Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Gonadotropin-releasing hormone receptor (Rattus norvegicus) | BDBM50187673 (5-(3,3,6-trimethyl-indan-5-yloxy)-furan-2-carboxyl...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.400 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research & Development Curated by ChEMBL | Assay Description Binding affinity to rat pituitary GnRH receptor | J Med Chem 49: 3362-7 (2006) Article DOI: 10.1021/jm060012g BindingDB Entry DOI: 10.7270/Q2F76C54 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50187673 (5-(3,3,6-trimethyl-indan-5-yloxy)-furan-2-carboxyl...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.400 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research & Development Curated by ChEMBL | Assay Description Binding affinity to human recombinant GnRH receptor | J Med Chem 49: 3362-7 (2006) Article DOI: 10.1021/jm060012g BindingDB Entry DOI: 10.7270/Q2F76C54 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Rattus norvegicus) | BDBM50121472 (5-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro-naphth...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 1.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development-La Jolla/Agouron Pharmaceuticals Curated by ChEMBL | Assay Description In vitro binding affinity towards rat gonadotropin-releasing hormone receptor | Bioorg Med Chem Lett 12: 3635-9 (2002) BindingDB Entry DOI: 10.7270/Q2XK8DXZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C beta type (Homo sapiens (Human)) | BDBM153901 (US8999981, A146) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 1.70 | -50.9 | n/a | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer Inc.; Pfizer Products Inc. US Patent | Assay Description Protein Kinase C beta 2 (PKC beta II) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe... | US Patent US8999981 (2015) BindingDB Entry DOI: 10.7270/Q2RR1X0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C beta type (Homo sapiens (Human)) | BDBM153898 (US8999981, A143) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | US Patent | 1.90 | -50.6 | n/a | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer Inc.; Pfizer Products Inc. US Patent | Assay Description Protein Kinase C beta 2 (PKC beta II) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe... | US Patent US8999981 (2015) BindingDB Entry DOI: 10.7270/Q2RR1X0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Rattus norvegicus) | BDBM50121475 (5-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro-naphth...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 2.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development-La Jolla/Agouron Pharmaceuticals Curated by ChEMBL | Assay Description In vitro binding affinity towards rat gonadotropin-releasing hormone receptor | Bioorg Med Chem Lett 12: 3635-9 (2002) BindingDB Entry DOI: 10.7270/Q2XK8DXZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Rattus norvegicus) | BDBM50121461 (5-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro-naphth...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development-La Jolla/Agouron Pharmaceuticals Curated by ChEMBL | Assay Description In vitro binding affinity towards rat gonadotropin-releasing hormone receptor | Bioorg Med Chem Lett 12: 3635-9 (2002) BindingDB Entry DOI: 10.7270/Q2XK8DXZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C beta type (Homo sapiens (Human)) | BDBM153757 (US8999981, A2) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 3.05 | -49.4 | n/a | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer Inc.; Pfizer Products Inc. US Patent | Assay Description Protein Kinase C beta 2 (PKC beta II) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe... | US Patent US8999981 (2015) BindingDB Entry DOI: 10.7270/Q2RR1X0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C beta type (Homo sapiens (Human)) | BDBM154004 (US8999981, F60) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 4.17 | -48.6 | n/a | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer Inc.; Pfizer Products Inc. US Patent | Assay Description Protein Kinase C beta 2 (PKC beta II) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe... | US Patent US8999981 (2015) BindingDB Entry DOI: 10.7270/Q2RR1X0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Rattus norvegicus) | BDBM50121484 (5-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro-naphth...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 4.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development-La Jolla/Agouron Pharmaceuticals Curated by ChEMBL | Assay Description Competitive inhibition of GnRH-stimulated extracellular acidification in cells expressing recombinant rat GnRH receptor | Bioorg Med Chem Lett 12: 3635-9 (2002) BindingDB Entry DOI: 10.7270/Q2XK8DXZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Rattus norvegicus) | BDBM50121484 (5-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro-naphth...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 4.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development-La Jolla/Agouron Pharmaceuticals Curated by ChEMBL | Assay Description In vitro binding affinity towards rat gonadotropin-releasing hormone receptor | Bioorg Med Chem Lett 12: 3635-9 (2002) BindingDB Entry DOI: 10.7270/Q2XK8DXZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C beta type (Homo sapiens (Human)) | BDBM153933 (US8999981, E3) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 5.51 | -47.9 | n/a | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer Inc.; Pfizer Products Inc. US Patent | Assay Description Protein Kinase C beta 2 (PKC beta II) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe... | US Patent US8999981 (2015) BindingDB Entry DOI: 10.7270/Q2RR1X0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Rattus norvegicus) | BDBM50121464 (5-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro-naphth...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development-La Jolla/Agouron Pharmaceuticals Curated by ChEMBL | Assay Description In vitro binding affinity towards rat gonadotropin-releasing hormone receptor | Bioorg Med Chem Lett 12: 3635-9 (2002) BindingDB Entry DOI: 10.7270/Q2XK8DXZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C beta type (Homo sapiens (Human)) | BDBM153934 (US8999981, E4) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 6.17 | -47.6 | n/a | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer Inc.; Pfizer Products Inc. US Patent | Assay Description Protein Kinase C beta 2 (PKC beta II) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe... | US Patent US8999981 (2015) BindingDB Entry DOI: 10.7270/Q2RR1X0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C beta type (Homo sapiens (Human)) | BDBM153936 (US8999981, E6) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 6.81 | -47.4 | n/a | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer Inc.; Pfizer Products Inc. US Patent | Assay Description Protein Kinase C beta 2 (PKC beta II) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe... | US Patent US8999981 (2015) BindingDB Entry DOI: 10.7270/Q2RR1X0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Rattus norvegicus) | BDBM50121462 (5-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro-naphth...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 7 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development-La Jolla/Agouron Pharmaceuticals Curated by ChEMBL | Assay Description In vitro binding affinity towards rat gonadotropin-releasing hormone receptor | Bioorg Med Chem Lett 12: 3635-9 (2002) BindingDB Entry DOI: 10.7270/Q2XK8DXZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Rattus norvegicus) | BDBM50121466 (5-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro-naphth...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 7.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development-La Jolla/Agouron Pharmaceuticals Curated by ChEMBL | Assay Description In vitro binding affinity towards rat gonadotropin-releasing hormone receptor | Bioorg Med Chem Lett 12: 3635-9 (2002) BindingDB Entry DOI: 10.7270/Q2XK8DXZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50121472 (5-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro-naphth...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 8 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development-La Jolla/Agouron Pharmaceuticals Curated by ChEMBL | Assay Description In vitro binding affinity towards human gonadotropin-releasing hormone receptor | Bioorg Med Chem Lett 12: 3635-9 (2002) BindingDB Entry DOI: 10.7270/Q2XK8DXZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C beta type (Homo sapiens (Human)) | BDBM153888 (US8999981, A133) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 8.58 | -46.8 | n/a | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer Inc.; Pfizer Products Inc. US Patent | Assay Description Protein Kinase C beta 2 (PKC beta II) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe... | US Patent US8999981 (2015) BindingDB Entry DOI: 10.7270/Q2RR1X0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Rattus norvegicus) | BDBM50121470 (5-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro-naphth...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 9 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development-La Jolla/Agouron Pharmaceuticals Curated by ChEMBL | Assay Description In vitro binding affinity towards rat gonadotropin-releasing hormone receptor | Bioorg Med Chem Lett 12: 3635-9 (2002) BindingDB Entry DOI: 10.7270/Q2XK8DXZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C beta type (Homo sapiens (Human)) | BDBM153850 (US8999981, A95) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 9.11 | -46.7 | n/a | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer Inc.; Pfizer Products Inc. US Patent | Assay Description Protein Kinase C beta 2 (PKC beta II) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe... | US Patent US8999981 (2015) BindingDB Entry DOI: 10.7270/Q2RR1X0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50121484 (5-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro-naphth...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 9.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development-La Jolla/Agouron Pharmaceuticals Curated by ChEMBL | Assay Description In vitro binding affinity towards human gonadotropin-releasing hormone receptor | Bioorg Med Chem Lett 12: 3635-9 (2002) BindingDB Entry DOI: 10.7270/Q2XK8DXZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C beta type (Homo sapiens (Human)) | BDBM153838 (US8999981, A83) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | US Patent | 9.53 | -46.5 | n/a | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer Inc.; Pfizer Products Inc. US Patent | Assay Description Protein Kinase C beta 2 (PKC beta II) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe... | US Patent US8999981 (2015) BindingDB Entry DOI: 10.7270/Q2RR1X0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C beta type (Homo sapiens (Human)) | BDBM154000 (US8999981, F56) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | <10 | <-46.4 | n/a | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer Inc.; Pfizer Products Inc. US Patent | Assay Description Protein Kinase C beta 2 (PKC beta II) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe... | US Patent US8999981 (2015) BindingDB Entry DOI: 10.7270/Q2RR1X0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C beta type (Homo sapiens (Human)) | BDBM154005 (US8999981, G1 | US8999981, G3) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | <10 | <-46.4 | n/a | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer Inc.; Pfizer Products Inc. US Patent | Assay Description Protein Kinase C beta 2 (PKC beta II) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe... | US Patent US8999981 (2015) BindingDB Entry DOI: 10.7270/Q2RR1X0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C beta type (Homo sapiens (Human)) | BDBM154005 (US8999981, G1 | US8999981, G3) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | <10 | <-46.4 | n/a | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer Inc.; Pfizer Products Inc. US Patent | Assay Description Protein Kinase C beta 2 (PKC beta II) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe... | US Patent US8999981 (2015) BindingDB Entry DOI: 10.7270/Q2RR1X0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50121475 (5-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro-naphth...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development-La Jolla/Agouron Pharmaceuticals Curated by ChEMBL | Assay Description In vitro binding affinity towards human gonadotropin-releasing hormone receptor | Bioorg Med Chem Lett 12: 3635-9 (2002) BindingDB Entry DOI: 10.7270/Q2XK8DXZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C beta type (Homo sapiens (Human)) | BDBM153902 (US8999981, A147) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | <10 | <-46.4 | n/a | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer Inc.; Pfizer Products Inc. US Patent | Assay Description Protein Kinase C beta 2 (PKC beta II) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe... | US Patent US8999981 (2015) BindingDB Entry DOI: 10.7270/Q2RR1X0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C beta type (Homo sapiens (Human)) | BDBM153904 (US8999981, A149) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | <10 | <-46.4 | n/a | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer Inc.; Pfizer Products Inc. US Patent | Assay Description Protein Kinase C beta 2 (PKC beta II) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe... | US Patent US8999981 (2015) BindingDB Entry DOI: 10.7270/Q2RR1X0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C beta type (Homo sapiens (Human)) | BDBM153973 (US8999981, F29) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | <10 | <-46.4 | n/a | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer Inc.; Pfizer Products Inc. US Patent | Assay Description Protein Kinase C beta 2 (PKC beta II) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe... | US Patent US8999981 (2015) BindingDB Entry DOI: 10.7270/Q2RR1X0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C beta type (Homo sapiens (Human)) | BDBM153978 (US8999981, F34) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | <10 | <-46.4 | n/a | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer Inc.; Pfizer Products Inc. US Patent | Assay Description Protein Kinase C beta 2 (PKC beta II) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe... | US Patent US8999981 (2015) BindingDB Entry DOI: 10.7270/Q2RR1X0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C beta type (Homo sapiens (Human)) | BDBM153988 (US8999981, F44) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | <10 | <-46.4 | n/a | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer Inc.; Pfizer Products Inc. US Patent | Assay Description Protein Kinase C beta 2 (PKC beta II) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe... | US Patent US8999981 (2015) BindingDB Entry DOI: 10.7270/Q2RR1X0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C beta type (Homo sapiens (Human)) | BDBM153991 (US8999981, F47) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | <10 | <-46.4 | n/a | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer Inc.; Pfizer Products Inc. US Patent | Assay Description Protein Kinase C beta 2 (PKC beta II) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe... | US Patent US8999981 (2015) BindingDB Entry DOI: 10.7270/Q2RR1X0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C beta type (Homo sapiens (Human)) | BDBM153995 (US8999981, F51) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | <10 | <-46.4 | n/a | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer Inc.; Pfizer Products Inc. US Patent | Assay Description Protein Kinase C beta 2 (PKC beta II) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe... | US Patent US8999981 (2015) BindingDB Entry DOI: 10.7270/Q2RR1X0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C beta type (Homo sapiens (Human)) | BDBM153996 (US8999981, F52) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | <10 | <-46.4 | n/a | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer Inc.; Pfizer Products Inc. US Patent | Assay Description Protein Kinase C beta 2 (PKC beta II) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe... | US Patent US8999981 (2015) BindingDB Entry DOI: 10.7270/Q2RR1X0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C beta type (Homo sapiens (Human)) | BDBM153999 (US8999981, F55) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | <10 | <-46.4 | n/a | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer Inc.; Pfizer Products Inc. US Patent | Assay Description Protein Kinase C beta 2 (PKC beta II) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe... | US Patent US8999981 (2015) BindingDB Entry DOI: 10.7270/Q2RR1X0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C beta type (Homo sapiens (Human)) | BDBM153829 (US8999981, A74) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 10.4 | -46.3 | n/a | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer Inc.; Pfizer Products Inc. US Patent | Assay Description Protein Kinase C beta 2 (PKC beta II) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe... | US Patent US8999981 (2015) BindingDB Entry DOI: 10.7270/Q2RR1X0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C beta type (Homo sapiens (Human)) | BDBM153940 (US8999981, E10) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 10.6 | -46.3 | n/a | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer Inc.; Pfizer Products Inc. US Patent | Assay Description Protein Kinase C beta 2 (PKC beta II) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe... | US Patent US8999981 (2015) BindingDB Entry DOI: 10.7270/Q2RR1X0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Rattus norvegicus) | BDBM50121483 (5-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro-naphth...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 11 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development-La Jolla/Agouron Pharmaceuticals Curated by ChEMBL | Assay Description In vitro binding affinity towards rat gonadotropin-releasing hormone receptor | Bioorg Med Chem Lett 12: 3635-9 (2002) BindingDB Entry DOI: 10.7270/Q2XK8DXZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50121483 (5-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro-naphth...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 11 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development-La Jolla/Agouron Pharmaceuticals Curated by ChEMBL | Assay Description In vitro binding affinity towards human gonadotropin-releasing hormone receptor | Bioorg Med Chem Lett 12: 3635-9 (2002) BindingDB Entry DOI: 10.7270/Q2XK8DXZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C beta type (Homo sapiens (Human)) | BDBM153990 (US8999981, F46) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 11.2 | -46.1 | n/a | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer Inc.; Pfizer Products Inc. US Patent | Assay Description Protein Kinase C beta 2 (PKC beta II) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe... | US Patent US8999981 (2015) BindingDB Entry DOI: 10.7270/Q2RR1X0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C beta type (Homo sapiens (Human)) | BDBM153974 (US8999981, F30) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 11.9 | -46.0 | n/a | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer Inc.; Pfizer Products Inc. US Patent | Assay Description Protein Kinase C beta 2 (PKC beta II) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe... | US Patent US8999981 (2015) BindingDB Entry DOI: 10.7270/Q2RR1X0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C beta type (Homo sapiens (Human)) | BDBM153998 (US8999981, F54) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 12.2 | -45.9 | n/a | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer Inc.; Pfizer Products Inc. US Patent | Assay Description Protein Kinase C beta 2 (PKC beta II) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe... | US Patent US8999981 (2015) BindingDB Entry DOI: 10.7270/Q2RR1X0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C beta type (Homo sapiens (Human)) | BDBM153937 (US8999981, E7) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 12.5 | -45.9 | n/a | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer Inc.; Pfizer Products Inc. US Patent | Assay Description Protein Kinase C beta 2 (PKC beta II) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe... | US Patent US8999981 (2015) BindingDB Entry DOI: 10.7270/Q2RR1X0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C beta type (Homo sapiens (Human)) | BDBM153976 (US8999981, F32) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 12.8 | -45.8 | n/a | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer Inc.; Pfizer Products Inc. US Patent | Assay Description Protein Kinase C beta 2 (PKC beta II) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe... | US Patent US8999981 (2015) BindingDB Entry DOI: 10.7270/Q2RR1X0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C beta type (Homo sapiens (Human)) | BDBM153970 (US8999981, F26) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 12.8 | -45.8 | n/a | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer Inc.; Pfizer Products Inc. US Patent | Assay Description Protein Kinase C beta 2 (PKC beta II) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe... | US Patent US8999981 (2015) BindingDB Entry DOI: 10.7270/Q2RR1X0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C beta type (Homo sapiens (Human)) | BDBM153858 (US8999981, A103) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 12.9 | -45.8 | n/a | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer Inc.; Pfizer Products Inc. US Patent | Assay Description Protein Kinase C beta 2 (PKC beta II) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe... | US Patent US8999981 (2015) BindingDB Entry DOI: 10.7270/Q2RR1X0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50121081 (5-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro-naphth...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 13 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development-La Jolla/Agouron Pharmaceuticals Curated by ChEMBL | Assay Description In vitro binding affinity to human gonadotropin-releasing hormone receptor | Bioorg Med Chem Lett 12: 3467-70 (2002) BindingDB Entry DOI: 10.7270/Q20K27X7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C beta type (Homo sapiens (Human)) | BDBM153878 (US8999981, A123) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 13.3 | -45.7 | n/a | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer Inc.; Pfizer Products Inc. US Patent | Assay Description Protein Kinase C beta 2 (PKC beta II) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe... | US Patent US8999981 (2015) BindingDB Entry DOI: 10.7270/Q2RR1X0K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C beta type (Homo sapiens (Human)) | BDBM153853 (US8999981, A122 | US8999981, A98) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 13.3 | -45.7 | n/a | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer Inc.; Pfizer Products Inc. US Patent | Assay Description Protein Kinase C beta 2 (PKC beta II) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe... | US Patent US8999981 (2015) BindingDB Entry DOI: 10.7270/Q2RR1X0K | |||||||||||
More data for this Ligand-Target Pair |
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