Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552303 (US11312727, Compound 123A) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.400 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552356 ((17a*R,*E)-24,25-difluoro-12-hydroxy-2,6,9,17a-tet...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552337 (US11312727, Compound 136A) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552377 (US11312727, Compound 152BA) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.20 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552440 (US11312727, Compound 175A) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.90 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552297 ((18*R,*Z)-4-fluoro-12-hydroxy-18-(2-(methylthio)ph...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552278 ((17a′*R,*E)-24′,25′-difluoro-12&...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552406 ((9*R,17a*R,*E)-24,25-difluoro-12-hydroxy-9-methyl-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552314 ((13*S,21a*R,Z)-13-ethyl-24,25-difluoro-16-hydroxy-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2.40 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552388 (US11312727, Compound 155A) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2.80 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552350 (US11312727, Compound 140B) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552344 (US11312727, Compound 138D) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552336 (US11312727, Compound 108D) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552147 (US11312727, Compound 46B) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552255 (US11312727, Compound 100AA) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552412 (US11312727, Compound 165A) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552313 (US11312727, Compound 126BA) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3.40 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552439 ((18′*R,*E)-3′,4′-difluoro-12R...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3.80 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552291 (US11312727, Compound 116A) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552341 (US11312727, Compound 138AA) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552287 (US11312727, Compound 114A) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552381 (US11312727, Compound 153BB) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552261 (US11312727, Compound 102A) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552292 (US11312727, Compound 117A) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552385 (US11312727, Compound 154BB) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 4.20 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552404 (US11312727, Compound 162B) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 4.30 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552369 (US11312727, Compound 148AA) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 4.60 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552378 (US11312727, Compound 152BB) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 4.80 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552259 (US11312727, Compound 101AA) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552444 ((3*R,17a′*R,*E)-24′,25′-difluoro...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 5.10 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552421 ((21a′*R,*E)-24′,25′-difluoro-16&...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 5.20 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552446 (US11312727, Compound 177AB) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 5.20 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552416 (US11312727, Compound 167AA) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 5.30 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552423 (US11312727, Compound 169BB) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 5.40 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552316 ((1a*S,11b*S,20a*S)-22,23-difluoro-17-hydroxy-1a,2,...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552324 (US11312727, Compound 131AB) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552418 (US11312727, Compound 167AB) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552276 ((17a′*R,*E)-12′-hydroxy-2′,17a...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552267 (US11312727, Compound 101AB) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552230 ((23b*R, Z)-16,17-difluoro-6-hydroxy-10,13,18,23b-t...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552225 (US11312727, Compound 88B) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552353 (US11312727, Compound 141AB) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552164 ((*Z)-4-hydroxy-15-phenyl-8,15-dihydro-7H-6,16-meth...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552195 ((18*R,Z)-3,4-difluoro-12-hydroxy-18-phenyl-6,9-dih...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552370 (US11312727, Compound 148BB) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 6.20 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552365 (US11312727, Compound 146A) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 6.30 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552443 (US11312727, Compound 176BA) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 6.5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552427 (US11312727, Compound 170BB) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 6.60 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552437 ((9*S,18*S,*E)-4-chloro-9-ethyl-3-fluoro-12-hydroxy...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 6.70 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polymerase basic protein 2 (Influenza A virus (strain A/WS/1933 H1N1)) | BDBM552363 (US11312727, Compound 145A) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 6.70 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description EN PA FRET inhibition assay was performed using a 19 nucleotide synthetic oligoribonucleotide substrate: 5′-FAM-AUUUUGUUUUUAAUAUUUC-BHQ-3′... | Citation and Details BindingDB Entry DOI: 10.7270/Q2P272BG | |||||||||||
More data for this Ligand-Target Pair |
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