Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Ovarian cancer G-protein coupled receptor 1 (Homo sapiens (Human)) | BDBM50175290 (CHEMBL3810385) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | 7.2 | n/a |
Hokkaido University Curated by ChEMBL | Assay Description Antagonist activity at N-terminal HA-tagged OGR1 (unknown origin) expressed in HEK293 cells assessed as inhibition of pH dependent nuclear factor of ... | ACS Med Chem Lett 7: 493-7 (2016) Article DOI: 10.1021/acsmedchemlett.6b00014 BindingDB Entry DOI: 10.7270/Q2833TZR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ovarian cancer G-protein coupled receptor 1 (Homo sapiens (Human)) | BDBM123510 (US8748435, 35) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institutes for BioMedical Research Curated by ChEMBL | Assay Description Inhibition of OGR1 (unknown origin) expressed in human HeLa cells assessed as reduction in cAMP accumulation | J Med Chem 60: 3672-3683 (2017) Article DOI: 10.1021/acs.jmedchem.6b01703 BindingDB Entry DOI: 10.7270/Q28P6349 | |||||||||||
More data for this Ligand-Target Pair |