Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
BH3-interacting domain death agonist [79-99] (Homo sapiens (Human)) | BDBM472688 ((R)-N-((4-(((1,4-dioxan-2-yl)methyl)amino)-3- nitr...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | >5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Bcl-2 and Bcl-xL Inhibition: Fluorescein labeled BIM (81-106), BAK (72-87), and BID (79-99) peptides, named as Flu-BIM, Flu-BAK, and Flu-BID, respect... | US Patent US10829488 (2020) BindingDB Entry DOI: 10.7270/Q28D00BQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
BH3-interacting domain death agonist [79-99] (Homo sapiens (Human)) | BDBM361577 ((S)-N-((4-(((1,4-dioxan-2-yl)methyl)amino)-3- nitr...) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | US Patent | n/a | n/a | >5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Bcl-2 and Bcl-xL Inhibition: Fluorescein labeled BIM (81-106), BAK (72-87), and BID (79-99) peptides, named as Flu-BIM, Flu-BAK, and Flu-BID, respect... | US Patent US10829488 (2020) BindingDB Entry DOI: 10.7270/Q28D00BQ | |||||||||||
More data for this Ligand-Target Pair |