Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Vesicular glutamate transporter 3 (Rattus norvegicus) | BDBM50366944 (Azovan Blue | Azovan sodium | EVANS BLUE) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | PubMed | 40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Montana Curated by ChEMBL | Assay Description Evaluated for competitive inhibition against Vesicular glutamate transporter (VGLUT), and Ki value was reported. | J Med Chem 45: 2260-76 (2002) BindingDB Entry DOI: 10.7270/Q2NK3FRR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vesicular glutamate transporter 3 (Rattus norvegicus) | BDBM50113317 (Bis[4-Amino-5-hydroxy-6-(2-methoxy-phenylazo)-naph...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | PubMed | 190 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Montana Curated by ChEMBL | Assay Description Evaluated for competitive inhibition against Vesicular glutamate transporter (VGLUT), and Ki value was reported. | J Med Chem 45: 2260-76 (2002) BindingDB Entry DOI: 10.7270/Q2NK3FRR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vesicular glutamate transporter 3 (Rattus norvegicus) | BDBM50089912 ((2S)-2-amino-4-methylidenepentanedioic acid | 4-me...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL KEGG PC cid PC sid UniChem Patents Similars | PubMed | 3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Montana Curated by ChEMBL | Assay Description Evaluated for competitive inhibition against Vesicular glutamate transporter (VGLUT), and Ki value was reported. | J Med Chem 45: 2260-76 (2002) BindingDB Entry DOI: 10.7270/Q2NK3FRR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vesicular glutamate transporter 3 (Rattus norvegicus) | BDBM50113314 (6-Biphenyl-4-yl-quinoline-2,4-dicarboxylic acid | ...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 4.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Montana Curated by ChEMBL | Assay Description Estimated inhibitory conc. against Vesicular glutamate transporter (VGLUT), using Cheng-Prushoff equation | J Med Chem 45: 2260-76 (2002) BindingDB Entry DOI: 10.7270/Q2NK3FRR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vesicular glutamate transporter 3 (Rattus norvegicus) | BDBM50113320 (6-(2-Biphenyl-4-yl-vinyl)-quinoline-2,4-dicarboxyl...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 6.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Montana Curated by ChEMBL | Assay Description Estimated inhibitory conc. against Vesicular glutamate transporter (VGLUT), using Cheng-Prushoff equation | J Med Chem 45: 2260-76 (2002) BindingDB Entry DOI: 10.7270/Q2NK3FRR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vesicular glutamate transporter 3 (Rattus norvegicus) | BDBM50113314 (6-Biphenyl-4-yl-quinoline-2,4-dicarboxylic acid | ...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 9.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Montana Curated by ChEMBL | Assay Description Inhibitory conc. against Vesicular glutamate transporter (VGLUT), derived from Lineweaver-Burke analysis | J Med Chem 45: 2260-76 (2002) BindingDB Entry DOI: 10.7270/Q2NK3FRR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vesicular glutamate transporter 3 (Rattus norvegicus) | BDBM50113318 (6-Styryl-quinoline-2,4-dicarboxylic acid | CHEMBL7...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.29E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Montana Curated by ChEMBL | Assay Description Inhibitory conc. against Vesicular glutamate transporter (VGLUT), derived from Lineweaver-Burke analysis | J Med Chem 45: 2260-76 (2002) BindingDB Entry DOI: 10.7270/Q2NK3FRR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vesicular glutamate transporter 3 (Rattus norvegicus) | BDBM50113321 (6-Phenethyl-quinoline-2,4-dicarboxylic acid | CHEM...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.43E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Montana Curated by ChEMBL | Assay Description Estimated inhibitory conc. against Vesicular glutamate transporter (VGLUT), using Cheng-Prushoff equation | J Med Chem 45: 2260-76 (2002) BindingDB Entry DOI: 10.7270/Q2NK3FRR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vesicular glutamate transporter 3 (Rattus norvegicus) | BDBM50113318 (6-Styryl-quinoline-2,4-dicarboxylic acid | CHEMBL7...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.67E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Montana Curated by ChEMBL | Assay Description Estimated inhibitory conc. against Vesicular glutamate transporter (VGLUT), using Cheng-Prushoff equation | J Med Chem 45: 2260-76 (2002) BindingDB Entry DOI: 10.7270/Q2NK3FRR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vesicular glutamate transporter 3 (Rattus norvegicus) | BDBM50113323 (6-Phenethyloxy-quinoline-2,4-dicarboxylic acid | C...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.89E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Montana Curated by ChEMBL | Assay Description Estimated inhibitory conc. against Vesicular glutamate transporter (VGLUT), using Cheng-Prushoff equation | J Med Chem 45: 2260-76 (2002) BindingDB Entry DOI: 10.7270/Q2NK3FRR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vesicular glutamate transporter 3 (Rattus norvegicus) | BDBM50113313 (4,8-Dihydroxy-quinoline-2-carboxylic acid anion | ...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid PDB UniChem Patents Similars | PubMed | 1.90E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Montana Curated by ChEMBL | Assay Description Evaluated for competitive inhibition against Vesicular glutamate transporter (VGLUT), and Ki value was reported. | J Med Chem 45: 2260-76 (2002) BindingDB Entry DOI: 10.7270/Q2NK3FRR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vesicular glutamate transporter 3 (Rattus norvegicus) | BDBM50081123 (6-Benzyloxy-quinoline-2,4-dicarboxylic acid | CHEM...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | PubMed | 2.04E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Montana Curated by ChEMBL | Assay Description Inhibitory conc. against Vesicular glutamate transporter (VGLUT), derived from Lineweaver-Burke analysis | J Med Chem 45: 2260-76 (2002) BindingDB Entry DOI: 10.7270/Q2NK3FRR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vesicular glutamate transporter 3 (Rattus norvegicus) | BDBM50113319 (8-Hydroxy-quinoline-2,4-dicarboxylic acid | CHEMBL...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 2.86E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Montana Curated by ChEMBL | Assay Description Estimated inhibitory conc. against Vesicular glutamate transporter (VGLUT), using Cheng-Prushoff equation | J Med Chem 45: 2260-76 (2002) BindingDB Entry DOI: 10.7270/Q2NK3FRR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vesicular glutamate transporter 3 (Rattus norvegicus) | BDBM50113322 (6-Phenylazo-quinoline-2,4-dicarboxylic acid | CHEM...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 2.88E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Montana Curated by ChEMBL | Assay Description Compound was evaluated for competitive inhibition against Vesicular glutamate transporter (VGLUT), and Ki value was reported,.using Cheng-Prushoff eq... | J Med Chem 45: 2260-76 (2002) BindingDB Entry DOI: 10.7270/Q2NK3FRR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vesicular glutamate transporter 3 (Rattus norvegicus) | BDBM50081123 (6-Benzyloxy-quinoline-2,4-dicarboxylic acid | CHEM...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | PubMed | 3.68E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Montana Curated by ChEMBL | Assay Description Estimated inhibitory conc. against Vesicular glutamate transporter (VGLUT), using Cheng-Prushoff equation | J Med Chem 45: 2260-76 (2002) BindingDB Entry DOI: 10.7270/Q2NK3FRR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vesicular glutamate transporter 3 (Rattus norvegicus) | BDBM50005001 (7-Chloro-4-hydroxy-quinoline-2-carboxylic acid | 7...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | 5.90E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Montana Curated by ChEMBL | Assay Description Evaluated for competitive inhibition against Vesicular glutamate transporter (VGLUT), and Ki value was reported. | J Med Chem 45: 2260-76 (2002) BindingDB Entry DOI: 10.7270/Q2NK3FRR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vesicular glutamate transporter 3 (Rattus norvegicus) | BDBM50060136 ((1R,3S)-1-Amino-cyclopentane-1,3-dicarboxylic acid...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | 7.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Montana Curated by ChEMBL | Assay Description Evaluated for competitive inhibition against Vesicular glutamate transporter (VGLUT), and Ki value was reported. | J Med Chem 45: 2260-76 (2002) BindingDB Entry DOI: 10.7270/Q2NK3FRR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vesicular glutamate transporter 3 (Rattus norvegicus) | BDBM81975 (4-hydroxyquinoline-2-carboxylic acid | CAS_492-27-...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid PDB UniChem Patents Similars | PubMed | 1.30E+6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Montana Curated by ChEMBL | Assay Description Compound was evaluated for the inhibition of Vesicular glutamate transporter (VGLUT) | J Med Chem 45: 2260-76 (2002) BindingDB Entry DOI: 10.7270/Q2NK3FRR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Vesicular glutamate transporter 3 (Rattus norvegicus) | BDBM50113315 (5-Bromo-7-methyl-4,6,6a,7,8,9-hexahydro-indolo[4,3...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Montana Curated by ChEMBL | Assay Description Compound was evaluated for competitive inhibition against Vesicular glutamate transporter (VGLUT), and Ki value was reported. | J Med Chem 45: 2260-76 (2002) BindingDB Entry DOI: 10.7270/Q2NK3FRR | |||||||||||
More data for this Ligand-Target Pair |