BindingDB PrimarySearch

Found 9 hits Enz. Inhib. hit(s) with Target = 'Dolichyl-diphosphooligosaccharide--protein glycosyltransferase subunit 1'
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Dolichyl-diphosphooligosaccharide--protein glycosyltransferase subunit 1 (Saccharomyces cerevisiae (Baker's yeast))	BDBM43866 (2-amino-4,6-dimethyl-3-oxo-1-N,9-N-bis[(3R,6S,7R,1...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	Purchase DrugBank KEGG PC cid PC sid UniChem Similars	Article PubMed	41	-38.6	n/a	n/a	n/a	n/a	n/a	7.5	0
Massachusetts Institute of Technology					Assay Description Competition assay using S. cerevisiae oligosaccharyl transferase (OT)with disaccharide donor Dol-P-P-(GlcNAc)2 and the tripeptide substrate Bz-Asn-Le...				Chem Biol 9: 1323-8 (2002) Article DOI: 10.1016/S1074-5521(02)00281-8 BindingDB Entry DOI: 10.7270/Q2736P9D
Massachusetts Institute of Technology					More data for this Ligand-Target Pair
Dolichyl-diphosphooligosaccharide--protein glycosyltransferase subunit 1 (Saccharomyces cerevisiae (Baker's yeast))	BDBM43865 (6-formyl-4,7-dihydroxy-9-keto-5H-phenazine-1-carbo...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	62	-37.7	n/a	n/a	n/a	n/a	n/a	7.5	0
Massachusetts Institute of Technology					Assay Description Competition assay using S. cerevisiae oligosaccharyl transferase (OT)with disaccharide donor Dol-P-P-(GlcNAc)2 and the tripeptide substrate Bz-Asn-Le...				Chem Biol 9: 1323-8 (2002) Article DOI: 10.1016/S1074-5521(02)00281-8 BindingDB Entry DOI: 10.7270/Q2736P9D
Massachusetts Institute of Technology					More data for this Ligand-Target Pair
Dolichyl-diphosphooligosaccharide--protein glycosyltransferase subunit 1 (Saccharomyces cerevisiae (Baker's yeast))	BDBM43863 (3-[[4-amino-6-(2,5-dimethoxyanilino)-5-nitro-pyrim...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	Purchase PC cid PC sid UniChem Similars	Article PubMed	1.10E+3	-31.2	n/a	n/a	n/a	n/a	n/a	7.5	0
Massachusetts Institute of Technology					Assay Description Competition assay using S. cerevisiae oligosaccharyl transferase (OT)with disaccharide donor Dol-P-P-(GlcNAc)2 and the tripeptide substrate Bz-Asn-Le...				Chem Biol 9: 1323-8 (2002) Article DOI: 10.1016/S1074-5521(02)00281-8 BindingDB Entry DOI: 10.7270/Q2736P9D
Massachusetts Institute of Technology					More data for this Ligand-Target Pair
Dolichyl-diphosphooligosaccharide--protein glycosyltransferase subunit 1 (Saccharomyces cerevisiae (Baker's yeast))	BDBM43860 (Glycopeptide, 2 \| MLS000517385 \| N-(4-acetamidophe...) Show SMILES CC(=O)Nc1ccc(NC(=O)c2ccc(Cl)nc2)cc1 Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	Purchase PC cid PC sid UniChem Similars	Article PubMed	2.50E+3	-29.3	n/a	n/a	n/a	n/a	n/a	7.5	0
Massachusetts Institute of Technology					Assay Description Competition assay using S. cerevisiae oligosaccharyl transferase (OT)with disaccharide donor Dol-P-P-(GlcNAc)2 and the tripeptide substrate Bz-Asn-Le...				Chem Biol 9: 1323-8 (2002) Article DOI: 10.1016/S1074-5521(02)00281-8 BindingDB Entry DOI: 10.7270/Q2736P9D
Massachusetts Institute of Technology					More data for this Ligand-Target Pair
Dolichyl-diphosphooligosaccharide--protein glycosyltransferase subunit 1 (Saccharomyces cerevisiae (Baker's yeast))	BDBM43864 (2-chloranyl-N1,N4-bis[4-(4,5-dihydro-1H-imidazol-2...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	Purchase MCE PC cid PC sid UniChem Similars	Article PubMed	4.00E+3	-28.2	n/a	n/a	n/a	n/a	n/a	7.5	0
Massachusetts Institute of Technology					Assay Description Competition assay using S. cerevisiae oligosaccharyl transferase (OT)with disaccharide donor Dol-P-P-(GlcNAc)2 and the tripeptide substrate Bz-Asn-Le...				Chem Biol 9: 1323-8 (2002) Article DOI: 10.1016/S1074-5521(02)00281-8 BindingDB Entry DOI: 10.7270/Q2736P9D
Massachusetts Institute of Technology					More data for this Ligand-Target Pair
Dolichyl-diphosphooligosaccharide--protein glycosyltransferase subunit 1 (Saccharomyces cerevisiae (Baker's yeast))	BDBM43861 (4-[7-[4-[diethyl(methyl)ammonio]butoxy]-9-keto-flu...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	4.50E+3	-28.0	n/a	n/a	n/a	n/a	n/a	7.5	0
Massachusetts Institute of Technology					Assay Description Competition assay using S. cerevisiae oligosaccharyl transferase (OT)with disaccharide donor Dol-P-P-(GlcNAc)2 and the tripeptide substrate Bz-Asn-Le...				Chem Biol 9: 1323-8 (2002) Article DOI: 10.1016/S1074-5521(02)00281-8 BindingDB Entry DOI: 10.7270/Q2736P9D
Massachusetts Institute of Technology					More data for this Ligand-Target Pair
Dolichyl-diphosphooligosaccharide--protein glycosyltransferase subunit 1 (Saccharomyces cerevisiae (Baker's yeast))	BDBM43862 (2-(aminocarbonylamino)-N-[4-[(4-methoxyphenyl)sulf...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	Purchase PC cid PC sid UniChem Similars	Article PubMed	3.40E+4	-23.4	n/a	n/a	n/a	n/a	n/a	7.5	0
Massachusetts Institute of Technology					Assay Description Competition assay using S. cerevisiae oligosaccharyl transferase (OT)with disaccharide donor Dol-P-P-(GlcNAc)2 and the tripeptide substrate Bz-Asn-Le...				Chem Biol 9: 1323-8 (2002) Article DOI: 10.1016/S1074-5521(02)00281-8 BindingDB Entry DOI: 10.7270/Q2736P9D
Massachusetts Institute of Technology					More data for this Ligand-Target Pair
Dolichyl-diphosphooligosaccharide--protein glycosyltransferase subunit 1 (Saccharomyces cerevisiae (Baker's yeast))	BDBM43859 (2-[[4-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfany...) Show SMILES COc1ccc(cc1)-n1cnnc1SCC(=O)Nc1cc(C)on1 Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	Purchase PC cid PC sid UniChem Similars	Article PubMed	1.00E+5	-20.9	n/a	n/a	n/a	n/a	n/a	7.5	0
Massachusetts Institute of Technology					Assay Description Competition assay using S. cerevisiae oligosaccharyl transferase (OT)with disaccharide donor Dol-P-P-(GlcNAc)2 and the tripeptide substrate Bz-Asn-Le...				Chem Biol 9: 1323-8 (2002) Article DOI: 10.1016/S1074-5521(02)00281-8 BindingDB Entry DOI: 10.7270/Q2736P9D
Massachusetts Institute of Technology					More data for this Ligand-Target Pair
Dolichyl-diphosphooligosaccharide--protein glycosyltransferase subunit 1 (Saccharomyces cerevisiae (Baker's yeast))	BDBM43867 (Glycopeptide, 1) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	KEGG PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	n/a	n/a	n/a	7.5	0
Massachusetts Institute of Technology					Assay Description Competition assay using S. cerevisiae oligosaccharyl transferase (OT)with disaccharide donor Dol-P-P-(GlcNAc)2 and the tripeptide substrate Bz-Asn-Le...				Chem Biol 9: 1323-8 (2002) Article DOI: 10.1016/S1074-5521(02)00281-8 BindingDB Entry DOI: 10.7270/Q2736P9D
Massachusetts Institute of Technology					More data for this Ligand-Target Pair