Compile Data Set for Download or QSAR

Found 253 hits Enz. Inhib. hit(s) with Target = 'Gamma-aminobutyric acid receptor subunit gamma-1'   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM50021185 (5-Aminomethyl-4,5-dihydro-isoxazol-3-ol | CHEMBL42...) Show SMILES NC[C@@H]1CC(O)=NO1 |c:5| Show InChI InChI=1S/C4H8N2O2/c5-2-3-1-4(7)6-8-3/h3H,1-2,5H2,(H,6,7)/t3-/m0/s1	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	4	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description In vitro inhibition of [3H]-GABA binding to Gamma-aminobutyric-acid receptor of rat brain synaptic membranes				J Med Chem 28: 1612-7 (1985) BindingDB Entry DOI: 10.7270/Q2PN94NZ
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM50000766 (CHEMBL12 | DIAZEPAM | US9271961, Diazepam) Show SMILES CN1c2ccc(Cl)cc2C(=NCC1=O)c1ccccc1 |c:10| Show InChI InChI=1S/C16H13ClN2O/c1-19-14-8-7-12(17)9-13(14)16(18-10-15(19)20)11-5-3-2-4-6-11/h2-9H,10H2,1H3	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	Purchase CHEMBL DrugBank KEGG MMDB PC cid PC sid PDB UniChem Patents Similars	PubMed	n/a	n/a	5	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Anxiolytic activity by displacement of [3H]diazepam from GABA-A receptor in rat synaptosomal membranes				J Med Chem 23: 952-5 (1980) BindingDB Entry DOI: 10.7270/Q25X27ZP
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM23183 (5-(aminomethyl)-1,2-oxazol-3-ol | Agarin | CHEMBL2...) Show SMILES NCc1cc(=O)[nH]o1 Show InChI InChI=1S/C4H6N2O2/c5-2-3-1-4(7)6-8-3/h1H,2,5H2,(H,6,7)	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	Purchase CHEMBL KEGG PC cid PC sid UniChem Patents	PubMed	n/a	n/a	6	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description In vitro inhibition of [3H]-GABA binding to Gamma-aminobutyric-acid receptor of rat brain synaptic membranes				J Med Chem 28: 1612-7 (1985) BindingDB Entry DOI: 10.7270/Q2PN94NZ
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM585854 (US11530237, Compound 10 | US11542297, Compound 10) Show SMILES C[C@]12CC[C@H]3[C@@H](CC[C@@H]4C[C@](C)(O)CC[C@]34C)[C@@H]1CC[C@@H]2C(=O)Cn1cc(cn1)C#N |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM585855 (US11530237, Compound 11 | US11542297, Compound 11) Show SMILES C[C@]12CC[C@H]3[C@@H](CC[C@@H]4C[C@](C)(O)CC[C@]34C)[C@@H]1CC[C@@H]2C(=O)Cn1nc2ccccc2n1 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM585856 (US11530237, Compound 12 | US11542297, Compound 12) Show SMILES C[C@]12CC[C@H]3[C@@H](CC[C@@H]4C[C@](C)(O)CC[C@]34C)[C@@H]1CC[C@@H]2C(=O)Cn1nnc2ccccc12 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM585858 (US11530237, Compound 14 | US11542297, Compound 14) Show SMILES COc1ccc2nn(CC(=O)[C@H]3CC[C@H]4[C@@H]5CC[C@@H]6C[C@](C)(O)CC[C@]6(C)[C@H]5CC[C@]34C)nc2c1 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM585859 (US11530237, Compound 15 | US11542297, Compound 15) Show SMILES COc1ccc2n(CC(=O)[C@H]3CC[C@H]4[C@@H]5CC[C@@H]6C[C@](C)(O)CC[C@]6(C)[C@H]5CC[C@]34C)nnc2c1 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM585877 (US11530237, Compound 35 | US11542297, Compound 35) Show SMILES C[C@]12CC[C@H]3[C@@H](CC[C@@H]4C[C@](C)(O)CC[C@]34C)[C@@H]1CC[C@@H]2C(=O)Cn1nc2ccc(Cl)cc2n1 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM588646 (US11542297, Compound 50) Show SMILES C[C@]12CC[C@H]3[C@@H](CC[C@@H]4C[C@](C)(O)CC[C@]34C)[C@@H]1CC[C@@H]2C(=O)Cn1nc2cc(Cl)cnc2n1 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM585895 (US11530237, Compound 54 | US11542297, Compound 54) Show SMILES C[C@]12CC[C@H]3[C@@H](CC[C@@H]4C[C@](C)(O)CC[C@]34C)[C@@H]1CC[C@@H]2C(=O)Cn1ncnn1 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM585946 (US11530237, Compound 117 | US11542297, Compound 11...) Show SMILES COc1cccc2nn(CC(=O)[C@H]3CC[C@H]4[C@@H]5CC[C@H]6C[C@](C)(O)CC[C@]6(C)[C@H]5CC[C@]34C)nc12 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM588727 (US11542297, Compound 146) Show SMILES C[C@]12CC[C@H]3[C@@H](CC[C@@H]4C[C@](C)(O)CC[C@]34C)[C@@H]1CC[C@@H]2C(=O)Cn1cc(cn1)[N+]([O-])=O |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM586009 (US11530237, Compound 185 | US11542297, Compound 18...) Show SMILES COC[C@@]1(O)CC[C@@]2(C)[C@@H](CC[C@H]3[C@@H]4CC[C@H](C(=O)Cn5nnc6ccc(Cl)cc56)[C@@]4(C)CC[C@H]23)C1 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM585860 (US11530237, Compound 16 | US11542297, Compound 16) Show SMILES COc1ccc2nnn(CC(=O)[C@H]3CC[C@H]4[C@@H]5CC[C@@H]6C[C@](C)(O)CC[C@]6(C)[C@H]5CC[C@]34C)c2c1 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM585862 (US11530237, Compound 18 | US11542297, Compound 18) Show SMILES C[C@]12CC[C@H]3[C@@H](CC[C@@H]4C[C@](C)(O)CC[C@]34C)[C@@H]1CC[C@@H]2C(=O)Cn1nnc2c(F)cccc12 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM585863 (US11530237, Compound 19 | US11542297, Compound 19) Show SMILES C[C@]12CC[C@H]3[C@@H](CC[C@@H]4C[C@](C)(O)CC[C@]34C)[C@@H]1CC[C@@H]2C(=O)Cn1ccc(n1)C(F)(F)F |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM585864 (US11530237, Compound 21 | US11542297, Compound 21) Show SMILES C[C@]12CC[C@H]3[C@@H](CC[C@@H]4C[C@](C)(O)CC[C@]34C)[C@@H]1CC[C@@H]2C(=O)Cn1nc2ccc(F)cc2n1 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM585865 (US11530237, Compound 22 | US11542297, Compound 22) Show SMILES C[C@]12CC[C@H]3[C@@H](CC[C@@H]4C[C@](C)(O)CC[C@]34C)[C@@H]1CC[C@@H]2C(=O)Cn1nnc2ccc(F)cc12 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM585866 (US11530237, Compound 23 | US11542297, Compound 23) Show SMILES C[C@]12CC[C@H]3[C@@H](CC[C@@H]4C[C@](C)(O)CC[C@]34C)[C@@H]1CC[C@@H]2C(=O)Cn1nnc2cc(F)ccc12 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM585867 (US11530237, Compound 24 | US11542297, Compound 24) Show SMILES C[C@]12CC[C@H]3[C@@H](CC[C@@H]4C[C@](C)(O)CC[C@]34C)[C@@H]1CC[C@@H]2C(=O)Cn1ccc(n1)C#N |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM585868 (US11530237, Compound 26 | US11542297, Compound 26) Show SMILES C[C@]12CC[C@H]3[C@@H](CC[C@@H]4C[C@](C)(O)CC[C@]34C)[C@@H]1CC[C@@H]2C(=O)Cn1cc2ccccc2n1 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM585870 (US11530237, Compound 28 | US11542297, Compound 28) Show SMILES C[C@]12CC[C@H]3[C@@H](CC[C@@H]4C[C@](C)(O)CC[C@]34C)[C@@H]1CC[C@@H]2C(=O)Cn1nc2cc(F)cc(F)c2n1 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM585871 (US11530237, Compound 29 | US11542297, Compound 29) Show SMILES C[C@]12CC[C@H]3[C@@H](CC[C@@H]4C[C@](C)(O)CC[C@]34C)[C@@H]1CC[C@@H]2C(=O)Cn1nnc2cc(F)cc(F)c12 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM588629 (US11542297, Compound 32) Show SMILES Cc1nnn(CC(=O)[C@H]2CC[C@H]3[C@@H]4CC[C@@H]5C[C@](C)(O)CC[C@]5(C)[C@H]4CC[C@]23C)n1 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM585878 (US11530237, Compound 36 | US11542297, Compound 36) Show SMILES C[C@]12CC[C@H]3[C@@H](CC[C@@H]4C[C@](C)(O)CC[C@]34C)[C@@H]1CC[C@@H]2C(=O)Cn1nnc2ccc(Cl)cc12 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM585882 (US11530237, Compound 40 | US11542297, Compound 40) Show SMILES CCO[C@H]1C[C@@]2(C)[C@@H](CC[C@H]3[C@@H]4CC[C@H](C(=O)Cn5ccc(n5)C(=O)OCC)[C@@]4(C)CC[C@H]23)C[C@@H]1O |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM585886 (US11530237, Compound 45 | US11542297, Compound 45) Show SMILES COc1cccc2n(CC(=O)[C@H]3CC[C@H]4[C@@H]5CC[C@@H]6C[C@](C)(O)CC[C@]6(C)[C@H]5CC[C@]34C)nnc12 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM585894 (US11530237, Compound 53 | US11542297, Compound 53) Show SMILES C[C@]12CC[C@H]3[C@@H](CC[C@@H]4C[C@](C)(O)CC[C@]34C)[C@@H]1CC[C@@H]2C(=O)Cn1nc2ccc(Cl)c(F)c2n1 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM585915 (US11530237, Compound 74 | US11542297, Compound 74) Show SMILES CSc1ccc2nn(CC(=O)[C@H]3CC[C@H]4[C@@H]5CC[C@@H]6C[C@](C)(O)CC[C@]6(C)[C@H]5CC[C@]34C)nc2c1 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM585919 (US11530237, Compound 78 | US11542297, Compound 78) Show SMILES C[C@]12CC[C@H]3[C@@H](CC[C@@H]4C[C@](C)(O)CC[C@]34C)[C@@H]1CC[C@@H]2C(=O)Cn1nnc2c(F)c(F)ccc12 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM588678 (US11542297, Compound 86) Show SMILES CN(C)C(=O)c1cnn(CC(=O)[C@H]2CC[C@H]3[C@@H]4CC[C@H]5C[C@](C)(O)CC[C@]5(C)[C@H]4CC[C@]23C)c1 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM588688 (US11542297, Compound 103) Show SMILES CS(=O)c1ccc2nn(CC(=O)[C@H]3CC[C@H]4[C@@H]5CC[C@@H]6C[C@](C)(O)CC[C@]6(C)[C@H]5CC[C@]34C)nc2c1 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM588689 (US11542297, Compound 104) Show SMILES C[C@]12CC[C@H]3[C@@H](CC[C@@H]4C[C@](C)(O)CC[C@]34C)[C@@H]1CC[C@@H]2C(=O)Cn1nc2ccc(cc2n1)S(C)(=O)=O |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM585951 (US11530237, Compound 124 | US11542297, Compound 12...) Show SMILES C[C@]12CC[C@H]3[C@@H](CC[C@H]4C[C@](C)(O)CC[C@]34C)[C@@H]1CC[C@@H]2C(=O)Cn1nnc2cc(F)c(F)cc12 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM585939 (US11530237, Compound 110 | US11530237, Compound 12...) Show SMILES C[C@]12CC[C@H]3[C@@H](CC[C@H]4C[C@](C)(O)CC[C@]34C)[C@@H]1CC[C@@H]2C(=O)Cn1nc2cccc(F)c2n1 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM585959 (US11530237, Compound 133 | US11542297, Compound 13...) Show SMILES C[C@]12CC[C@H]3[C@@H](CC[C@@H]4C[C@](C)(O)CC[C@]34C)[C@@H]1CC[C@@H]2C(=O)Cn1cc(Cl)cn1 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM585990 (US11530237, Compound 165 | US11542297, Compound 16...) Show SMILES COC[C@@]1(O)CC[C@@]2(C)[C@@H](CC[C@H]3[C@@H]4CC[C@H](C(=O)Cn5nc6ccc(Cl)cc6n5)[C@@]4(C)CC[C@H]23)C1 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM586015 (US11530237, Compound 191 | US11542297, Compound 19...) Show SMILES COC[C@@]1(O)CC[C@@]2(C)[C@@H](CC[C@H]3[C@@H]4CC[C@H](C(=O)Cn5cc6cc(Cl)ccc6n5)[C@@]4(C)CC[C@H]23)C1 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM586026 (US11530237, Compound 204 | US11542297, Compound 20...) Show SMILES CCOC(=O)c1cnn(CC(=O)[C@H]2CC[C@H]3[C@@H]4CC[C@@H]5C[C@](C)(O)CC[C@]5(C)[C@H]4CC[C@]23C)c1 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM585939 (US11530237, Compound 110 | US11530237, Compound 12...) Show SMILES C[C@]12CC[C@H]3[C@@H](CC[C@H]4C[C@](C)(O)CC[C@]34C)[C@@H]1CC[C@@H]2C(=O)Cn1nc2cccc(F)c2n1 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM588823 (US11542297, Compound 248) Show SMILES CSc1ccc2cnn(CC(=O)[C@H]3CC[C@H]4[C@@H]5CC[C@H]6C[C@](C)(O)CC[C@]6(C)[C@H]5CC[C@]34C)c2c1 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM586067 (US11530237, Compound 248 | US11542297, Compound 24...) Show SMILES CSc1ccc2nn(CC(=O)[C@H]3CC[C@H]4[C@@H]5CC[C@H]6C[C@](C)(O)CC[C@]6(C)[C@H]5CC[C@]34C)nc2c1 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM586078 (US11530237, Compound 259 | US11542297, Compound 25...) Show SMILES C[C@]12CC[C@H]3[C@@H](CC[C@@H]4C[C@](C)(O)CC[C@]34C)[C@@H]1CC[C@@H]2C(=O)Cn1cnc(F)c1 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM586079 (US11530237, Compound 260 | US11542297, Compound 26...) Show SMILES CCCN(C)C(=O)c1cnn(CC(=O)[C@H]2CC[C@H]3[C@@H]4CC[C@@H]5C[C@](C)(O)CC[C@]5(C)[C@H]4CC[C@]23C)n1 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM50018800 (4-tert-Butyl-1-(4-ethynyl-phenyl)-2,6,7-trioxa-bic...) Show SMILES CC(C)(C)C12COC(OC1)(OC2C#N)c1ccc(cc1)C#C Show InChI InChI=1S/C18H19NO3/c1-5-13-6-8-14(9-7-13)18-20-11-17(12-21-18,16(2,3)4)15(10-19)22-18/h1,6-9,15H,11-12H2,2-4H3	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents	PubMed	n/a	n/a	25	n/a	n/a	n/a	n/a	n/a	n/a
University of California Curated by ChEMBL					Assay Description Inhibition of GABA-stimulated 36Cl- uptakeby membrane vesicles of rat cerebral cortex				J Med Chem 31: 1064-6 (1988) BindingDB Entry DOI: 10.7270/Q2VH5MTN
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM585970 (US11530237, Compound 145 | US11542297, Compound 14...) Show SMILES CCOc1cnn(CC(=O)[C@H]2CC[C@H]3[C@@H]4CC[C@@H]5C[C@](C)(O)CC[C@]5(C)[C@H]4CC[C@]23C)c1 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	30	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM585972 (US11530237, Compound 147 | US11542297, Compound 14...) Show SMILES Cc1cnn(CC(=O)[C@H]2CC[C@H]3[C@@H]4CC[C@@H]5C[C@](C)(O)CC[C@]5(C)[C@H]4CC[C@]23C)c1 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	30	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM585973 (US11530237, Compound 148 | US11542297, Compound 14...) Show SMILES COc1cnn(CC(=O)[C@H]2CC[C@H]3[C@@H]4CC[C@H]5C[C@](C)(O)CC[C@]5(C)[C@H]4CC[C@]23C)c1 |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	30	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair
Gamma-aminobutyric acid receptor subunit gamma-1 (Rattus norvegicus)	BDBM588732 (US11542297, Compound 151) Show SMILES C[C@]12CC[C@H]3[C@@H](CC[C@H]4C[C@](C)(O)CC[C@]34C)[C@@H]1CC[C@@H]2C(=O)Cn1cc(cn1)[N+](O)=O |r| Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	UniChem	US Patent	n/a	n/a	30	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...				Citation and Details BindingDB Entry DOI: 10.7270/Q2VD73BW
					More data for this Ligand-Target Pair

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