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77 molecules are shown

Wt: 264.2
BDBM50433070Purchase		Wt: 321.3
BDBM50438627Purchase
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50433070,50438627   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kcal/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Aminopeptidase N


(Sus scrofa (Pig))		BDBM50433070
PNG
(CHEMBL2376106)
Show SMILES ONC(=O)CN1C(=O)C2(OCCO2)c2ccccc12
Show InChI InChI=1S/C12H12N2O5/c15-10(13-17)7-14-9-4-2-1-3-8(9)12(11(14)16)18-5-6-19-12/h1-4,17H,5-7H2,(H,13,15)
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Article
PubMed
n/an/a 2.09E+5n/an/an/an/an/an/a



Shandong University

Curated by ChEMBL


Assay Description
Inhibition of pig kidney microsome aminopeptidase-N using L-leu-p-nitroanilide as substrate incubated for 5 mins prior to substrate addition measured...

Bioorg Med Chem 21: 2663-70 (2013)


Article DOI: 10.1016/j.bmc.2012.06.024
BindingDB Entry DOI: 10.7270/Q2J67J8H
More data for this
Ligand-Target Pair
Aminopeptidase N


(Sus scrofa (Pig))		BDBM50438627
PNG
(CHEMBL2414225)
Show SMILES COC(=O)CC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C |r|
Show InChI InChI=1S/C17H23NO5/c1-17(2,3)23-16(21)18-13(14(19)11-15(20)22-4)10-12-8-6-5-7-9-12/h5-9,13H,10-11H2,1-4H3,(H,18,21)/t13-/m1/s1
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PubMed
n/an/a>1.00E+6n/an/an/an/an/an/a



Shandong University

Curated by ChEMBL


Assay Description
Inhibition of pig microsomal aminopeptidase N using L-leu-p-nitroanilide as substrate incubated for 5 mins prior to substrate addition measured after...

Bioorg Med Chem Lett 23: 4948-52 (2013)


Article DOI: 10.1016/j.bmcl.2013.06.058
BindingDB Entry DOI: 10.7270/Q2377B4J
More data for this
Ligand-Target Pair