Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50482402 (CHEMBL1209692) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 0.220 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet assessed as reduction of ADP-induced platelet aggregation | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50482409 (CHEMBL1208912) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 0.400 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet assessed as reduction of ADP-induced platelet aggregation | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50482414 (CHEMBL1208853) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 0.630 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet assessed as reduction of ADP-induced platelet aggregation | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50323320 (3-(3,4-dimethoxyphenyl)-3-(3-(1,2,3,4-tetrahydrois...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.700 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet assessed as reduction of ADP-induced platelet aggregation | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50482419 (CHEMBL1208980) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 0.780 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet assessed as reduction of ADP-induced platelet aggregation | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50323319 (3-(3-(carbamoyl)benzamido)-3-(4-methoxyphenyl)prop...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.800 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet assessed as reduction of ADP-induced platelet aggregation | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50482412 (CHEMBL1208850) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 0.900 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet assessed as reduction of ADP-induced platelet aggregation | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50323318 (3-(3-(carbamoyl)benzamido)-3-phenylpropanoic acid ...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet assessed as reduction of ADP-induced platelet aggregation | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50482403 (CHEMBL1209774) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet assessed as reduction of ADP-induced platelet aggregation | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50482404 (CHEMBL1209860) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet assessed as reduction of ADP-induced platelet aggregation | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50482415 (CHEMBL1209773) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.20 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet assessed as reduction of ADP-induced platelet aggregation | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50482400 (CHEMBL1209622) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.60 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet assessed as reduction of ADP-induced platelet aggregation | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50482407 (CHEMBL1208851) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.5 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet assessed as reduction of ADP-induced platelet aggregation | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50482416 (CHEMBL1209862) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet assessed as reduction of ADP-induced platelet aggregation | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50482411 (CHEMBL1208979) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet assessed as reduction of ADP-induced platelet aggregation | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50482401 (CHEMBL1209690) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet assessed as reduction of ADP-induced platelet aggregation | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50155250 (3-[3-(2,3-Dihydro-1H-isoindol-5-ylcarbamoyl)-propi...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8.30 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet assessed as reduction of ADP-induced platelet aggregation | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50482404 (CHEMBL1209860) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 8.90 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet rich plasma | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50482413 (CHEMBL1209691) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 9 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet assessed as reduction of ADP-induced platelet aggregation | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50323320 (3-(3,4-dimethoxyphenyl)-3-(3-(1,2,3,4-tetrahydrois...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet rich plasma | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50482403 (CHEMBL1209774) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 13 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet rich plasma | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50323319 (3-(3-(carbamoyl)benzamido)-3-(4-methoxyphenyl)prop...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 17 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet rich plasma | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50482410 (CHEMBL1208914) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet assessed as reduction of ADP-induced platelet aggregation | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50323318 (3-(3-(carbamoyl)benzamido)-3-phenylpropanoic acid ...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 25 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet rich plasma | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50482415 (CHEMBL1209773) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet rich plasma | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50482402 (CHEMBL1209692) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 31 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet rich plasma | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50482419 (CHEMBL1208980) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 53 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet rich plasma | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3 (Homo sapiens (Human)) | BDBM50254203 (2-((3S,6R,11R,14R,20S,28aS)-11-amino-3-(2-amino-2-...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 57 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description Binding affinity to integrin alpha3 (unknown origin) expressed in human MDA-MB-231 cells by flow cytometry | J Med Chem 52: 126-33 (2009) Article DOI: 10.1021/jm801062d BindingDB Entry DOI: 10.7270/Q2VM4C4F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50482414 (CHEMBL1208853) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 64 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet rich plasma | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50482406 (CHEMBL1209863) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 65 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet assessed as reduction of ADP-induced platelet aggregation | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3 (Homo sapiens (Human)) | BDBM50254205 (2-((3S,6R,11R,14R,20S,28aS)-11-amino-6-carbamoyl-2...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 68 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description Binding affinity to integrin alpha3 (unknown origin) expressed in human MDA-MB-231 cells by flow cytometry | J Med Chem 52: 126-33 (2009) Article DOI: 10.1021/jm801062d BindingDB Entry DOI: 10.7270/Q2VM4C4F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50482408 (CHEMBL1208852) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 87 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet rich plasma | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50482409 (CHEMBL1208912) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 90 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet rich plasma | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50482412 (CHEMBL1208850) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 96 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet rich plasma | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50482401 (CHEMBL1209690) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 105 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet rich plasma | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50482411 (CHEMBL1208979) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 127 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet rich plasma | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50482400 (CHEMBL1209622) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 160 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet rich plasma | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3 (Homo sapiens (Human)) | BDBM50254204 (2-((3S,6R,11R,14R,20S,28aS)-11-amino-6-carbamoyl-2...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 190 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description Binding affinity to integrin alpha3 (unknown origin) expressed in human MDA-MB-231 cells by flow cytometry | J Med Chem 52: 126-33 (2009) Article DOI: 10.1021/jm801062d BindingDB Entry DOI: 10.7270/Q2VM4C4F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3 (Homo sapiens (Human)) | BDBM50254206 (2-((3S,6R,11R,14R,20S,28aS)-11-amino-6-carbamoyl-2...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 220 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description Binding affinity to integrin alpha3 (unknown origin) expressed in human MDA-MB-231 cells by flow cytometry | J Med Chem 52: 126-33 (2009) Article DOI: 10.1021/jm801062d BindingDB Entry DOI: 10.7270/Q2VM4C4F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3 (Homo sapiens (Human)) | BDBM50254208 (2-((3S,6R,11R,14R,20S,28aS)-11-amino-6-carbamoyl-2...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 290 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description Binding affinity to integrin alpha3 (unknown origin) expressed in human MDA-MB-231 cells by flow cytometry | J Med Chem 52: 126-33 (2009) Article DOI: 10.1021/jm801062d BindingDB Entry DOI: 10.7270/Q2VM4C4F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50482407 (CHEMBL1208851) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 310 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet rich plasma | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3 (Homo sapiens (Human)) | BDBM50254207 (2-((3S,6R,11R,14R,20S,28aS)-11-amino-6-carbamoyl-2...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 340 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description Binding affinity to integrin alpha3 (unknown origin) expressed in human MDA-MB-231 cells by flow cytometry | J Med Chem 52: 126-33 (2009) Article DOI: 10.1021/jm801062d BindingDB Entry DOI: 10.7270/Q2VM4C4F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50482418 (CHEMBL1208911) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 510 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet rich plasma | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3 (Homo sapiens (Human)) | BDBM50254202 (2-((3S,6R,11R,14R,20S,28aS)-11-amino-3-(2-amino-2-...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 550 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description Binding affinity to integrin alpha3 (unknown origin) expressed in human MDA-MB-231 cells by flow cytometry | J Med Chem 52: 126-33 (2009) Article DOI: 10.1021/jm801062d BindingDB Entry DOI: 10.7270/Q2VM4C4F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50482416 (CHEMBL1209862) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 570 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet rich plasma | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50155250 (3-[3-(2,3-Dihydro-1H-isoindol-5-ylcarbamoyl)-propi...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 860 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet rich plasma | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50482413 (CHEMBL1209691) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 890 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet rich plasma | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50482405 (CHEMBL1209861) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet assessed as reduction of ADP-induced platelet aggregation | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50482406 (CHEMBL1209863) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet rich plasma | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Integrin alpha-3/beta-3 (Homo sapiens (Human)) | BDBM50482410 (CHEMBL1208914) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine Curated by ChEMBL | Assay Description Antagonist activity at FITC-tagged alpha3beta3 integrin in human platelet rich plasma | Bioorg Med Chem Lett 20: 4444-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.051 BindingDB Entry DOI: 10.7270/Q2H134T5 | |||||||||||
More data for this Ligand-Target Pair |
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