Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
5'-nucleotidase (Rattus norvegicus (Rat)) | BDBM50336767 (CHEMBL257495 | PSB-716 | sodium 1-amino-4-(2-metho...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bonn Curated by ChEMBL | Assay Description Inhibition of rat ecto-5'-nucleotidase | Bioorg Med Chem Lett 18: 223-7 (2008) Article DOI: 10.1016/j.bmcl.2007.10.082 BindingDB Entry DOI: 10.7270/Q2RX9CXT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ectonucleoside triphosphate diphosphohydrolase 1 (Rattus norvegicus) | BDBM50336767 (CHEMBL257495 | PSB-716 | sodium 1-amino-4-(2-metho...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bonn Curated by ChEMBL | Assay Description Inhibition of rat NTPDase 1 | Bioorg Med Chem Lett 18: 223-7 (2008) Article DOI: 10.1016/j.bmcl.2007.10.082 BindingDB Entry DOI: 10.7270/Q2RX9CXT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 2 (Homo sapiens (Human)) | BDBM50271558 (CHEMBL4082045) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 57 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced intracellular calcium influx preincu... | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111789 BindingDB Entry DOI: 10.7270/Q2CJ8J5F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Uracil nucleotide/cysteinyl leukotriene receptor (Homo sapiens (Human)) | BDBM50558931 (CHEMBL4748101) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.33E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human GPR17 expressed in human 1321N1 cells assessed as inhibition of ATP-induced intracellular calcium influx preincubated fo... | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111789 BindingDB Entry DOI: 10.7270/Q2CJ8J5F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Uracil nucleotide/cysteinyl leukotriene receptor (Homo sapiens (Human)) | BDBM50558929 (CHEMBL4752357) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human GPR17 expressed in human 1321N1 cells assessed as inhibition of ATP-induced intracellular calcium influx preincubated fo... | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111789 BindingDB Entry DOI: 10.7270/Q2CJ8J5F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Uracil nucleotide/cysteinyl leukotriene receptor (Homo sapiens (Human)) | BDBM50558925 (CHEMBL4748522) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.65E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human GPR17 expressed in human 1321N1 cells assessed as inhibition of ATP-induced intracellular calcium influx preincubated fo... | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111789 BindingDB Entry DOI: 10.7270/Q2CJ8J5F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Uracil nucleotide/cysteinyl leukotriene receptor (Homo sapiens (Human)) | BDBM50558921 (CHEMBL4743510) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.67E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human GPR17 expressed in human 1321N1 cells assessed as inhibition of ATP-induced intracellular calcium influx preincubated fo... | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111789 BindingDB Entry DOI: 10.7270/Q2CJ8J5F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 2 (Homo sapiens (Human)) | BDBM50029031 (1-Amino-4-{4-[4-chloro-6-(3-sulfo-phenylamino)-[1,...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.85E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bonn Curated by ChEMBL | Assay Description Antagonist activity at human recombinant P2Y2 receptor in 1321N1 cells assessed as inhibition of UTP-induced calcium mobilization | Bioorg Med Chem Lett 18: 223-7 (2008) Article DOI: 10.1016/j.bmcl.2007.10.082 BindingDB Entry DOI: 10.7270/Q2RX9CXT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Uracil nucleotide/cysteinyl leukotriene receptor (Homo sapiens (Human)) | BDBM50558932 (CHEMBL4780920) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.92E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human GPR17 expressed in human 1321N1 cells assessed as inhibition of ATP-induced intracellular calcium influx preincubated fo... | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111789 BindingDB Entry DOI: 10.7270/Q2CJ8J5F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Uracil nucleotide/cysteinyl leukotriene receptor (Homo sapiens (Human)) | BDBM50558916 (CHEMBL4777444) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.32E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human GPR17 expressed in human 1321N1 cells assessed as inhibition of ATP-induced intracellular calcium influx preincubated fo... | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111789 BindingDB Entry DOI: 10.7270/Q2CJ8J5F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Uracil nucleotide/cysteinyl leukotriene receptor (Homo sapiens (Human)) | BDBM50558923 (CHEMBL4743246) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human GPR17 expressed in human 1321N1 cells assessed as inhibition of ATP-induced intracellular calcium influx preincubated fo... | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111789 BindingDB Entry DOI: 10.7270/Q2CJ8J5F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 2 (Homo sapiens (Human)) | BDBM50558923 (CHEMBL4743246) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.01E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced intracellular calcium influx preincu... | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111789 BindingDB Entry DOI: 10.7270/Q2CJ8J5F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 2 (Homo sapiens (Human)) | BDBM50336787 (CHEMBL445413 | sodium 1-amino-9,10-dioxo-4-(m-toly...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.04E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bonn Curated by ChEMBL | Assay Description Antagonist activity at human recombinant P2Y2 receptor in 1321N1 cells assessed as inhibition of UTP-induced calcium mobilization | Bioorg Med Chem Lett 18: 223-7 (2008) Article DOI: 10.1016/j.bmcl.2007.10.082 BindingDB Entry DOI: 10.7270/Q2RX9CXT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Uracil nucleotide/cysteinyl leukotriene receptor (Homo sapiens (Human)) | BDBM50558915 (CHEMBL4750852) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.06E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human GPR17 expressed in human 1321N1 cells assessed as inhibition of ATP-induced intracellular calcium influx preincubated fo... | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111789 BindingDB Entry DOI: 10.7270/Q2CJ8J5F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 2 (Homo sapiens (Human)) | BDBM50558922 (CHEMBL4753843) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.17E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced intracellular calcium influx preincu... | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111789 BindingDB Entry DOI: 10.7270/Q2CJ8J5F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Uracil nucleotide/cysteinyl leukotriene receptor (Homo sapiens (Human)) | BDBM50558933 (CHEMBL4796857) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human GPR17 expressed in human 1321N1 cells assessed as inhibition of ATP-induced intracellular calcium influx preincubated fo... | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111789 BindingDB Entry DOI: 10.7270/Q2CJ8J5F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Uracil nucleotide/cysteinyl leukotriene receptor (Homo sapiens (Human)) | BDBM50558920 (CHEMBL4783980) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.33E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human GPR17 expressed in human 1321N1 cells assessed as inhibition of ATP-induced intracellular calcium influx preincubated fo... | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111789 BindingDB Entry DOI: 10.7270/Q2CJ8J5F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Uracil nucleotide/cysteinyl leukotriene receptor (Homo sapiens (Human)) | BDBM50558922 (CHEMBL4753843) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.37E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human GPR17 expressed in human 1321N1 cells assessed as inhibition of ATP-induced intracellular calcium influx preincubated fo... | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111789 BindingDB Entry DOI: 10.7270/Q2CJ8J5F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 2 (Homo sapiens (Human)) | BDBM50558932 (CHEMBL4780920) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.43E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced intracellular calcium influx preincu... | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111789 BindingDB Entry DOI: 10.7270/Q2CJ8J5F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Uracil nucleotide/cysteinyl leukotriene receptor (Homo sapiens (Human)) | BDBM50558917 (CHEMBL4797060) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.61E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human GPR17 expressed in human 1321N1 cells assessed as inhibition of ATP-induced intracellular calcium influx preincubated fo... | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111789 BindingDB Entry DOI: 10.7270/Q2CJ8J5F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Uracil nucleotide/cysteinyl leukotriene receptor (Homo sapiens (Human)) | BDBM50558928 (CHEMBL4764999) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.88E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human GPR17 expressed in human 1321N1 cells assessed as inhibition of ATP-induced intracellular calcium influx preincubated fo... | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111789 BindingDB Entry DOI: 10.7270/Q2CJ8J5F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 2 (Homo sapiens (Human)) | BDBM50227016 (CHEMBL401859 | Sodium 1-amino-4-(4-anilinophenylam...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 3.93E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bonn Curated by ChEMBL | Assay Description Antagonist activity at human recombinant P2Y2 receptor in 1321N1 cells assessed as inhibition of UTP-induced calcium mobilization | Bioorg Med Chem Lett 18: 223-7 (2008) Article DOI: 10.1016/j.bmcl.2007.10.082 BindingDB Entry DOI: 10.7270/Q2RX9CXT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Uracil nucleotide/cysteinyl leukotriene receptor (Homo sapiens (Human)) | BDBM50558903 (CHEMBL4799394) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.07E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human GPR17 expressed in human 1321N1 cells assessed as inhibition of ATP-induced intracellular calcium influx preincubated fo... | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111789 BindingDB Entry DOI: 10.7270/Q2CJ8J5F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Uracil nucleotide/cysteinyl leukotriene receptor (Homo sapiens (Human)) | BDBM50558919 (CHEMBL4741242) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.18E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human GPR17 expressed in human 1321N1 cells assessed as inhibition of ATP-induced intracellular calcium influx preincubated fo... | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111789 BindingDB Entry DOI: 10.7270/Q2CJ8J5F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Uracil nucleotide/cysteinyl leukotriene receptor (Homo sapiens (Human)) | BDBM50558924 (CHEMBL4741688) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.62E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human GPR17 expressed in human 1321N1 cells assessed as inhibition of ATP-induced intracellular calcium influx preincubated fo... | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111789 BindingDB Entry DOI: 10.7270/Q2CJ8J5F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 2 (Mus musculus) | BDBM50029031 (1-Amino-4-{4-[4-chloro-6-(3-sulfo-phenylamino)-[1,...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bonn Curated by ChEMBL | Assay Description Antagonist activity at mouse P2Y2 receptor in mouse NG108-15 cells assessed as inhibition of UTP-induced calcium mobilization | Bioorg Med Chem Lett 18: 223-7 (2008) Article DOI: 10.1016/j.bmcl.2007.10.082 BindingDB Entry DOI: 10.7270/Q2RX9CXT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 2 (Homo sapiens (Human)) | BDBM50227019 (CHEMBL271673 | sodium 1-amino-4-(4-chlorophenylami...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 5.31E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bonn Curated by ChEMBL | Assay Description Antagonist activity at human recombinant P2Y2 receptor in 1321N1 cells assessed as inhibition of UTP-induced calcium mobilization | Bioorg Med Chem Lett 18: 223-7 (2008) Article DOI: 10.1016/j.bmcl.2007.10.082 BindingDB Entry DOI: 10.7270/Q2RX9CXT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 2 (Homo sapiens (Human)) | BDBM50336792 (CHEMBL256688 | sodium 1-amino-4-(2,4-dimethylpheny...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.43E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bonn Curated by ChEMBL | Assay Description Antagonist activity at human recombinant P2Y2 receptor in 1321N1 cells assessed as inhibition of UTP-induced calcium mobilization | Bioorg Med Chem Lett 18: 223-7 (2008) Article DOI: 10.1016/j.bmcl.2007.10.082 BindingDB Entry DOI: 10.7270/Q2RX9CXT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 2 (Homo sapiens (Human)) | BDBM50558924 (CHEMBL4741688) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.55E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced intracellular calcium influx preincu... | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111789 BindingDB Entry DOI: 10.7270/Q2CJ8J5F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 2 (Homo sapiens (Human)) | BDBM50227032 (CHEMBL256057 | acid blue 25 | sodium 1-amino-9,10-...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 5.61E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bonn Curated by ChEMBL | Assay Description Antagonist activity at human recombinant P2Y2 receptor in 1321N1 cells assessed as inhibition of UTP-induced calcium mobilization | Bioorg Med Chem Lett 18: 223-7 (2008) Article DOI: 10.1016/j.bmcl.2007.10.082 BindingDB Entry DOI: 10.7270/Q2RX9CXT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Uracil nucleotide/cysteinyl leukotriene receptor (Homo sapiens (Human)) | BDBM50558914 (CHEMBL4758186) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.75E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human GPR17 expressed in human 1321N1 cells assessed as inhibition of ATP-induced intracellular calcium influx preincubated fo... | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111789 BindingDB Entry DOI: 10.7270/Q2CJ8J5F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 2 (Homo sapiens (Human)) | BDBM50558921 (CHEMBL4743510) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.78E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced intracellular calcium influx preincu... | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111789 BindingDB Entry DOI: 10.7270/Q2CJ8J5F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 2 (Homo sapiens (Human)) | BDBM50227015 (CHEMBL271688 | Sodium 1-amino-4-(4-acetylaminophen...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 5.81E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bonn Curated by ChEMBL | Assay Description Antagonist activity at human recombinant P2Y2 receptor in 1321N1 cells assessed as inhibition of UTP-induced calcium mobilization | Bioorg Med Chem Lett 18: 223-7 (2008) Article DOI: 10.1016/j.bmcl.2007.10.082 BindingDB Entry DOI: 10.7270/Q2RX9CXT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Uracil nucleotide/cysteinyl leukotriene receptor (Homo sapiens (Human)) | BDBM50558918 (CHEMBL4756398) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.18E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human GPR17 expressed in human 1321N1 cells assessed as inhibition of ATP-induced intracellular calcium influx preincubated fo... | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111789 BindingDB Entry DOI: 10.7270/Q2CJ8J5F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 6 (Rattus norvegicus) | BDBM50558932 (CHEMBL4780920) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.19E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at rat P2Y6 receptor expressed in human 1321N1 cells assessed as inhibition of UDP-induced intracellular calcium influx preincuba... | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111789 BindingDB Entry DOI: 10.7270/Q2CJ8J5F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 2 (Homo sapiens (Human)) | BDBM50227018 (CHEMBL404659 | Sodium 1-amino-4-(3-nitrophenylamin...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.52E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bonn Curated by ChEMBL | Assay Description Antagonist activity at human recombinant P2Y2 receptor in 1321N1 cells assessed as inhibition of UTP-induced calcium mobilization | Bioorg Med Chem Lett 18: 223-7 (2008) Article DOI: 10.1016/j.bmcl.2007.10.082 BindingDB Entry DOI: 10.7270/Q2RX9CXT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 2 (Homo sapiens (Human)) | BDBM50336791 (CHEMBL402239 | sodium 1-amino-4-(2,3-dimethylpheny...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.95E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bonn Curated by ChEMBL | Assay Description Antagonist activity at human recombinant P2Y2 receptor in 1321N1 cells assessed as inhibition of UTP-induced calcium mobilization | Bioorg Med Chem Lett 18: 223-7 (2008) Article DOI: 10.1016/j.bmcl.2007.10.082 BindingDB Entry DOI: 10.7270/Q2RX9CXT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 2 (Mus musculus) | BDBM50336767 (CHEMBL257495 | PSB-716 | sodium 1-amino-4-(2-metho...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bonn Curated by ChEMBL | Assay Description Antagonist activity at mouse P2Y2 receptor in mouse NG108-15 cells assessed as inhibition of UTP-induced calcium mobilization | Bioorg Med Chem Lett 18: 223-7 (2008) Article DOI: 10.1016/j.bmcl.2007.10.082 BindingDB Entry DOI: 10.7270/Q2RX9CXT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 2 (Mus musculus) | BDBM50336792 (CHEMBL256688 | sodium 1-amino-4-(2,4-dimethylpheny...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bonn Curated by ChEMBL | Assay Description Antagonist activity at mouse P2Y2 receptor in mouse NG108-15 cells assessed as inhibition of UTP-induced calcium mobilization | Bioorg Med Chem Lett 18: 223-7 (2008) Article DOI: 10.1016/j.bmcl.2007.10.082 BindingDB Entry DOI: 10.7270/Q2RX9CXT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 2 (Mus musculus) | BDBM50371701 (CHEMBL271881) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bonn Curated by ChEMBL | Assay Description Antagonist activity at mouse P2Y2 receptor in mouse NG108-15 cells assessed as inhibition of UTP-induced calcium mobilization | Bioorg Med Chem Lett 18: 223-7 (2008) Article DOI: 10.1016/j.bmcl.2007.10.082 BindingDB Entry DOI: 10.7270/Q2RX9CXT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 2 (Homo sapiens (Human)) | BDBM50371702 (CHEMBL402238) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.26E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bonn Curated by ChEMBL | Assay Description Antagonist activity at human recombinant P2Y2 receptor in 1321N1 cells assessed as inhibition of UTP-induced calcium mobilization | Bioorg Med Chem Lett 18: 223-7 (2008) Article DOI: 10.1016/j.bmcl.2007.10.082 BindingDB Entry DOI: 10.7270/Q2RX9CXT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 2 (Homo sapiens (Human)) | BDBM50336767 (CHEMBL257495 | PSB-716 | sodium 1-amino-4-(2-metho...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.82E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bonn Curated by ChEMBL | Assay Description Antagonist activity at human recombinant P2Y2 receptor in 1321N1 cells assessed as inhibition of UTP-induced calcium mobilization | Bioorg Med Chem Lett 18: 223-7 (2008) Article DOI: 10.1016/j.bmcl.2007.10.082 BindingDB Entry DOI: 10.7270/Q2RX9CXT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Uracil nucleotide/cysteinyl leukotriene receptor (Homo sapiens (Human)) | BDBM50558904 (CHEMBL4751881) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human GPR17 expressed in human 1321N1 cells assessed as inhibition of ATP-induced intracellular calcium influx preincubated fo... | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111789 BindingDB Entry DOI: 10.7270/Q2CJ8J5F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Uracil nucleotide/cysteinyl leukotriene receptor (Homo sapiens (Human)) | BDBM50558905 (CHEMBL4750327) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human GPR17 expressed in human 1321N1 cells assessed as inhibition of ATP-induced intracellular calcium influx preincubated fo... | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111789 BindingDB Entry DOI: 10.7270/Q2CJ8J5F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Uracil nucleotide/cysteinyl leukotriene receptor (Homo sapiens (Human)) | BDBM50558906 (CHEMBL4753686) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human GPR17 expressed in human 1321N1 cells assessed as inhibition of ATP-induced intracellular calcium influx preincubated fo... | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111789 BindingDB Entry DOI: 10.7270/Q2CJ8J5F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Uracil nucleotide/cysteinyl leukotriene receptor (Homo sapiens (Human)) | BDBM50558907 (CHEMBL4795664) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human GPR17 expressed in human 1321N1 cells assessed as inhibition of ATP-induced intracellular calcium influx preincubated fo... | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111789 BindingDB Entry DOI: 10.7270/Q2CJ8J5F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Uracil nucleotide/cysteinyl leukotriene receptor (Homo sapiens (Human)) | BDBM50558908 (CHEMBL4762760) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human GPR17 expressed in human 1321N1 cells assessed as inhibition of ATP-induced intracellular calcium influx preincubated fo... | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111789 BindingDB Entry DOI: 10.7270/Q2CJ8J5F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Uracil nucleotide/cysteinyl leukotriene receptor (Homo sapiens (Human)) | BDBM50558909 (CHEMBL4763683) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human GPR17 expressed in human 1321N1 cells assessed as inhibition of ATP-induced intracellular calcium influx preincubated fo... | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111789 BindingDB Entry DOI: 10.7270/Q2CJ8J5F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Uracil nucleotide/cysteinyl leukotriene receptor (Homo sapiens (Human)) | BDBM50558910 (CHEMBL4742739) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human GPR17 expressed in human 1321N1 cells assessed as inhibition of ATP-induced intracellular calcium influx preincubated fo... | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111789 BindingDB Entry DOI: 10.7270/Q2CJ8J5F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Uracil nucleotide/cysteinyl leukotriene receptor (Homo sapiens (Human)) | BDBM50558911 (CHEMBL4763168) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human GPR17 expressed in human 1321N1 cells assessed as inhibition of ATP-induced intracellular calcium influx preincubated fo... | Citation and Details Article DOI: 10.1016/j.ejmech.2019.111789 BindingDB Entry DOI: 10.7270/Q2CJ8J5F | |||||||||||
More data for this Ligand-Target Pair |
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