Compounds in cluster

200 molecules are shown

Wt: 252.2 BDBM3863 Purchase	Wt: 222.2 BDBM3790 Purchase	Wt: 193.2 BDBM3791 Purchase	Wt: 194.2 BDBM3792 Purchase	Wt: 195.2 BDBM3793 Purchase
Wt: 237.2 BDBM3827 Purchase	Wt: 239.2 BDBM3828 Purchase	Wt: 209.2 BDBM3829 Purchase	Wt: 194.2 BDBM3794 Purchase	Wt: 224.2 BDBM3796 Purchase
Wt: 236.2 BDBM3830 Purchase	Wt: 222.2 BDBM3831 Purchase	Wt: 219.2 BDBM3832 Purchase	Wt: 210.2 BDBM3797 Purchase	Wt: 238.2 BDBM3799 Purchase

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 33 hits for monomerid = 3863,3790,3791,3792,3793,3827,3828,3829,3794,3796,3830,3831,3832,3797,3799
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Platelet-derived growth factor receptor beta (Homo sapiens (Human))	BDBM3790 (1-Phenylbenzimidazole Analog 7 \| 4-phenyl-2,3-dihy...) Show SMILES C1CC(=Nc2ccccc2N1)c1ccccc1 \|c:2\| Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase PC cid PC sid UniChem	Article PubMed	n/a	n/a	>5.00E+4	n/a	n/a	n/a	n/a	7.4	25
University of Auckland					Assay Description IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...				J Med Chem 41: 5457-65 (1998) Article DOI: 10.1021/jm9804681 BindingDB Entry DOI: 10.7270/Q24T6GJC
University of Auckland					More data for this Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (Homo sapiens (Human))	BDBM3794 (1-Phenylbenzimidazole 3 \| 1-Phenylbenzimidazole de...) Show SMILES c1nc2ccccc2n1-c1ccccc1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase MCE PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	>5.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Auckland					Assay Description IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...				J Med Chem 42: 2373-82 (1999) Article DOI: 10.1021/jm980658b BindingDB Entry DOI: 10.7270/Q2W957B2
University of Auckland					More data for this Ligand-Target Pair
Platelet-derived growth factor receptor beta (Homo sapiens (Human))	BDBM3792 (1-Phenylbenzimidazole deriv. 9 \| 1-phenyl-1H-indaz...) Show SMILES c1nn(-c2ccccc2)c2ccccc12 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	>5.00E+4	n/a	n/a	n/a	n/a	7.4	25
University of Auckland					Assay Description IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...				J Med Chem 41: 5457-65 (1998) Article DOI: 10.1021/jm9804681 BindingDB Entry DOI: 10.7270/Q24T6GJC
University of Auckland					More data for this Ligand-Target Pair
Platelet-derived growth factor receptor beta (Homo sapiens (Human))	BDBM3793 (1-Phenylbenzimidazole deriv. 10 \| 1-phenyl-1H-1,2,...) Show SMILES c1ccc(cc1)-n1nnc2ccccc12 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase MCE PC cid PC sid UniChem Patents	Article PubMed	n/a	n/a	>5.00E+4	n/a	n/a	n/a	n/a	7.4	25
University of Auckland					Assay Description IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...				J Med Chem 41: 5457-65 (1998) Article DOI: 10.1021/jm9804681 BindingDB Entry DOI: 10.7270/Q24T6GJC
University of Auckland					More data for this Ligand-Target Pair
Platelet-derived growth factor receptor beta (Homo sapiens (Human))	BDBM3794 (1-Phenylbenzimidazole 3 \| 1-Phenylbenzimidazole de...) Show SMILES c1nc2ccccc2n1-c1ccccc1 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase MCE PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	9.30E+3	n/a	n/a	n/a	n/a	7.4	25
University of Auckland					Assay Description IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...				J Med Chem 41: 5457-65 (1998) Article DOI: 10.1021/jm9804681 BindingDB Entry DOI: 10.7270/Q24T6GJC
University of Auckland					More data for this Ligand-Target Pair
Platelet-derived growth factor receptor beta (Homo sapiens (Human))	BDBM3796 (1-(2-Methoxyphenyl)benzimidazole Hydrochloride \| 1...) Show SMILES COc1ccccc1-n1cnc2ccccc12 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>5.00E+4	n/a	n/a	n/a	n/a	7.4	25
University of Auckland					Assay Description IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...				J Med Chem 41: 5457-65 (1998) Article DOI: 10.1021/jm9804681 BindingDB Entry DOI: 10.7270/Q24T6GJC
University of Auckland					More data for this Ligand-Target Pair
Fibroblast growth factor receptor 1 (Homo sapiens (Human))	BDBM3790 (1-Phenylbenzimidazole Analog 7 \| 4-phenyl-2,3-dihy...) Show SMILES C1CC(=Nc2ccccc2N1)c1ccccc1 \|c:2\| Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase PC cid PC sid UniChem	Article PubMed	n/a	n/a	>5.00E+4	n/a	n/a	n/a	n/a	7.4	25
University of Auckland					Assay Description IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...				J Med Chem 41: 5457-65 (1998) Article DOI: 10.1021/jm9804681 BindingDB Entry DOI: 10.7270/Q24T6GJC
University of Auckland					More data for this Ligand-Target Pair
Fibroblast growth factor receptor 1 (Homo sapiens (Human))	BDBM3791 (1-Phenylbenzimidazole deriv. 8 \| 1-phenyl-1H-indol...) Show SMILES c1cc2ccccc2n1-c1ccccc1 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase MCE PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	>5.00E+4	n/a	n/a	n/a	n/a	7.4	25
University of Auckland					Assay Description IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...				J Med Chem 41: 5457-65 (1998) Article DOI: 10.1021/jm9804681 BindingDB Entry DOI: 10.7270/Q24T6GJC
University of Auckland					More data for this Ligand-Target Pair
Fibroblast growth factor receptor 1 (Homo sapiens (Human))	BDBM3792 (1-Phenylbenzimidazole deriv. 9 \| 1-phenyl-1H-indaz...) Show SMILES c1nn(-c2ccccc2)c2ccccc12 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	>5.00E+4	n/a	n/a	n/a	n/a	7.4	25
University of Auckland					Assay Description IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...				J Med Chem 41: 5457-65 (1998) Article DOI: 10.1021/jm9804681 BindingDB Entry DOI: 10.7270/Q24T6GJC
University of Auckland					More data for this Ligand-Target Pair
Fibroblast growth factor receptor 1 (Homo sapiens (Human))	BDBM3793 (1-Phenylbenzimidazole deriv. 10 \| 1-phenyl-1H-1,2,...) Show SMILES c1ccc(cc1)-n1nnc2ccccc12 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase MCE PC cid PC sid UniChem Patents	Article PubMed	n/a	n/a	>5.00E+4	n/a	n/a	n/a	n/a	7.4	25
University of Auckland					Assay Description IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...				J Med Chem 41: 5457-65 (1998) Article DOI: 10.1021/jm9804681 BindingDB Entry DOI: 10.7270/Q24T6GJC
University of Auckland					More data for this Ligand-Target Pair
Fibroblast growth factor receptor 1 (Homo sapiens (Human))	BDBM3794 (1-Phenylbenzimidazole 3 \| 1-Phenylbenzimidazole de...) Show SMILES c1nc2ccccc2n1-c1ccccc1 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase MCE PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	>5.00E+4	n/a	n/a	n/a	n/a	7.4	25
University of Auckland					Assay Description IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...				J Med Chem 41: 5457-65 (1998) Article DOI: 10.1021/jm9804681 BindingDB Entry DOI: 10.7270/Q24T6GJC
University of Auckland					More data for this Ligand-Target Pair
Fibroblast growth factor receptor 1 (Homo sapiens (Human))	BDBM3796 (1-(2-Methoxyphenyl)benzimidazole Hydrochloride \| 1...) Show SMILES COc1ccccc1-n1cnc2ccccc12 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>5.00E+4	n/a	n/a	n/a	n/a	7.4	25
University of Auckland					Assay Description IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...				J Med Chem 41: 5457-65 (1998) Article DOI: 10.1021/jm9804681 BindingDB Entry DOI: 10.7270/Q24T6GJC
University of Auckland					More data for this Ligand-Target Pair
Platelet-derived growth factor receptor beta (Homo sapiens (Human))	BDBM3797 (1-Phenylbenzimidazole deriv. 14 \| 2-(1H-1,3-benzod...) Show SMILES Oc1ccccc1-n1cnc2ccccc12 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>5.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Auckland					Assay Description IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...				J Med Chem 41: 5457-65 (1998) Article DOI: 10.1021/jm9804681 BindingDB Entry DOI: 10.7270/Q24T6GJC
University of Auckland					More data for this Ligand-Target Pair
Platelet-derived growth factor receptor beta (Homo sapiens (Human))	BDBM3799 (1-Phenylbenzimidazole deriv. 16 \| 2-(1H-1,3-benzod...) Show SMILES OC(=O)c1ccccc1-n1cnc2ccccc12 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>5.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Auckland					Assay Description IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...				J Med Chem 41: 5457-65 (1998) Article DOI: 10.1021/jm9804681 BindingDB Entry DOI: 10.7270/Q24T6GJC
University of Auckland					More data for this Ligand-Target Pair
Fibroblast growth factor receptor 1 (Homo sapiens (Human))	BDBM3797 (1-Phenylbenzimidazole deriv. 14 \| 2-(1H-1,3-benzod...) Show SMILES Oc1ccccc1-n1cnc2ccccc12 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>5.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Auckland					Assay Description IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...				J Med Chem 41: 5457-65 (1998) Article DOI: 10.1021/jm9804681 BindingDB Entry DOI: 10.7270/Q24T6GJC
University of Auckland					More data for this Ligand-Target Pair
Fibroblast growth factor receptor 1 (Homo sapiens (Human))	BDBM3799 (1-Phenylbenzimidazole deriv. 16 \| 2-(1H-1,3-benzod...) Show SMILES OC(=O)c1ccccc1-n1cnc2ccccc12 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>5.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Auckland					Assay Description IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...				J Med Chem 41: 5457-65 (1998) Article DOI: 10.1021/jm9804681 BindingDB Entry DOI: 10.7270/Q24T6GJC
University of Auckland					More data for this Ligand-Target Pair
Platelet-derived growth factor receptor beta (Homo sapiens (Human))	BDBM3827 (1-(4-Carboxamidophenyl)benzimidazole \| 1-Phenylben...) Show SMILES NC(=O)c1ccc(cc1)-n1cnc2ccccc12 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	2.30E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Auckland					Assay Description IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...				J Med Chem 41: 5457-65 (1998) Article DOI: 10.1021/jm9804681 BindingDB Entry DOI: 10.7270/Q24T6GJC
University of Auckland					More data for this Ligand-Target Pair
Platelet-derived growth factor receptor beta (Homo sapiens (Human))	BDBM3828 (1-(4-nitrophenyl)-1H-1,3-benzodiazole \| 1-Phenylbe...) Show SMILES [O-][N+](=O)c1ccc(cc1)-n1cnc2ccccc12 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase MCE PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	3.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Auckland					Assay Description IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...				J Med Chem 41: 5457-65 (1998) Article DOI: 10.1021/jm9804681 BindingDB Entry DOI: 10.7270/Q24T6GJC
University of Auckland					More data for this Ligand-Target Pair
Platelet-derived growth factor receptor beta (Homo sapiens (Human))	BDBM3829 (1-Phenylbenzimidazole deriv. 46 \| 4-(1H-1,3-benzod...) Show SMILES Nc1ccc(cc1)-n1cnc2ccccc12 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase MCE PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	5.60E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Auckland					Assay Description IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...				J Med Chem 41: 5457-65 (1998) Article DOI: 10.1021/jm9804681 BindingDB Entry DOI: 10.7270/Q24T6GJC
University of Auckland					More data for this Ligand-Target Pair
Platelet-derived growth factor receptor beta (Homo sapiens (Human))	BDBM3830 (1-Phenylbenzimidazole deriv. 47 \| 1-[4-(1H-1,3-ben...) Show SMILES CC(=O)c1ccc(cc1)-n1cnc2ccccc12 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	2.40E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Auckland					Assay Description IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...				J Med Chem 41: 5457-65 (1998) Article DOI: 10.1021/jm9804681 BindingDB Entry DOI: 10.7270/Q24T6GJC
University of Auckland					More data for this Ligand-Target Pair
Platelet-derived growth factor receptor beta (Homo sapiens (Human))	BDBM3831 (1-Phenylbenzimidazole deriv. 48 \| 4-(1H-1,3-benzod...) Show SMILES O=Cc1ccc(cc1)-n1cnc2ccccc12 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase MCE PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	1.30E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Auckland					Assay Description IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...				J Med Chem 41: 5457-65 (1998) Article DOI: 10.1021/jm9804681 BindingDB Entry DOI: 10.7270/Q24T6GJC
University of Auckland					More data for this Ligand-Target Pair
Platelet-derived growth factor receptor beta (Homo sapiens (Human))	BDBM3832 (1-Phenylbenzimidazole deriv. 49 \| 4-(1H-1,3-benzod...) Show SMILES N#Cc1ccc(cc1)-n1cnc2ccccc12 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.60E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Auckland					Assay Description IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...				J Med Chem 41: 5457-65 (1998) Article DOI: 10.1021/jm9804681 BindingDB Entry DOI: 10.7270/Q24T6GJC
University of Auckland					More data for this Ligand-Target Pair
Fibroblast growth factor receptor 1 (Homo sapiens (Human))	BDBM3827 (1-(4-Carboxamidophenyl)benzimidazole \| 1-Phenylben...) Show SMILES NC(=O)c1ccc(cc1)-n1cnc2ccccc12 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>5.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Auckland					Assay Description IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...				J Med Chem 41: 5457-65 (1998) Article DOI: 10.1021/jm9804681 BindingDB Entry DOI: 10.7270/Q24T6GJC
University of Auckland					More data for this Ligand-Target Pair
Fibroblast growth factor receptor 1 (Homo sapiens (Human))	BDBM3828 (1-(4-nitrophenyl)-1H-1,3-benzodiazole \| 1-Phenylbe...) Show SMILES [O-][N+](=O)c1ccc(cc1)-n1cnc2ccccc12 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase MCE PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	>5.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Auckland					Assay Description IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...				J Med Chem 41: 5457-65 (1998) Article DOI: 10.1021/jm9804681 BindingDB Entry DOI: 10.7270/Q24T6GJC
University of Auckland					More data for this Ligand-Target Pair
Fibroblast growth factor receptor 1 (Homo sapiens (Human))	BDBM3829 (1-Phenylbenzimidazole deriv. 46 \| 4-(1H-1,3-benzod...) Show SMILES Nc1ccc(cc1)-n1cnc2ccccc12 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase MCE PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	>5.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Auckland					Assay Description IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...				J Med Chem 41: 5457-65 (1998) Article DOI: 10.1021/jm9804681 BindingDB Entry DOI: 10.7270/Q24T6GJC
University of Auckland					More data for this Ligand-Target Pair
Fibroblast growth factor receptor 1 (Homo sapiens (Human))	BDBM3830 (1-Phenylbenzimidazole deriv. 47 \| 1-[4-(1H-1,3-ben...) Show SMILES CC(=O)c1ccc(cc1)-n1cnc2ccccc12 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	>5.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Auckland					Assay Description IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...				J Med Chem 41: 5457-65 (1998) Article DOI: 10.1021/jm9804681 BindingDB Entry DOI: 10.7270/Q24T6GJC
University of Auckland					More data for this Ligand-Target Pair
Fibroblast growth factor receptor 1 (Homo sapiens (Human))	BDBM3831 (1-Phenylbenzimidazole deriv. 48 \| 4-(1H-1,3-benzod...) Show SMILES O=Cc1ccc(cc1)-n1cnc2ccccc12 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase MCE PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	>5.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Auckland					Assay Description IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...				J Med Chem 41: 5457-65 (1998) Article DOI: 10.1021/jm9804681 BindingDB Entry DOI: 10.7270/Q24T6GJC
University of Auckland					More data for this Ligand-Target Pair
Fibroblast growth factor receptor 1 (Homo sapiens (Human))	BDBM3832 (1-Phenylbenzimidazole deriv. 49 \| 4-(1H-1,3-benzod...) Show SMILES N#Cc1ccc(cc1)-n1cnc2ccccc12 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>5.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Auckland					Assay Description IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...				J Med Chem 41: 5457-65 (1998) Article DOI: 10.1021/jm9804681 BindingDB Entry DOI: 10.7270/Q24T6GJC
University of Auckland					More data for this Ligand-Target Pair
Platelet-derived growth factor receptor beta (Homo sapiens (Human))	BDBM3863 (1-Phenylbenzimidazole deriv. 80 \| methyl 1-phenyl-...) Show SMILES COC(=O)c1ccc2ncn(-c3ccccc3)c2c1 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	1.30E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Auckland					Assay Description IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...				J Med Chem 41: 5457-65 (1998) Article DOI: 10.1021/jm9804681 BindingDB Entry DOI: 10.7270/Q24T6GJC
University of Auckland					More data for this Ligand-Target Pair
Fibroblast growth factor receptor 1 (Homo sapiens (Human))	BDBM3863 (1-Phenylbenzimidazole deriv. 80 \| methyl 1-phenyl-...) Show SMILES COC(=O)c1ccc2ncn(-c3ccccc3)c2c1 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	>5.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Auckland					Assay Description IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...				J Med Chem 41: 5457-65 (1998) Article DOI: 10.1021/jm9804681 BindingDB Entry DOI: 10.7270/Q24T6GJC
University of Auckland					More data for this Ligand-Target Pair
Platelet-derived growth factor receptor beta (Homo sapiens (Human))	BDBM3794 (1-Phenylbenzimidazole 3 \| 1-Phenylbenzimidazole de...) Show SMILES c1nc2ccccc2n1-c1ccccc1 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase MCE PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	9.30E+3	n/a	n/a	n/a	n/a	7.4	25
University of Auckland					Assay Description IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...				J Med Chem 42: 2373-82 (1999) Article DOI: 10.1021/jm980658b BindingDB Entry DOI: 10.7270/Q2W957B2
University of Auckland					More data for this Ligand-Target Pair
Fibroblast growth factor receptor 1 (Homo sapiens (Human))	BDBM3794 (1-Phenylbenzimidazole 3 \| 1-Phenylbenzimidazole de...) Show SMILES c1nc2ccccc2n1-c1ccccc1 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase MCE PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	>5.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Auckland					Assay Description IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...				J Med Chem 42: 2373-82 (1999) Article DOI: 10.1021/jm980658b BindingDB Entry DOI: 10.7270/Q2W957B2
University of Auckland					More data for this Ligand-Target Pair
Platelet-derived growth factor receptor beta (Homo sapiens (Human))	BDBM3791 (1-Phenylbenzimidazole deriv. 8 \| 1-phenyl-1H-indol...) Show SMILES c1cc2ccccc2n1-c1ccccc1 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase MCE PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	>5.00E+4	n/a	n/a	n/a	n/a	7.4	25
University of Auckland					Assay Description IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...				J Med Chem 41: 5457-65 (1998) Article DOI: 10.1021/jm9804681 BindingDB Entry DOI: 10.7270/Q24T6GJC
University of Auckland					More data for this Ligand-Target Pair