Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Telomere resolvase ResT (Borrelia burgdorferi) | BDBM50335561 ((R)-4-((5S,8R,9S,10S,13S,14S,17R)-10,13-dimethylhe...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.96E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Calgary Curated by ChEMBL | Assay Description Inhibition of Borrelia burgdorferi telomere resolvase by gel-based telomere resolution assay | Antimicrob Agents Chemother 53: 4441-9 (2009) Article DOI: 10.1128/AAC.00529-09 BindingDB Entry DOI: 10.7270/Q26W9BBG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Telomere resolvase ResT (Borrelia burgdorferi) | BDBM50335562 (13-(cyclopent-2-enyl)tridecanoic acid | CHEMBL1649...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 2.62E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Calgary Curated by ChEMBL | Assay Description Inhibition of Borrelia burgdorferi telomere resolvase by gel-based telomere resolution assay | Antimicrob Agents Chemother 53: 4441-9 (2009) Article DOI: 10.1128/AAC.00529-09 BindingDB Entry DOI: 10.7270/Q26W9BBG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Telomere resolvase ResT (Borrelia burgdorferi) | BDBM50335560 (2,2'-(3,4,6-trihydroxy-5-oxo-5H-benzo[7]annulene-1...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.73E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Calgary Curated by ChEMBL | Assay Description Inhibition of Borrelia burgdorferi telomere resolvase by gel-based telomere resolution assay | Antimicrob Agents Chemother 53: 4441-9 (2009) Article DOI: 10.1128/AAC.00529-09 BindingDB Entry DOI: 10.7270/Q26W9BBG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Telomere resolvase ResT (Borrelia burgdorferi) | BDBM50335558 (2-(4-(6-(6-carboxy-1,3-dioxo-1H-benzo[de]isoquinol...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.16E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Calgary Curated by ChEMBL | Assay Description Inhibition of Borrelia burgdorferi telomere resolvase by gel-based telomere resolution assay | Antimicrob Agents Chemother 53: 4441-9 (2009) Article DOI: 10.1128/AAC.00529-09 BindingDB Entry DOI: 10.7270/Q26W9BBG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Telomere resolvase ResT (Borrelia burgdorferi) | BDBM50096619 (1,8,9-Trihydroxy-3-methoxy-benzo[4,5]furo[3,2-c]ch...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 8.67E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Calgary Curated by ChEMBL | Assay Description Inhibition of Borrelia burgdorferi telomere resolvase by gel-based telomere resolution assay | Antimicrob Agents Chemother 53: 4441-9 (2009) Article DOI: 10.1128/AAC.00529-09 BindingDB Entry DOI: 10.7270/Q26W9BBG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Telomere resolvase ResT (Borrelia burgdorferi) | BDBM50335559 (4-(4,5-di(biphenyl-4-yl)-1H-imidazol-2-yl)benzoic ...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.52E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Calgary Curated by ChEMBL | Assay Description Inhibition of Borrelia burgdorferi telomere resolvase by gel-based telomere resolution assay | Antimicrob Agents Chemother 53: 4441-9 (2009) Article DOI: 10.1128/AAC.00529-09 BindingDB Entry DOI: 10.7270/Q26W9BBG | |||||||||||
More data for this Ligand-Target Pair |