Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Low-density lipoprotein receptor-related protein 6 (Homo sapiens (Human)) | BDBM50135174 (CHEMBL3747431) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Aristotle University of Thessaloniki Curated by ChEMBL | Assay Description Binding affinity to human LRP6 expressed in HEK293 cells assessed as inhibition of DKK1/LRP6 interaction using compound pre-treated DKK1 conditioned ... | Bioorg Med Chem 24: 1014-22 (2016) Article DOI: 10.1016/j.bmc.2016.01.025 BindingDB Entry DOI: 10.7270/Q2J67JRS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Low-density lipoprotein receptor-related protein 6 (Homo sapiens (Human)) | BDBM50145410 (CHEMBL3764819) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.38E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Aristotle University of Thessaloniki Curated by ChEMBL | Assay Description Binding affinity to human LRP6 expressed in HEK293 cells assessed as inhibition of DKK1/LRP6 interaction using compound pre-treated DKK1 conditioned ... | Bioorg Med Chem 24: 1014-22 (2016) Article DOI: 10.1016/j.bmc.2016.01.025 BindingDB Entry DOI: 10.7270/Q2J67JRS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Low-density lipoprotein receptor-related protein 6 (Homo sapiens (Human)) | BDBM50145403 (CHEMBL3764323) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.74E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Aristotle University of Thessaloniki Curated by ChEMBL | Assay Description Binding affinity to human LRP6 expressed in HEK293 cells assessed as inhibition of DKK1/LRP6 interaction using compound pre-treated DKK1 conditioned ... | Bioorg Med Chem 24: 1014-22 (2016) Article DOI: 10.1016/j.bmc.2016.01.025 BindingDB Entry DOI: 10.7270/Q2J67JRS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Low-density lipoprotein receptor-related protein 6 (Homo sapiens (Human)) | BDBM50145379 (CHEMBL3765769) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.77E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Aristotle University of Thessaloniki Curated by ChEMBL | Assay Description Binding affinity to human LRP6 expressed in HEK293 cells assessed as inhibition of DKK1/LRP6 interaction using compound pre-treated DKK1 conditioned ... | Bioorg Med Chem 24: 1014-22 (2016) Article DOI: 10.1016/j.bmc.2016.01.025 BindingDB Entry DOI: 10.7270/Q2J67JRS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Low-density lipoprotein receptor-related protein 6 (Homo sapiens (Human)) | BDBM50145384 (CHEMBL3764205) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.06E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Aristotle University of Thessaloniki Curated by ChEMBL | Assay Description Binding affinity to human LRP6 expressed in HEK293 cells assessed as inhibition of DKK1/LRP6 interaction using compound pre-treated DKK1 conditioned ... | Bioorg Med Chem 24: 1014-22 (2016) Article DOI: 10.1016/j.bmc.2016.01.025 BindingDB Entry DOI: 10.7270/Q2J67JRS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Low-density lipoprotein receptor-related protein 6 (Homo sapiens (Human)) | BDBM50145382 (CHEMBL3765415) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.33E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Aristotle University of Thessaloniki Curated by ChEMBL | Assay Description Binding affinity to human LRP6 expressed in HEK293 cells assessed as inhibition of DKK1/LRP6 interaction using compound pre-treated DKK1 conditioned ... | Bioorg Med Chem 24: 1014-22 (2016) Article DOI: 10.1016/j.bmc.2016.01.025 BindingDB Entry DOI: 10.7270/Q2J67JRS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Low-density lipoprotein receptor-related protein 6 (Homo sapiens (Human)) | BDBM50145409 (CHEMBL3765394) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.61E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Aristotle University of Thessaloniki Curated by ChEMBL | Assay Description Binding affinity to human LRP6 expressed in HEK293 cells assessed as inhibition of DKK1/LRP6 interaction using compound pre-treated DKK1 conditioned ... | Bioorg Med Chem 24: 1014-22 (2016) Article DOI: 10.1016/j.bmc.2016.01.025 BindingDB Entry DOI: 10.7270/Q2J67JRS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Low-density lipoprotein receptor-related protein 6 (Homo sapiens (Human)) | BDBM50145380 (CHEMBL3765591) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.71E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Aristotle University of Thessaloniki Curated by ChEMBL | Assay Description Binding affinity to human LRP6 expressed in HEK293 cells assessed as inhibition of DKK1/LRP6 interaction using compound pre-treated DKK1 conditioned ... | Bioorg Med Chem 24: 1014-22 (2016) Article DOI: 10.1016/j.bmc.2016.01.025 BindingDB Entry DOI: 10.7270/Q2J67JRS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Low-density lipoprotein receptor-related protein 6 (Homo sapiens (Human)) | BDBM50145381 (CHEMBL3763214) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.87E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Aristotle University of Thessaloniki Curated by ChEMBL | Assay Description Binding affinity to human LRP6 expressed in HEK293 cells assessed as inhibition of DKK1/LRP6 interaction using compound pre-treated DKK1 conditioned ... | Bioorg Med Chem 24: 1014-22 (2016) Article DOI: 10.1016/j.bmc.2016.01.025 BindingDB Entry DOI: 10.7270/Q2J67JRS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Low-density lipoprotein receptor-related protein 6 (Homo sapiens (Human)) | BDBM50145377 (CHEMBL3764713) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.23E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Aristotle University of Thessaloniki Curated by ChEMBL | Assay Description Binding affinity to human LRP6 expressed in HEK293 cells assessed as inhibition of DKK1/LRP6 interaction using compound pre-treated DKK1 conditioned ... | Bioorg Med Chem 24: 1014-22 (2016) Article DOI: 10.1016/j.bmc.2016.01.025 BindingDB Entry DOI: 10.7270/Q2J67JRS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Low-density lipoprotein receptor-related protein 6 (Homo sapiens (Human)) | BDBM50145383 (CHEMBL3763953) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Aristotle University of Thessaloniki Curated by ChEMBL | Assay Description Binding affinity to human LRP6 expressed in HEK293 cells assessed as inhibition of DKK1/LRP6 interaction using compound pre-treated DKK1 conditioned ... | Bioorg Med Chem 24: 1014-22 (2016) Article DOI: 10.1016/j.bmc.2016.01.025 BindingDB Entry DOI: 10.7270/Q2J67JRS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Low-density lipoprotein receptor-related protein 6 (Homo sapiens (Human)) | BDBM50145378 (CHEMBL3764972) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.16E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Aristotle University of Thessaloniki Curated by ChEMBL | Assay Description Binding affinity to human LRP6 expressed in HEK293 cells assessed as inhibition of DKK1/LRP6 interaction using compound pre-treated DKK1 conditioned ... | Bioorg Med Chem 24: 1014-22 (2016) Article DOI: 10.1016/j.bmc.2016.01.025 BindingDB Entry DOI: 10.7270/Q2J67JRS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Low-density lipoprotein receptor-related protein 6 (Homo sapiens (Human)) | BDBM50135174 (CHEMBL3747431) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.38E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Aristotle University of Thessaloniki Curated by ChEMBL | Assay Description Binding affinity to human LRP6 expressed in HEK293 cells assessed as inhibition of DKK1/LRP6 interaction using compound pre-treated DKK1 conditioned ... | Bioorg Med Chem 24: 1014-22 (2016) Article DOI: 10.1016/j.bmc.2016.01.025 BindingDB Entry DOI: 10.7270/Q2J67JRS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Low-density lipoprotein receptor (Homo sapiens (Human)) | BDBM50052689 (CHEMBL115205 | N-[5-(4-Cyclohexyl-butyrylamino)-2-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 4.00E+3 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Concentration at which one-half of the maximum Low density lipoprotein receptor is upregulated in HepG2 cells | J Med Chem 39: 3343-56 (1996) Article DOI: 10.1021/jm960153q BindingDB Entry DOI: 10.7270/Q2FT8K4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Low-density lipoprotein receptor (Homo sapiens (Human)) | BDBM50052691 (CHEMBL114199 | N-[5-(4-Cyclohexyl-butyryl)-2-methy...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Concentration at which one-half the maximum Low density lipoprotein receptor upregulation is observed in HepG2 cells | J Med Chem 39: 3343-56 (1996) Article DOI: 10.1021/jm960153q BindingDB Entry DOI: 10.7270/Q2FT8K4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Low-density lipoprotein receptor (Homo sapiens (Human)) | BDBM50052692 (5-(3-Cyclohexyl-propionylamino)-N-(4-hydroxy-pheny...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 7.00E+3 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Concentration at which one-half of the maximum Low density lipoprotein receptor is upregulated in HepG2 cells | J Med Chem 39: 3343-56 (1996) Article DOI: 10.1021/jm960153q BindingDB Entry DOI: 10.7270/Q2FT8K4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Low-density lipoprotein receptor (Homo sapiens (Human)) | BDBM50052690 (Acetic acid 4-[5-(3-cyclohexyl-propionylamino)-2-m...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.50E+3 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Concentration at which one-half of the maximum Low density lipoprotein receptor is upregulated in HepG2 cells | J Med Chem 39: 3343-56 (1996) Article DOI: 10.1021/jm960153q BindingDB Entry DOI: 10.7270/Q2FT8K4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Low-density lipoprotein receptor (Homo sapiens (Human)) | BDBM50052687 (CHEMBL114705 | N-[5-(3-Cyclohexyl-propionylamino)-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Concentration at which one-half of the maximum Low density lipoprotein receptor is upregulated in HepG2 cells | J Med Chem 39: 3343-56 (1996) Article DOI: 10.1021/jm960153q BindingDB Entry DOI: 10.7270/Q2FT8K4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Low-density lipoprotein receptor (Homo sapiens (Human)) | BDBM50052686 (CHEMBL115992 | N-{3-[(Benzo[1,3]dioxol-5-ylmethyl)...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 600 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Concentration at which one-half of the maximum Low density lipoprotein receptor is upregulated in HepG2 cells | J Med Chem 39: 3343-56 (1996) Article DOI: 10.1021/jm960153q BindingDB Entry DOI: 10.7270/Q2FT8K4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Low-density lipoprotein receptor (Homo sapiens (Human)) | BDBM50052688 (CHEMBL419042 | N-[5-(3-Cyclohexyl-propionylamino)-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Concentration at which one-half of the maximum Low density lipoprotein receptor is upregulated in HepG2 cells | J Med Chem 39: 3343-56 (1996) Article DOI: 10.1021/jm960153q BindingDB Entry DOI: 10.7270/Q2FT8K4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Low-density lipoprotein receptor (Homo sapiens (Human)) | BDBM50052684 (CHEMBL112106 | N-[5-(3-Cyclohexyl-propionylamino)-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 7.60E+3 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Concentration at which one-half of the maximum Low density lipoprotein receptor is upregulated in HepG2 cells | J Med Chem 39: 3343-56 (1996) Article DOI: 10.1021/jm960153q BindingDB Entry DOI: 10.7270/Q2FT8K4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Low-density lipoprotein receptor (Homo sapiens (Human)) | BDBM50052685 (4-Amino-N-[5-(3-cyclohexyl-propionylamino)-2-methy...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.80E+3 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Concentration at which one-half of the maximum Low density lipoprotein receptor is upregulated in HepG2 cells | J Med Chem 39: 3343-56 (1996) Article DOI: 10.1021/jm960153q BindingDB Entry DOI: 10.7270/Q2FT8K4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Low-density lipoprotein receptor (Homo sapiens (Human)) | BDBM50052680 (CHEMBL419763 | N-[5-(3-Cyclohexyl-propionylamino)-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.70E+3 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Concentration at which one-half of the maximum Low density lipoprotein receptor is upregulated in HepG2 cells | J Med Chem 39: 3343-56 (1996) Article DOI: 10.1021/jm960153q BindingDB Entry DOI: 10.7270/Q2FT8K4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Low-density lipoprotein receptor (Homo sapiens (Human)) | BDBM50052683 (CHEMBL112449 | N-[3-((Z)-2-Cyano-2-pyridin-3-yl-vi...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Concentration at which one-half of the maximum Low density lipoprotein receptor is upregulated in HepG2 cells | J Med Chem 39: 3343-56 (1996) Article DOI: 10.1021/jm960153q BindingDB Entry DOI: 10.7270/Q2FT8K4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Low-density lipoprotein receptor (Homo sapiens (Human)) | BDBM50052682 (3-Cyclohexyl-N-[3-(5-hydroxy-1H-benzoimidazol-2-yl...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 700 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Concentration at which one-half of the maximum Low density lipoprotein receptor is upregulated in HepG2 cells | J Med Chem 39: 3343-56 (1996) Article DOI: 10.1021/jm960153q BindingDB Entry DOI: 10.7270/Q2FT8K4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Low-density lipoprotein receptor (Homo sapiens (Human)) | BDBM50052681 (CHEMBL114890 | N-[3-((Z)-2-Benzo[1,3]dioxol-5-yl-2...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 700 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Concentration at which one-half of the maximum Low density lipoprotein receptor is upregulated in HepG2 cells | J Med Chem 39: 3343-56 (1996) Article DOI: 10.1021/jm960153q BindingDB Entry DOI: 10.7270/Q2FT8K4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Low-density lipoprotein receptor (Homo sapiens (Human)) | BDBM50052679 (CHEMBL112537 | N-[5-(3-Cyclohexyl-propionylamino)-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Concentration at which one-half of the maximum Low density lipoprotein receptor is upregulated in HepG2 cells | J Med Chem 39: 3343-56 (1996) Article DOI: 10.1021/jm960153q BindingDB Entry DOI: 10.7270/Q2FT8K4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Low-density lipoprotein receptor (Homo sapiens (Human)) | BDBM50052678 (3-Cyclohexyl-N-[4-methyl-3-(5-methyl-1H-benzoimida...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.30E+3 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Concentration at which one-half of the maximum Low density lipoprotein receptor is upregulated in HepG2 cells | J Med Chem 39: 3343-56 (1996) Article DOI: 10.1021/jm960153q BindingDB Entry DOI: 10.7270/Q2FT8K4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Low-density lipoprotein receptor (Homo sapiens (Human)) | BDBM50052676 (CHEMBL115304 | N-[3-(1H-Benzoimidazol-2-yl)-4-meth...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.30E+3 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Concentration at which one-half of the maximum Low density lipoprotein receptor is upregulated in HepG2 cells | J Med Chem 39: 3343-56 (1996) Article DOI: 10.1021/jm960153q BindingDB Entry DOI: 10.7270/Q2FT8K4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Low-density lipoprotein receptor (Homo sapiens (Human)) | BDBM50052677 (CHEMBL115779 | N-(2-Cyclohexyl-ethyl)-3-(4-hydroxy...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Concentration at which one-half of the maximum Low density lipoprotein receptor is upregulated in HepG2 cells | J Med Chem 39: 3343-56 (1996) Article DOI: 10.1021/jm960153q BindingDB Entry DOI: 10.7270/Q2FT8K4S | |||||||||||
More data for this Ligand-Target Pair |