Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Deoxyribonuclease-2-alpha (Homo sapiens (Human)) | BDBM50326048 ((2R,5S,8S,11S,14S,17S,20S,23S,26S,29S,32S,35R)-8,1...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 200 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Laboratory of Molecular Biology, Medical Research Council Curated by ChEMBL | Assay Description Binding affinity to Dnase 2 | Nat Chem Biol 5: 502-7 (2009) Article DOI: 10.1038/nchembio.184 BindingDB Entry DOI: 10.7270/Q2Z60P9P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Deoxyribonuclease-2-alpha (Sus scrofa) | BDBM22984 ((8S,10S)-10-{[(2R,4S,5S,6S)-4-amino-5-hydroxy-6-me...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | PubMed | n/a | n/a | >2.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kumamoto University Curated by ChEMBL | Assay Description Inhibition of porcine spleen DNase 2 assessed as undigested supercoiled pBR322 DNA concentration | J Nat Prod 64: 204-7 (2001) BindingDB Entry DOI: 10.7270/Q2W37W21 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Deoxyribonuclease-2-alpha (Sus scrofa) | BDBM50242374 (CHEMBL505529 | topostatin) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem | PubMed | n/a | n/a | >2.50E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kumamoto University Curated by ChEMBL | Assay Description Inhibition of porcine spleen DNase 2 assessed as undigested supercoiled pBR322 DNA concentration | J Nat Prod 64: 204-7 (2001) BindingDB Entry DOI: 10.7270/Q2W37W21 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Deoxyribonuclease-2-alpha (Sus scrofa) | BDBM50008923 ((S)-4-ethyl-4-hydroxy-1,12-dihydro-4H-2-oxa-6,12a-...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid PDB UniChem Patents Similars | PubMed | n/a | n/a | >3.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kumamoto University Curated by ChEMBL | Assay Description Inhibition of porcine spleen DNase 2 assessed as undigested supercoiled pBR322 DNA concentration | J Nat Prod 64: 204-7 (2001) BindingDB Entry DOI: 10.7270/Q2W37W21 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Deoxyribonuclease-2-alpha (Sus scrofa) | BDBM50164888 (6-Hydroxy-3-[1-(4-hydroxy-phenyl)-meth-(E)-ylidene...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >4.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kumamoto University Curated by ChEMBL | Assay Description Inhibition of porcine spleen DNase 2 assessed as undigested supercoiled pBR322 DNA concentration | J Nat Prod 64: 204-7 (2001) BindingDB Entry DOI: 10.7270/Q2W37W21 | |||||||||||
More data for this Ligand-Target Pair |