Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM86478 (A-317491) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem Patents Similars | PDB Article PubMed | 9 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Plc Curated by ChEMBL | Assay Description Antagonist activity at human P2X2/3 expressed in human1321N1 cells assessed as inhibition of alpha,beta-methylene-ATP-stimulated Ca2+ influx preincub... | Bioorg Med Chem Lett 26: 3896-904 (2016) Article DOI: 10.1016/j.bmcl.2016.07.009 BindingDB Entry DOI: 10.7270/Q26W9FJD | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM86478 (A-317491) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem Patents Similars | PDB Article PubMed | 9 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Plc Curated by ChEMBL | Assay Description Antagonist activity at human P2X2/3 expressed in human1321N1 cells assessed as inhibition of alpha,beta-methylene-ATP-stimulated Ca2+ influx preincub... | Bioorg Med Chem Lett 26: 3896-904 (2016) Article DOI: 10.1016/j.bmcl.2016.07.009 BindingDB Entry DOI: 10.7270/Q26W9FJD | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM86480 (A-317344) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | Article PubMed | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Plc Curated by ChEMBL | Assay Description Antagonist activity at human P2X2/3 expressed in human1321N1 cells assessed as inhibition of alpha,beta-methylene-ATP-stimulated Ca2+ influx preincub... | Bioorg Med Chem Lett 26: 3896-904 (2016) Article DOI: 10.1016/j.bmcl.2016.07.009 BindingDB Entry DOI: 10.7270/Q26W9FJD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM86480 (A-317344) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | Article PubMed | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Gedeon Richter Plc Curated by ChEMBL | Assay Description Antagonist activity at human P2X2/3 expressed in human1321N1 cells assessed as inhibition of alpha,beta-methylene-ATP-stimulated Ca2+ influx preincub... | Bioorg Med Chem Lett 26: 3896-904 (2016) Article DOI: 10.1016/j.bmcl.2016.07.009 BindingDB Entry DOI: 10.7270/Q26W9FJD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM50594498 (CHEMBL4583478) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 8.30 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Citation and Details Article DOI: 10.1021/acs.jmedchem.2c00812 BindingDB Entry DOI: 10.7270/Q2XS60DK | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM320093 (3-(5-ethyl-1,3- thiazol-2-yl)-5- [(3R)- tetrahydro...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 14 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FLEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelati... | US Patent US10202369 (2019) BindingDB Entry DOI: 10.7270/Q2TT4T2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM319936 (3-[(2- Methylpyridin- 4-yl)oxy]-5- (5-methyl- 1,3-...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 14 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FILEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelat... | US Patent US10472354 (2019) BindingDB Entry DOI: 10.7270/Q2KD2197 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM320093 (3-(5-ethyl-1,3- thiazol-2-yl)-5- [(3R)- tetrahydro...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 14 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FILEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelat... | US Patent US10472354 (2019) BindingDB Entry DOI: 10.7270/Q2KD2197 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM319936 (3-[(2- Methylpyridin- 4-yl)oxy]-5- (5-methyl- 1,3-...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 14 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FLEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelati... | US Patent US10202369 (2019) BindingDB Entry DOI: 10.7270/Q2TT4T2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM319933 (N-[(1R)-1-(6- Methyl- pyridazin-3- yl)ethyl]-3- [(...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 16 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FILEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelat... | US Patent US10472354 (2019) BindingDB Entry DOI: 10.7270/Q2KD2197 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM319933 (N-[(1R)-1-(6- Methyl- pyridazin-3- yl)ethyl]-3- [(...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 16 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FLEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelati... | US Patent US10202369 (2019) BindingDB Entry DOI: 10.7270/Q2TT4T2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM319940 (N-[(1R)-1-(6- Methylpyridin- 3-yl)ethyl]- 3-[(2- m...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 17 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FILEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelat... | US Patent US10472354 (2019) BindingDB Entry DOI: 10.7270/Q2KD2197 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM319940 (N-[(1R)-1-(6- Methylpyridin- 3-yl)ethyl]- 3-[(2- m...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 17 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FLEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelati... | US Patent US10202369 (2019) BindingDB Entry DOI: 10.7270/Q2TT4T2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM319931 (3-(5-Methyl- 1,3-thiazol-2- yl)-5- (tetrahydro- 2H...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 19 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FLEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelati... | US Patent US10202369 (2019) BindingDB Entry DOI: 10.7270/Q2TT4T2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM319931 (3-(5-Methyl- 1,3-thiazol-2- yl)-5- (tetrahydro- 2H...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 19 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FILEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelat... | US Patent US10472354 (2019) BindingDB Entry DOI: 10.7270/Q2KD2197 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM320075 (3-(5-ethyl-1,3- thiazol-2-yl)-5- [(3R)- tetrahydro...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 22 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FILEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelat... | US Patent US10472354 (2019) BindingDB Entry DOI: 10.7270/Q2KD2197 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM320075 (3-(5-ethyl-1,3- thiazol-2-yl)-5- [(3R)- tetrahydro...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 22 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FLEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelati... | US Patent US10202369 (2019) BindingDB Entry DOI: 10.7270/Q2TT4T2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM320111 (3-(5-ethyl-1,3- thiazol-2-yl)-5- [(3S)- tetrahydro...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 23 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FILEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelat... | US Patent US10472354 (2019) BindingDB Entry DOI: 10.7270/Q2KD2197 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM320102 (3-(5-ethyl-1,3- thiazol-2-yl)-5- [(2R)- tetrahydro...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 23 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FLEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelati... | US Patent US10202369 (2019) BindingDB Entry DOI: 10.7270/Q2TT4T2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM320137 (3-{[1-(2,2- difluoroethyl) piperidin-4-yl]oxy}- 5-...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 27 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FLEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelati... | US Patent US10202369 (2019) BindingDB Entry DOI: 10.7270/Q2TT4T2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM319958 (3-(5-Ethyl-1,3-thiazol-2-yl)-N-[(1R)-1-(2-methylpy...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 27 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FLEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelati... | US Patent US10202369 (2019) BindingDB Entry DOI: 10.7270/Q2TT4T2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM319958 (3-(5-Ethyl-1,3-thiazol-2-yl)-N-[(1R)-1-(2-methylpy...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 27 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FILEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelat... | US Patent US10472354 (2019) BindingDB Entry DOI: 10.7270/Q2KD2197 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM320137 (3-{[1-(2,2- difluoroethyl) piperidin-4-yl]oxy}- 5-...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 27 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FILEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelat... | US Patent US10472354 (2019) BindingDB Entry DOI: 10.7270/Q2KD2197 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM319932 (N-[(1R)-1-(6- Methyl- pyridazin-3- yl)ethyl]-3- (5...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 27 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FILEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelat... | US Patent US10472354 (2019) BindingDB Entry DOI: 10.7270/Q2KD2197 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM319932 (N-[(1R)-1-(6- Methyl- pyridazin-3- yl)ethyl]-3- (5...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 27 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FLEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelati... | US Patent US10202369 (2019) BindingDB Entry DOI: 10.7270/Q2TT4T2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM322574 (US10183937, Example 385 | US10202369, Example 385) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 28 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FLEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelati... | US Patent US10202369 (2019) BindingDB Entry DOI: 10.7270/Q2TT4T2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM320217 (3-{[4,4-difluoro-1-methylpiperidin-3-yl]methoxy}-5...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 28 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FILEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelat... | US Patent US10472354 (2019) BindingDB Entry DOI: 10.7270/Q2KD2197 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM319962 (3-(5-Ethyl-1,3-thiazol-2-yl)-5-(tetrahydro-2H-pyra...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 33 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FILEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelat... | US Patent US10472354 (2019) BindingDB Entry DOI: 10.7270/Q2KD2197 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM319962 (3-(5-Ethyl-1,3-thiazol-2-yl)-5-(tetrahydro-2H-pyra...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 33 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FLEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelati... | US Patent US10202369 (2019) BindingDB Entry DOI: 10.7270/Q2TT4T2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM319914 (N-[1-(5- Chloro-3- fluoropyridin- 2-yl)ethyl]-3- (...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 34 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FLEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelati... | US Patent US10202369 (2019) BindingDB Entry DOI: 10.7270/Q2TT4T2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM319914 (N-[1-(5- Chloro-3- fluoropyridin- 2-yl)ethyl]-3- (...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 34 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FILEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelat... | US Patent US10472354 (2019) BindingDB Entry DOI: 10.7270/Q2KD2197 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM320144 (N-[(1R)-1-(6- methylpyridazin-3- yl)ethyl]-3-(5- m...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 35 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FLEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelati... | US Patent US10202369 (2019) BindingDB Entry DOI: 10.7270/Q2TT4T2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM320216 (3-{[4,4- difluoro-1- methylpiperidin- 3-yl]methoxy...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 35 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FILEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelat... | US Patent US10472354 (2019) BindingDB Entry DOI: 10.7270/Q2KD2197 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM320073 (3-(5-ethyl-1,3- thiazol-2-yl)-N- [(1R)-1-(6- methy...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 35 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FLEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelati... | US Patent US10202369 (2019) BindingDB Entry DOI: 10.7270/Q2TT4T2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM320111 (3-(5-ethyl-1,3- thiazol-2-yl)-5- [(3S)- tetrahydro...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 35 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FILEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelat... | US Patent US10472354 (2019) BindingDB Entry DOI: 10.7270/Q2KD2197 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM320102 (3-(5-ethyl-1,3- thiazol-2-yl)-5- [(2R)- tetrahydro...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 35 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FLEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelati... | US Patent US10202369 (2019) BindingDB Entry DOI: 10.7270/Q2TT4T2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM320144 (N-[(1R)-1-(6- methylpyridazin-3- yl)ethyl]-3-(5- m...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 35 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FILEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelat... | US Patent US10472354 (2019) BindingDB Entry DOI: 10.7270/Q2KD2197 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM320073 (3-(5-ethyl-1,3- thiazol-2-yl)-N- [(1R)-1-(6- methy...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 35 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FILEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelat... | US Patent US10472354 (2019) BindingDB Entry DOI: 10.7270/Q2KD2197 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM320216 (3-{[4,4- difluoro-1- methylpiperidin- 3-yl]methoxy...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 35 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FLEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelati... | US Patent US10202369 (2019) BindingDB Entry DOI: 10.7270/Q2TT4T2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM319918 (3-(5-Methyl- 1,3-thiazol-2- yl)-5- (tetrahydro- 2H...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 36 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FLEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelati... | US Patent US10202369 (2019) BindingDB Entry DOI: 10.7270/Q2TT4T2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM319918 (3-(5-Methyl- 1,3-thiazol-2- yl)-5- (tetrahydro- 2H...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 36 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FILEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelat... | US Patent US10472354 (2019) BindingDB Entry DOI: 10.7270/Q2KD2197 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM320084 (3-(5-ethyl-1,3- thiazol-2-yl)-5- [(3S)- tetrahydro...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 38 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FLEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelati... | US Patent US10202369 (2019) BindingDB Entry DOI: 10.7270/Q2TT4T2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM320091 (3-(5-ethyl-1,3- thiazol-2-yl)-N- [(1R)-1-(6- methy...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 38 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FLEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelati... | US Patent US10202369 (2019) BindingDB Entry DOI: 10.7270/Q2TT4T2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM319839 (N-[1-(5-Chloro-3-fluoropyridin-2-yl)ethyl]-3-(cycl...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 38 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FLEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelati... | US Patent US10202369 (2019) BindingDB Entry DOI: 10.7270/Q2TT4T2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM319839 (N-[1-(5-Chloro-3-fluoropyridin-2-yl)ethyl]-3-(cycl...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 38 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FILEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelat... | US Patent US10472354 (2019) BindingDB Entry DOI: 10.7270/Q2KD2197 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM320136 (3-(5-methyl-1,3- thiazol-2-yl)-5-{[1- (2,2,2- trif...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 38 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FILEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelat... | US Patent US10472354 (2019) BindingDB Entry DOI: 10.7270/Q2KD2197 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM320084 (3-(5-ethyl-1,3- thiazol-2-yl)-5- [(3S)- tetrahydro...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 38 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FILEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelat... | US Patent US10472354 (2019) BindingDB Entry DOI: 10.7270/Q2KD2197 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM320091 (3-(5-ethyl-1,3- thiazol-2-yl)-N- [(1R)-1-(6- methy...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 38 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FILEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelat... | US Patent US10472354 (2019) BindingDB Entry DOI: 10.7270/Q2KD2197 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM320136 (3-(5-methyl-1,3- thiazol-2-yl)-5-{[1- (2,2,2- trif...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 38 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FLEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelati... | US Patent US10202369 (2019) BindingDB Entry DOI: 10.7270/Q2TT4T2P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2X purinoceptor 2/3 (Homo sapiens (Human)) | BDBM319938 (3-[(2- Methylpyridin- 4-yl)oxy]-5- (5-methyl- 1,3-...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 39 | n/a | n/a | n/a | n/a | n/a | n/a |
Bayer Aktiengesellschaft US Patent | Assay Description A fluorescent imaging plate reader (FILEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelat... | US Patent US10472354 (2019) BindingDB Entry DOI: 10.7270/Q2KD2197 | |||||||||||
More data for this Ligand-Target Pair |
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