.2015.03.062 BindingDB Entry DOI: 10.7270/Q2KD20PR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
N-formyl peptide receptor 2 (Homo sapiens (Human)) | BDBM50098178 (CHEMBL3588925) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 140 | n/a | n/a | n/a | n/a |
University of Warsaw Curated by ChEMBL | Assay Description Agonist activity against human FPR2 expressed in human HL60 cells by Fluo-4AM dye based intracellular Ca2+ mobilization assay | Bioorg Med Chem 23: 4072-81 (2015) Article DOI: 10.1016/j.bmc.2015.03.062 BindingDB Entry DOI: 10.7270/Q2KD20PR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
N-formyl peptide receptor 2 (Homo sapiens (Human)) | BDBM50098179 (CHEMBL3588924) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 300 | n/a | n/a | n/a | n/a |
University of Warsaw Curated by ChEMBL | Assay Description Agonist activity against human FPR2 expressed in human HL60 cells by Fluo-4AM dye based intracellular Ca2+ mobilization assay | Bioorg Med Chem 23: 4072-81 (2015) Article DOI: 10.1016/j.bmc.2015.03.062 BindingDB Entry DOI: 10.7270/Q2KD20PR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
N-formyl peptide receptor 2 (Homo sapiens (Human)) | BDBM50098180 (CHEMBL3588923) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 130 | n/a | n/a | n/a | n/a |
University of Warsaw Curated by ChEMBL | Assay Description Agonist activity against human FPR2 expressed in human HL60 cells by Fluo-4AM dye based intracellular Ca2+ mobilization assay | Bioorg Med Chem 23: 4072-81 (2015) Article DOI: 10.1016/j.bmc.2015.03.062 BindingDB Entry DOI: 10.7270/Q2KD20PR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
N-formyl peptide receptor 2 (Homo sapiens (Human)) | BDBM50098181 (CHEMBL1289381) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | n/a | n/a | 100 | n/a | n/a | n/a | n/a |
University of Warsaw Curated by ChEMBL | Assay Description Agonist activity against human FPR2 expressed in human HL60 cells by Fluo-4AM dye based intracellular Ca2+ mobilization assay | Bioorg Med Chem 23: 4072-81 (2015) Article DOI: 10.1016/j.bmc.2015.03.062 BindingDB Entry DOI: 10.7270/Q2KD20PR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
N-formyl peptide receptor 2 (Homo sapiens (Human)) | BDBM50098182 (CHEMBL1289379) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 900 | n/a | n/a | n/a | n/a |
University of Warsaw Curated by ChEMBL | Assay Description Agonist activity against human FPR2 expressed in human HL60 cells by Fluo-4AM dye based intracellular Ca2+ mobilization assay | Bioorg Med Chem 23: 4072-81 (2015) Article DOI: 10.1016/j.bmc.2015.03.062 BindingDB Entry DOI: 10.7270/Q2KD20PR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
N-formyl peptide receptor 2 (Homo sapiens (Human)) | BDBM50098183 (CHEMBL1288648) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 3.00E+3 | n/a | n/a | n/a | n/a |
University of Warsaw Curated by ChEMBL | Assay Description Agonist activity against human FPR2 expressed in human HL60 cells by Fluo-4AM dye based intracellular Ca2+ mobilization assay | Bioorg Med Chem 23: 4072-81 (2015) Article DOI: 10.1016/j.bmc.2015.03.062 BindingDB Entry DOI: 10.7270/Q2KD20PR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
N-formyl peptide receptor 2 (Homo sapiens (Human)) | BDBM50098184 (AG-26 | CHEMBL1289260) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 400 | n/a | n/a | n/a | n/a |
University of Warsaw Curated by ChEMBL | Assay Description Agonist activity against human FPR2 expressed in human HL60 cells by Fluo-4AM dye based intracellular Ca2+ mobilization assay | Bioorg Med Chem 23: 4072-81 (2015) Article DOI: 10.1016/j.bmc.2015.03.062 BindingDB Entry DOI: 10.7270/Q2KD20PR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Oxoeicosanoid receptor 1 (Homo sapiens (Human)) | BDBM50027524 (5-Oxo-icosa-6,8,11,14-tetraenoic acid methyl ester...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.54E+3 | n/a | n/a | n/a | n/a |
Hospital del Mar Medical Research Institute (IMIM) Curated by ChEMBL | Assay Description Agonist activity at human PK-tagged OXER1 expressed in CHOK1 cells assessed as EA-tagged beta-arrestin recruitment by beta-galactosidase enzyme fragm... | Bioorg Med Chem 26: 3580-3587 (2018) Article DOI: 10.1016/j.bmc.2018.05.036 BindingDB Entry DOI: 10.7270/Q2X63QFQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Oxoeicosanoid receptor 1 (Homo sapiens (Human)) | BDBM50024458 (5-oxo-ETE | CHEMBL18028 | ETE-5-Oxo) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 220 | n/a | n/a | n/a | n/a |
Hospital del Mar Medical Research Institute (IMIM) Curated by ChEMBL | Assay Description Agonist activity at human PK-tagged OXER1 expressed in CHOK1 cells assessed as EA-tagged beta-arrestin recruitment by beta-galactosidase enzyme fragm... | Bioorg Med Chem 26: 3580-3587 (2018) Article DOI: 10.1016/j.bmc.2018.05.036 BindingDB Entry DOI: 10.7270/Q2X63QFQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Oxoeicosanoid receptor 1 (Homo sapiens (Human)) | BDBM50275215 (CHEMBL4128585) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a |
Hospital del Mar Medical Research Institute (IMIM) Curated by ChEMBL | Assay Description Agonist activity at human PK-tagged OXER1 expressed in CHOK1 cells assessed as EA-tagged beta-arrestin recruitment by beta-galactosidase enzyme fragm... | Bioorg Med Chem 26: 3580-3587 (2018) Article DOI: 10.1016/j.bmc.2018.05.036 BindingDB Entry DOI: 10.7270/Q2X63QFQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Oxoeicosanoid receptor 1 (Homo sapiens (Human)) | BDBM50275216 (CHEMBL4130040) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.08E+3 | n/a | n/a | n/a | n/a |
Hospital del Mar Medical Research Institute (IMIM) Curated by ChEMBL | Assay Description Agonist activity at human PK-tagged OXER1 expressed in CHOK1 cells assessed as EA-tagged beta-arrestin recruitment by beta-galactosidase enzyme fragm... | Bioorg Med Chem 26: 3580-3587 (2018) Article DOI: 10.1016/j.bmc.2018.05.036 BindingDB Entry DOI: 10.7270/Q2X63QFQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Oxoeicosanoid receptor 1 (Homo sapiens (Human)) | BDBM50275217 (CHEMBL4127146) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 380 | n/a | n/a | n/a | n/a |
Hospital del Mar Medical Research Institute (IMIM) Curated by ChEMBL | Assay Description Agonist activity at human PK-tagged OXER1 expressed in CHOK1 cells assessed as EA-tagged beta-arrestin recruitment by beta-galactosidase enzyme fragm... | Bioorg Med Chem 26: 3580-3587 (2018) Article DOI: 10.1016/j.bmc.2018.05.036 BindingDB Entry DOI: 10.7270/Q2X63QFQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
N-formyl peptide receptor 2 (Homo sapiens (Human)) | BDBM50098048 (CHEMBL1290698) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 4.70E+3 | n/a | n/a | n/a | n/a |
University of Warsaw Curated by ChEMBL | Assay Description Agonist activity against human FPR2 expressed in human HL60 cells by Fluo-4AM dye based intracellular Ca2+ mobilization assay | Bioorg Med Chem 23: 4072-81 (2015) Article DOI: 10.1016/j.bmc.2015.03.062 BindingDB Entry DOI: 10.7270/Q2KD20PR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
N-formyl peptide receptor 2 (Homo sapiens (Human)) | BDBM50098047 (CHEMBL3590214) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | n/a | n/a | 1.00E+4 | n/a | n/a | n/a | n/a |
University of Warsaw Curated by ChEMBL | Assay Description Agonist activity against human FPR2 expressed in human HL60 cells by Fluo-4AM dye based intracellular Ca2+ mobilization assay | Bioorg Med Chem 23: 4072-81 (2015) Article DOI: 10.1016/j.bmc.2015.03.062 BindingDB Entry DOI: 10.7270/Q2KD20PR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
N-formyl peptide receptor 2 (Homo sapiens (Human)) | BDBM50098007 (CHEMBL3590216) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.48E+3 | n/a | n/a | n/a | n/a |
University of Warsaw Curated by ChEMBL | Assay Description Agonist activity at human FPR2 expressed in rat RBL-2H3 cells by intracellular Ca2+ mobilization assay | Bioorg Med Chem 23: 4072-81 (2015) Article DOI: 10.1016/j.bmc.2015.03.062 BindingDB Entry DOI: 10.7270/Q2KD20PR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
N-formyl peptide receptor 2 (Homo sapiens (Human)) | BDBM50098001 (CHEMBL3590217) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | n/a | n/a | 470 | n/a | n/a | n/a | n/a |
University of Warsaw Curated by ChEMBL | Assay Description Agonist activity at human FPR2 expressed in rat RBL-2H3 cells by intracellular Ca2+ mobilization assay | Bioorg Med Chem 23: 4072-81 (2015) Article DOI: 10.1016/j.bmc.2015.03.062 BindingDB Entry DOI: 10.7270/Q2KD20PR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Oxoeicosanoid receptor 1 (Homo sapiens (Human)) | BDBM50275229 (CHEMBL4128214) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a |
Hospital del Mar Medical Research Institute (IMIM) Curated by ChEMBL | Assay Description Agonist activity at human PK-tagged OXER1 expressed in CHOK1 cells assessed as EA-tagged beta-arrestin recruitment by beta-galactosidase enzyme fragm... | Bioorg Med Chem 26: 3580-3587 (2018) Article DOI: 10.1016/j.bmc.2018.05.036 BindingDB Entry DOI: 10.7270/Q2X63QFQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
N-formyl peptide receptor 2 (Homo sapiens (Human)) | BDBM50098000 (CHEMBL3588922) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 140 | n/a | n/a | n/a | n/a |
University of Warsaw Curated by ChEMBL | Assay Description Agonist activity at FPR2 (unknown origin) by Fluo4 florescence based intracellular Ca2+ mobilization assay | Bioorg Med Chem 23: 4072-81 (2015) Article DOI: 10.1016/j.bmc.2015.03.062 BindingDB Entry DOI: 10.7270/Q2KD20PR | |||||||||||
More data for this Ligand-Target Pair |