Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Dolichyl-diphosphooligosaccharide--protein glycosyltransferase subunit 1 (Saccharomyces cerevisiae (Baker's yeast)) | BDBM43866 (2-amino-4,6-dimethyl-3-oxo-1-N,9-N-bis[(3R,6S,7R,1...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase DrugBank KEGG PC cid PC sid UniChem Similars | Article PubMed | 41 | -38.6 | n/a | n/a | n/a | n/a | n/a | 7.5 | 0 |
Massachusetts Institute of Technology | Assay Description Competition assay using S. cerevisiae oligosaccharyl transferase (OT)with disaccharide donor Dol-P-P-(GlcNAc)2 and the tripeptide substrate Bz-Asn-Le... | Chem Biol 9: 1323-8 (2002) Article DOI: 10.1016/S1074-5521(02)00281-8 BindingDB Entry DOI: 10.7270/Q2736P9D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dolichyl-diphosphooligosaccharide--protein glycosyltransferase subunit 1 (Saccharomyces cerevisiae (Baker's yeast)) | BDBM43865 (6-formyl-4,7-dihydroxy-9-keto-5H-phenazine-1-carbo...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 62 | -37.7 | n/a | n/a | n/a | n/a | n/a | 7.5 | 0 |
Massachusetts Institute of Technology | Assay Description Competition assay using S. cerevisiae oligosaccharyl transferase (OT)with disaccharide donor Dol-P-P-(GlcNAc)2 and the tripeptide substrate Bz-Asn-Le... | Chem Biol 9: 1323-8 (2002) Article DOI: 10.1016/S1074-5521(02)00281-8 BindingDB Entry DOI: 10.7270/Q2736P9D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dolichyl-diphosphooligosaccharide--protein glycosyltransferase subunit 1 (Saccharomyces cerevisiae (Baker's yeast)) | BDBM43863 (3-[[4-amino-6-(2,5-dimethoxyanilino)-5-nitro-pyrim...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | Article PubMed | 1.10E+3 | -31.2 | n/a | n/a | n/a | n/a | n/a | 7.5 | 0 |
Massachusetts Institute of Technology | Assay Description Competition assay using S. cerevisiae oligosaccharyl transferase (OT)with disaccharide donor Dol-P-P-(GlcNAc)2 and the tripeptide substrate Bz-Asn-Le... | Chem Biol 9: 1323-8 (2002) Article DOI: 10.1016/S1074-5521(02)00281-8 BindingDB Entry DOI: 10.7270/Q2736P9D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dolichyl-diphosphooligosaccharide--protein glycosyltransferase subunit 1 (Saccharomyces cerevisiae (Baker's yeast)) | BDBM43860 (Glycopeptide, 2 | MLS000517385 | N-(4-acetamidophe...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | Article PubMed | 2.50E+3 | -29.3 | n/a | n/a | n/a | n/a | n/a | 7.5 | 0 |
Massachusetts Institute of Technology | Assay Description Competition assay using S. cerevisiae oligosaccharyl transferase (OT)with disaccharide donor Dol-P-P-(GlcNAc)2 and the tripeptide substrate Bz-Asn-Le... | Chem Biol 9: 1323-8 (2002) Article DOI: 10.1016/S1074-5521(02)00281-8 BindingDB Entry DOI: 10.7270/Q2736P9D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dolichyl-diphosphooligosaccharide--protein glycosyltransferase subunit 1 (Saccharomyces cerevisiae (Baker's yeast)) | BDBM43864 (2-chloranyl-N1,N4-bis[4-(4,5-dihydro-1H-imidazol-2...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | 4.00E+3 | -28.2 | n/a | n/a | n/a | n/a | n/a | 7.5 | 0 |
Massachusetts Institute of Technology | Assay Description Competition assay using S. cerevisiae oligosaccharyl transferase (OT)with disaccharide donor Dol-P-P-(GlcNAc)2 and the tripeptide substrate Bz-Asn-Le... | Chem Biol 9: 1323-8 (2002) Article DOI: 10.1016/S1074-5521(02)00281-8 BindingDB Entry DOI: 10.7270/Q2736P9D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dolichyl-diphosphooligosaccharide--protein glycosyltransferase subunit 1 (Saccharomyces cerevisiae (Baker's yeast)) | BDBM43861 (4-[7-[4-[diethyl(methyl)ammonio]butoxy]-9-keto-flu...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 4.50E+3 | -28.0 | n/a | n/a | n/a | n/a | n/a | 7.5 | 0 |
Massachusetts Institute of Technology | Assay Description Competition assay using S. cerevisiae oligosaccharyl transferase (OT)with disaccharide donor Dol-P-P-(GlcNAc)2 and the tripeptide substrate Bz-Asn-Le... | Chem Biol 9: 1323-8 (2002) Article DOI: 10.1016/S1074-5521(02)00281-8 BindingDB Entry DOI: 10.7270/Q2736P9D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dolichyl-diphosphooligosaccharide--protein glycosyltransferase subunit 1 (Saccharomyces cerevisiae (Baker's yeast)) | BDBM43862 (2-(aminocarbonylamino)-N-[4-[(4-methoxyphenyl)sulf...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | Article PubMed | 3.40E+4 | -23.4 | n/a | n/a | n/a | n/a | n/a | 7.5 | 0 |
Massachusetts Institute of Technology | Assay Description Competition assay using S. cerevisiae oligosaccharyl transferase (OT)with disaccharide donor Dol-P-P-(GlcNAc)2 and the tripeptide substrate Bz-Asn-Le... | Chem Biol 9: 1323-8 (2002) Article DOI: 10.1016/S1074-5521(02)00281-8 BindingDB Entry DOI: 10.7270/Q2736P9D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dolichyl-diphosphooligosaccharide--protein glycosyltransferase subunit 1 (Saccharomyces cerevisiae (Baker's yeast)) | BDBM43859 (2-[[4-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfany...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | Article PubMed | 1.00E+5 | -20.9 | n/a | n/a | n/a | n/a | n/a | 7.5 | 0 |
Massachusetts Institute of Technology | Assay Description Competition assay using S. cerevisiae oligosaccharyl transferase (OT)with disaccharide donor Dol-P-P-(GlcNAc)2 and the tripeptide substrate Bz-Asn-Le... | Chem Biol 9: 1323-8 (2002) Article DOI: 10.1016/S1074-5521(02)00281-8 BindingDB Entry DOI: 10.7270/Q2736P9D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dolichyl-diphosphooligosaccharide--protein glycosyltransferase subunit 1 (Saccharomyces cerevisiae (Baker's yeast)) | BDBM43867 (Glycopeptide, 1) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | n/a | n/a | n/a | 7.5 | 0 |
Massachusetts Institute of Technology | Assay Description Competition assay using S. cerevisiae oligosaccharyl transferase (OT)with disaccharide donor Dol-P-P-(GlcNAc)2 and the tripeptide substrate Bz-Asn-Le... | Chem Biol 9: 1323-8 (2002) Article DOI: 10.1016/S1074-5521(02)00281-8 BindingDB Entry DOI: 10.7270/Q2736P9D | |||||||||||
More data for this Ligand-Target Pair |