BindingDB PrimarySearch

Found 399 hits with Last Name = 'zhong' and Initial = 'j'
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Sodium-dependent dopamine transporter (Homo sapiens (Human))	BDBM50398789 (CHEMBL2180073) Show SMILES Show InChI	NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	293	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Pfizer Inc. Curated by ChEMBL					Assay Description Inhibition of human DAT				J Med Chem 55: 9055-68 (2012) Article DOI: 10.1021/jm3009635 BindingDB Entry DOI: 10.7270/Q2CR5VHK
Pfizer Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium-dependent dopamine transporter (Homo sapiens (Human))	BDBM50398807 (CHEMBL2180074) Show SMILES Show InChI	NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	1.20E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Pfizer Inc. Curated by ChEMBL					Assay Description Inhibition of human DAT				J Med Chem 55: 9055-68 (2012) Article DOI: 10.1021/jm3009635 BindingDB Entry DOI: 10.7270/Q2CR5VHK
Pfizer Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium-dependent dopamine transporter (Homo sapiens (Human))	BDBM50398804 (CHEMBL2177497) Show SMILES Show InChI	NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Pfizer Inc. Curated by ChEMBL					Assay Description Inhibition of human DAT				J Med Chem 55: 9055-68 (2012) Article DOI: 10.1021/jm3009635 BindingDB Entry DOI: 10.7270/Q2CR5VHK
Pfizer Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium-dependent dopamine transporter (Homo sapiens (Human))	BDBM50398800 (CHEMBL2180069) Show SMILES Show InChI	NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Pfizer Inc. Curated by ChEMBL					Assay Description Inhibition of human DAT				J Med Chem 55: 9055-68 (2012) Article DOI: 10.1021/jm3009635 BindingDB Entry DOI: 10.7270/Q2CR5VHK
Pfizer Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Receptor-type tyrosine-protein kinase FLT3 (Homo sapiens (Human))	BDBM50553656 (CHEMBL4744130) Show SMILES Show InChI	PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	0.0150	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of FLT3 ITD mutant (unknown origin) expressed in mouse BaF3 cells				Citation and Details Article DOI: 10.1016/j.bmcl.2020.127532 BindingDB Entry DOI: 10.7270/Q2154MQ1
TBA					More data for this Ligand-Target Pair
Receptor-type tyrosine-protein kinase FLT3 (Homo sapiens (Human))	BDBM50533653 (CHEMBL4519741) Show SMILES Show InChI	PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	0.0380	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of FLT3 ITD mutant (unknown origin) expressed in mouse BaF3 cells				Citation and Details Article DOI: 10.1016/j.bmcl.2020.127532 BindingDB Entry DOI: 10.7270/Q2154MQ1
TBA					More data for this Ligand-Target Pair
Receptor-type tyrosine-protein kinase FLT3 (Homo sapiens (Human))	BDBM50553658 (CHEMBL4790915) Show SMILES Show InChI	PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	0.0720	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of FLT3 ITD mutant (unknown origin) expressed in mouse BaF3 cells				Citation and Details Article DOI: 10.1016/j.bmcl.2020.127532 BindingDB Entry DOI: 10.7270/Q2154MQ1
TBA					More data for this Ligand-Target Pair
Receptor-type tyrosine-protein kinase FLT3 (Homo sapiens (Human))	BDBM50553655 (CHEMBL4749639) Show SMILES Show InChI	PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	0.292	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of FLT3 ITD mutant (unknown origin) expressed in mouse BaF3 cells				Citation and Details Article DOI: 10.1016/j.bmcl.2020.127532 BindingDB Entry DOI: 10.7270/Q2154MQ1
TBA					More data for this Ligand-Target Pair
Serine/threonine-protein kinase PLK1 (Homo sapiens (Human))	BDBM50565570 (CHEMBL4798376) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	<0.508	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assay				Citation and Details Article DOI: 10.1016/j.ejmech.2020.112697 BindingDB Entry DOI: 10.7270/Q2PK0KWC
TBA					More data for this Ligand-Target Pair
Serine/threonine-protein kinase PLK1 (Homo sapiens (Human))	BDBM50565559 (CHEMBL4792017) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	<0.508	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assay				Citation and Details Article DOI: 10.1016/j.ejmech.2020.112697 BindingDB Entry DOI: 10.7270/Q2PK0KWC
TBA					More data for this Ligand-Target Pair
Serine/threonine-protein kinase PLK1 (Homo sapiens (Human))	BDBM50565572 (CHEMBL4800688) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase MCE PC cid PC sid UniChem	Article PubMed	n/a	n/a	<0.508	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assay				Citation and Details Article DOI: 10.1016/j.ejmech.2020.112697 BindingDB Entry DOI: 10.7270/Q2PK0KWC
TBA					More data for this Ligand-Target Pair
Serine/threonine-protein kinase PLK1 (Homo sapiens (Human))	BDBM50565556 (CHEMBL4787929) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	<0.508	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assay				Citation and Details Article DOI: 10.1016/j.ejmech.2020.112697 BindingDB Entry DOI: 10.7270/Q2PK0KWC
TBA					More data for this Ligand-Target Pair
Serine/threonine-protein kinase PLK1 (Homo sapiens (Human))	BDBM50565569 (CHEMBL4780069) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	<0.508	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assay				Citation and Details Article DOI: 10.1016/j.ejmech.2020.112697 BindingDB Entry DOI: 10.7270/Q2PK0KWC
TBA					More data for this Ligand-Target Pair
Serine/threonine-protein kinase PLK1 (Homo sapiens (Human))	BDBM50565571 (CHEMBL4790038) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	0.577	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assay				Citation and Details Article DOI: 10.1016/j.ejmech.2020.112697 BindingDB Entry DOI: 10.7270/Q2PK0KWC
TBA					More data for this Ligand-Target Pair
Receptor-type tyrosine-protein kinase FLT3 (Homo sapiens (Human))	BDBM50553660 (CHEMBL4761091) Show SMILES Show InChI	PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.20	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of FLT3 ITD mutant (unknown origin) expressed in mouse BaF3 cells				Citation and Details Article DOI: 10.1016/j.bmcl.2020.127532 BindingDB Entry DOI: 10.7270/Q2154MQ1
TBA					More data for this Ligand-Target Pair
Receptor-type tyrosine-protein kinase FLT3 (Homo sapiens (Human))	BDBM50533653 (CHEMBL4519741) Show SMILES Show InChI	PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.30	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human partial length FLT3 ITD mutant expressed in bacterial expression system by Kinomescan method				Citation and Details Article DOI: 10.1016/j.bmcl.2020.127532 BindingDB Entry DOI: 10.7270/Q2154MQ1
TBA					More data for this Ligand-Target Pair
Serine/threonine-protein kinase PLK1 (Homo sapiens (Human))	BDBM50565558 (CHEMBL4783888) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.30	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assay				Citation and Details Article DOI: 10.1016/j.ejmech.2020.112697 BindingDB Entry DOI: 10.7270/Q2PK0KWC
TBA					More data for this Ligand-Target Pair
Serine/threonine-protein kinase PLK1 (Homo sapiens (Human))	BDBM50565583 (CHEMBL4780169) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.40	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assay				Citation and Details Article DOI: 10.1016/j.ejmech.2020.112697 BindingDB Entry DOI: 10.7270/Q2PK0KWC
TBA					More data for this Ligand-Target Pair
Receptor-type tyrosine-protein kinase FLT3 (Homo sapiens (Human))	BDBM50553661 (CHEMBL4781811) Show SMILES Show InChI	PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.5	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of FLT3 ITD mutant (unknown origin) expressed in mouse BaF3 cells				Citation and Details Article DOI: 10.1016/j.bmcl.2020.127532 BindingDB Entry DOI: 10.7270/Q2154MQ1
TBA					More data for this Ligand-Target Pair
Serine/threonine-protein kinase PLK1 (Homo sapiens (Human))	BDBM50565555 (CHEMBL4795375) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.60	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assay				Citation and Details Article DOI: 10.1016/j.ejmech.2020.112697 BindingDB Entry DOI: 10.7270/Q2PK0KWC
TBA					More data for this Ligand-Target Pair
Serine/threonine-protein kinase PLK1 (Homo sapiens (Human))	BDBM50565586 (CHEMBL4799529) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.90	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assay				Citation and Details Article DOI: 10.1016/j.ejmech.2020.112697 BindingDB Entry DOI: 10.7270/Q2PK0KWC
TBA					More data for this Ligand-Target Pair
Receptor-type tyrosine-protein kinase FLT3 (Homo sapiens (Human))	BDBM50533659 (CHEMBL4444648) Show SMILES Show InChI	PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	2	n/a	n/a	n/a	n/a	n/a	n/a
Sichuan University/Collaborative Innovation Center of Biotherapy Curated by ChEMBL					Assay Description Inhibition of recombinant human N-terminal GST-tagged FLT3 (564 to end residues) expressed by baculovirus in Sf21 insect cells measured after 10 mins...				J Med Chem 59: 8293-305 (2016) Article DOI: 10.1021/acs.jmedchem.6b00604 BindingDB Entry DOI: 10.7270/Q20Z76SQ
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase PLK1 (Homo sapiens (Human))	BDBM50565585 (CHEMBL4776291) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	2.20	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assay				Citation and Details Article DOI: 10.1016/j.ejmech.2020.112697 BindingDB Entry DOI: 10.7270/Q2PK0KWC
TBA					More data for this Ligand-Target Pair
Serine/threonine-protein kinase PLK1 (Homo sapiens (Human))	BDBM50402023 (BI 6727 \| VOLASERTIB) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase MCE MMDB PC cid PC sid PDB UniChem Similars	MMDB PDB Article PubMed	n/a	n/a	2.40	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assay				Citation and Details Article DOI: 10.1016/j.ejmech.2020.112697 BindingDB Entry DOI: 10.7270/Q2PK0KWC
TBA					More data for this Ligand-Target Pair				3D Structure (crystal)
Serine/threonine-protein kinase PLK1 (Homo sapiens (Human))	BDBM50565577 (CHEMBL4784741) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	2.70	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assay				Citation and Details Article DOI: 10.1016/j.ejmech.2020.112697 BindingDB Entry DOI: 10.7270/Q2PK0KWC
TBA					More data for this Ligand-Target Pair
Receptor-type tyrosine-protein kinase FLT3 (Homo sapiens (Human))	BDBM50300690 (1-(5-Tert-Butyl-1,2-Oxazol-3-Yl)-3-(4-{7-[2-(Morph...) Show SMILES Show InChI	PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars	Article PubMed	n/a	n/a	3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of FLT3 ITD mutant (unknown origin) expressed in mouse BaF3 cells				Citation and Details Article DOI: 10.1016/j.bmcl.2020.127532 BindingDB Entry DOI: 10.7270/Q2154MQ1
TBA					More data for this Ligand-Target Pair
Receptor-type tyrosine-protein kinase FLT3 (Homo sapiens (Human))	BDBM50553674 (CHEMBL4763034) Show SMILES Show InChI	PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	3.10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of FLT3 ITD mutant (unknown origin) expressed in mouse BaF3 cells				Citation and Details Article DOI: 10.1016/j.bmcl.2020.127532 BindingDB Entry DOI: 10.7270/Q2154MQ1
TBA					More data for this Ligand-Target Pair
Receptor-type tyrosine-protein kinase FLT3 (Homo sapiens (Human))	BDBM50553664 (CHEMBL4765203) Show SMILES Show InChI	PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	3.20	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of FLT3 ITD mutant (unknown origin) expressed in mouse BaF3 cells				Citation and Details Article DOI: 10.1016/j.bmcl.2020.127532 BindingDB Entry DOI: 10.7270/Q2154MQ1
TBA					More data for this Ligand-Target Pair
Serine/threonine-protein kinase PLK1 (Homo sapiens (Human))	BDBM50565573 (CHEMBL4785567) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	3.30	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assay				Citation and Details Article DOI: 10.1016/j.ejmech.2020.112697 BindingDB Entry DOI: 10.7270/Q2PK0KWC
TBA					More data for this Ligand-Target Pair
Serine/threonine-protein kinase PLK1 (Homo sapiens (Human))	BDBM50565582 (CHEMBL4790028) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	3.40	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assay				Citation and Details Article DOI: 10.1016/j.ejmech.2020.112697 BindingDB Entry DOI: 10.7270/Q2PK0KWC
TBA					More data for this Ligand-Target Pair
Receptor-type tyrosine-protein kinase FLT3 (Homo sapiens (Human))	BDBM50553658 (CHEMBL4790915) Show SMILES Show InChI	PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	3.5	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of FLT3 ITD/D835Y double mutant (unknown origin) expressed in mouse BaF3 cells				Citation and Details Article DOI: 10.1016/j.bmcl.2020.127532 BindingDB Entry DOI: 10.7270/Q2154MQ1
TBA					More data for this Ligand-Target Pair
Serine/threonine-protein kinase PLK1 (Homo sapiens (Human))	BDBM50565564 (CHEMBL4784781) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	3.70	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assay				Citation and Details Article DOI: 10.1016/j.ejmech.2020.112697 BindingDB Entry DOI: 10.7270/Q2PK0KWC
TBA					More data for this Ligand-Target Pair
Serine/threonine-protein kinase PLK1 (Homo sapiens (Human))	BDBM50565576 (CHEMBL4779654) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	3.80	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assay				Citation and Details Article DOI: 10.1016/j.ejmech.2020.112697 BindingDB Entry DOI: 10.7270/Q2PK0KWC
TBA					More data for this Ligand-Target Pair
Serine/threonine-protein kinase PLK1 (Homo sapiens (Human))	BDBM50565581 (CHEMBL4800085) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	4.30	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assay				Citation and Details Article DOI: 10.1016/j.ejmech.2020.112697 BindingDB Entry DOI: 10.7270/Q2PK0KWC
TBA					More data for this Ligand-Target Pair
Serine/threonine-protein kinase PLK1 (Homo sapiens (Human))	BDBM50565557 (CHEMBL4800017) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	4.40	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assay				Citation and Details Article DOI: 10.1016/j.ejmech.2020.112697 BindingDB Entry DOI: 10.7270/Q2PK0KWC
TBA					More data for this Ligand-Target Pair
Serine/threonine-protein kinase PLK1 (Homo sapiens (Human))	BDBM50565574 (CHEMBL4783122) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	4.60	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assay				Citation and Details Article DOI: 10.1016/j.ejmech.2020.112697 BindingDB Entry DOI: 10.7270/Q2PK0KWC
TBA					More data for this Ligand-Target Pair
Serine/threonine-protein kinase PLK1 (Homo sapiens (Human))	BDBM50565552 (CHEMBL4787496) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	4.70	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assay				Citation and Details Article DOI: 10.1016/j.ejmech.2020.112697 BindingDB Entry DOI: 10.7270/Q2PK0KWC
TBA					More data for this Ligand-Target Pair
Receptor-type tyrosine-protein kinase FLT3 (Homo sapiens (Human))	BDBM50553665 (CHEMBL4763828) Show SMILES Show InChI	PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	4.70	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of FLT3 ITD mutant (unknown origin) expressed in mouse BaF3 cells				Citation and Details Article DOI: 10.1016/j.bmcl.2020.127532 BindingDB Entry DOI: 10.7270/Q2154MQ1
TBA					More data for this Ligand-Target Pair
Serine/threonine-protein kinase PLK1 (Homo sapiens (Human))	BDBM50565584 (CHEMBL4778470) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	4.70	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assay				Citation and Details Article DOI: 10.1016/j.ejmech.2020.112697 BindingDB Entry DOI: 10.7270/Q2PK0KWC
TBA					More data for this Ligand-Target Pair
Receptor-type tyrosine-protein kinase FLT3 (Homo sapiens (Human))	BDBM50553672 (CHEMBL4791482) Show SMILES Show InChI	PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	4.90	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of FLT3 ITD mutant (unknown origin) expressed in mouse BaF3 cells				Citation and Details Article DOI: 10.1016/j.bmcl.2020.127532 BindingDB Entry DOI: 10.7270/Q2154MQ1
TBA					More data for this Ligand-Target Pair
Serine/threonine-protein kinase PLK1 (Homo sapiens (Human))	BDBM50565575 (CHEMBL4778422) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	4.90	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assay				Citation and Details Article DOI: 10.1016/j.ejmech.2020.112697 BindingDB Entry DOI: 10.7270/Q2PK0KWC
TBA					More data for this Ligand-Target Pair
Serine/threonine-protein kinase PLK1 (Homo sapiens (Human))	BDBM50565565 (CHEMBL4796797) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	5	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assay				Citation and Details Article DOI: 10.1016/j.ejmech.2020.112697 BindingDB Entry DOI: 10.7270/Q2PK0KWC
TBA					More data for this Ligand-Target Pair
Receptor-type tyrosine-protein kinase FLT3 (Homo sapiens (Human))	BDBM50533653 (CHEMBL4519741) Show SMILES Show InChI	PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	5	n/a	n/a	n/a	n/a	n/a	n/a
Sichuan University/Collaborative Innovation Center of Biotherapy Curated by ChEMBL					Assay Description Inhibition of recombinant human N-terminal GST-tagged FLT3 (564 to end residues) expressed by baculovirus in Sf21 insect cells measured after 10 mins...				J Med Chem 59: 8293-305 (2016) Article DOI: 10.1021/acs.jmedchem.6b00604 BindingDB Entry DOI: 10.7270/Q20Z76SQ
					More data for this Ligand-Target Pair
Receptor-type tyrosine-protein kinase FLT3 (Homo sapiens (Human))	BDBM50553664 (CHEMBL4765203) Show SMILES Show InChI	PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	5.10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of FLT3 ITD/D835Y double mutant (unknown origin) expressed in mouse BaF3 cells				Citation and Details Article DOI: 10.1016/j.bmcl.2020.127532 BindingDB Entry DOI: 10.7270/Q2154MQ1
TBA					More data for this Ligand-Target Pair
Serine/threonine-protein kinase PLK1 (Homo sapiens (Human))	BDBM50565561 (CHEMBL4799183) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	5.10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assay				Citation and Details Article DOI: 10.1016/j.ejmech.2020.112697 BindingDB Entry DOI: 10.7270/Q2PK0KWC
TBA					More data for this Ligand-Target Pair
Receptor-type tyrosine-protein kinase FLT3 (Homo sapiens (Human))	BDBM50553662 (CHEMBL4795857) Show SMILES Show InChI	PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	5.20	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of FLT3 ITD mutant (unknown origin) expressed in mouse BaF3 cells				Citation and Details Article DOI: 10.1016/j.bmcl.2020.127532 BindingDB Entry DOI: 10.7270/Q2154MQ1
TBA					More data for this Ligand-Target Pair
Receptor-type tyrosine-protein kinase FLT3 (Homo sapiens (Human))	BDBM50553675 (CHEMBL4750430) Show SMILES Show InChI	PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	5.20	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of FLT3 ITD mutant (unknown origin) expressed in mouse BaF3 cells				Citation and Details Article DOI: 10.1016/j.bmcl.2020.127532 BindingDB Entry DOI: 10.7270/Q2154MQ1
TBA					More data for this Ligand-Target Pair
Serine/threonine-protein kinase PLK1 (Homo sapiens (Human))	BDBM50565562 (CHEMBL4790807) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	5.30	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assay				Citation and Details Article DOI: 10.1016/j.ejmech.2020.112697 BindingDB Entry DOI: 10.7270/Q2PK0KWC
TBA					More data for this Ligand-Target Pair
Receptor-type tyrosine-protein kinase FLT3 (Homo sapiens (Human))	BDBM50553665 (CHEMBL4763828) Show SMILES Show InChI	PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	5.40	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of FLT3 ITD/D835Y double mutant (unknown origin) expressed in mouse BaF3 cells				Citation and Details Article DOI: 10.1016/j.bmcl.2020.127532 BindingDB Entry DOI: 10.7270/Q2154MQ1
TBA					More data for this Ligand-Target Pair
Receptor-type tyrosine-protein kinase FLT3 (Homo sapiens (Human))	BDBM50553671 (CHEMBL4749484) Show SMILES Show InChI	PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	5.80	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of FLT3 ITD mutant (unknown origin) expressed in mouse BaF3 cells				Citation and Details Article DOI: 10.1016/j.bmcl.2020.127532 BindingDB Entry DOI: 10.7270/Q2154MQ1
TBA					More data for this Ligand-Target Pair

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