Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Catenin beta-1/Transcription factor 7-like 2 (Homo sapiens (Human)) | BDBM40314 (3-(4-Chloro-phenyl)-1,6-dimethyl-1H-pyrimido[5,4-e...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 300 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Michigan Curated by ChEMBL | Assay Description Inhibition of human TCF4/ flag epitope-tagged beta-catenin (unknown origin) interaction transfected in human HCT116 cells after 24 hrs by beta-galact... | Bioorg Med Chem Lett 23: 5814-20 (2013) Article DOI: 10.1016/j.bmcl.2013.08.111 BindingDB Entry DOI: 10.7270/Q2RV0Q4J | |||||||||||
More data for this Ligand-Target Pair |