Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Cannabinoid receptor 1 (Homo sapiens (Human)) | BDBM50180022 (5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 0.400 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Corbus Pharmaceuticals, Inc. Curated by ChEMBL | Assay Description Displacement of [3H]-CP-55940 from human CB1 receptor expressed in HEK293T cell membranes by scintillation counting | Bioorg Med Chem 22: 3245-51 (2014) Article DOI: 10.1016/j.bmc.2014.04.062 BindingDB Entry DOI: 10.7270/Q22Z173H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM21278 (5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 1.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Corbus Pharmaceuticals, Inc. Curated by ChEMBL | Assay Description Displacement of [3H]-CP-55940 from human CB2 receptor expressed in HEK293T cell membranes by scintillation counting | Bioorg Med Chem 22: 3245-51 (2014) Article DOI: 10.1016/j.bmc.2014.04.062 BindingDB Entry DOI: 10.7270/Q22Z173H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM50019392 (CHEMBL3290053) | PDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 51 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Corbus Pharmaceuticals, Inc. Curated by ChEMBL | Assay Description Displacement of [3H]-CP-55940 from human CB2 receptor expressed in HEK293T cell membranes by scintillation counting | Bioorg Med Chem 22: 3245-51 (2014) Article DOI: 10.1016/j.bmc.2014.04.062 BindingDB Entry DOI: 10.7270/Q22Z173H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Homo sapiens (Human)) | BDBM50019392 (CHEMBL3290053) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 628 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Corbus Pharmaceuticals, Inc. Curated by ChEMBL | Assay Description Displacement of [3H]-CP-55940 from human CB1 receptor expressed in HEK293T cell membranes by scintillation counting | Bioorg Med Chem 22: 3245-51 (2014) Article DOI: 10.1016/j.bmc.2014.04.062 BindingDB Entry DOI: 10.7270/Q22Z173H | |||||||||||
More data for this Ligand-Target Pair |